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Sheep tail fat inhibits the proliferation of non-small-cell lung cancer cells in vitro and in vivo 期刊论文
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13
作者:  Xu, Changzhi;  Zhang, Lanlan;  He, Huimin;  Liu, Xiaoyi;  Pei, Xinxin
收藏  |  浏览/下载:22/0  |  提交时间:2022/12/23
The Novel RET Inhibitor SYHA1815 Inhibits RET-Driven Cancers and Overcomes Gatekeeper Mutations by Inducing G1 Cell-Cycle Arrest through c-Myc Downregulation 期刊论文
MOLECULAR CANCER THERAPEUTICS, 2021, 卷号: 20, 期号: 11, 页码: 2198-2206
作者:  Jiang, Yuchen;  Peng, Xia;  Ji, Yinchun;  Dai, Yang;  Fang, Yanfen
收藏  |  浏览/下载:28/0  |  提交时间:2021/12/16
Discovery and Development of a Potent, Selective, and Orally Bioavailable CHK1 Inhibitor Candidate: 5-((4-((3-Amino-3-methylbutyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino)picolinonitrile 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 20, 页码: 15069-15090
作者:  Jin, Tingting;  Xu, Lei;  Wang, Peipei;  Hu, Xiaobei;  Zhang, Runyuan
收藏  |  浏览/下载:20/0  |  提交时间:2022/01/04
Design, synthesis and pharmacological evaluation of bicyclic and tetracyclic pyridopyrimidinone analogues as new KRAS(G12C) inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 213, 页码: 17
作者:  Xiao, Xuanzheng;  Lai, Mengzhen;  Song, Zilan;  Geng, Meiyu;  Ding, Jian
收藏  |  浏览/下载:47/0  |  提交时间:2021/05/24
Divalent tranylcypromine derivative as lysine-specific demethylase 1 inhibitor 期刊论文
MEDICINAL CHEMISTRY RESEARCH, 2021, 页码: 8
作者:  Sun, Yin;  Li, Na;  Su, Mingbo;  Wang, Xiaowen;  Zhao, Dongmei
收藏  |  浏览/下载:58/0  |  提交时间:2021/05/24
DW14383 is an irreversible pan-FGFR inhibitor that suppresses FGFR-dependent tumor growth in vitro and in vivo 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9
作者:  Dai, Meng-di;  Wang, Yue-liang;  Fan, Jun;  Dai, Yang;  Ji, Yin-chun
收藏  |  浏览/下载:32/0  |  提交时间:2021/05/24
The dual HDAC-PI3K inhibitor CUDC-907 displays single-agent activity and synergizes with PARP inhibitor olaparib in small cell lung cancer 期刊论文
JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH, 2020, 卷号: 39
作者:  Ma, Liying;  Bian, Xing;  Lin, Wenchu
收藏  |  浏览/下载:37/0  |  提交时间:2020/11/30
Bungsteroid A: One Unusual C 34 Pentacyclic Steroid Analogue from Zanthoxylum bungeanum Maxim 期刊论文
the Journal of Organic Chemistry, 2020, 卷号: 85, 期号: 16, 页码: 10806−10812
作者:  Meng XH(孟宪华);  Chai T(柴甜);  Shi YP(师彦平);  Yang JL(杨军丽)
收藏  |  浏览/下载:15/0  |  提交时间:2020/11/16
Studies on Proximate Composition and Phytochemical Profiling of Turbinaria ornata and its Antiproliferative Effect on Y79 Cell Lines 期刊论文
THALASSAS, 2019, 卷号: 35, 期号: 2, 页码: 495-502
作者:  Remya, R. R.;  Rajasree, S. R. Radhika;  Suman, T. Y.;  Aranganathan, L.;  Gayathri, S.
收藏  |  浏览/下载:58/0  |  提交时间:2019/12/03
Design of wogonin-inspired selective cyclin-dependent kinase 9 (CDK9) inhibitors with potent in vitro and in vivo antitumor activity 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 178, 页码: 782-801
作者:  Wang, Jubo;  Li, Tinghan;  Zhao, Tengteng;  Wu, Tizhi;  Liu, Chuang
收藏  |  浏览/下载:21/0  |  提交时间:2020/07/01


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