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Discovery and optimization of a series of 3-substituted indazole derivatives as multi-target kinase inhibitors for the treatment of lung squamous cell carcinoma 期刊论文
European journal of medicinal chemistry, 2018, 卷号: 163, 页码: 671-689
作者:  Wang, Qi;  Dai, Yang;  Ji, Yinchun;  Shi, Huanyu;  Guo, Zuhao
收藏  |  浏览/下载:85/0  |  提交时间:2019/01/08
High-throughput screening campaigns against a PI3K alpha isoform bearing the H1047R mutation identified potential inhibitors with novel scaffolds 期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 11, 页码: 1816-1822
作者:  Wang, Jia;  Gong, Grace Qun;  Zhou, Yan;  Lee, Woo-Jeong;  Buchanan, Christina Maree
收藏  |  浏览/下载:84/0  |  提交时间:2019/01/08
Molecular-docking-guided design and synthesis of new IAA-tacrine hybrids as multifunctional AChE/BChE inhibitors 期刊论文
Bioorganic chemistry, 2018, 卷号: 83, 页码: 277-288
作者:  Cheng, Zhi-Qiang;  Zhu, Kong-Kai;  Zhang, Juan;  Song, Jia-Li;  Muehlmann, Luis Alexandre
收藏  |  浏览/下载:48/0  |  提交时间:2019/01/08
Novel nor-monoterpenoid indole alkaloids inhibiting glioma stem cells from fruits of Alstonia scholaris 期刊论文
PHYTOMEDICINE, 2018, 卷号: 48, 页码: 170-178
作者:  Wang, Bei;  Dai, Zhi;  Yang, Xiong-Wu;  Liu, Ya-Ping;  Khan, Afsar
收藏  |  浏览/下载:33/0  |  提交时间:2018/10/04
Enhancement of Glucose Utilization by Loesenerine through AMPK Activation in Myotubes 期刊论文
CHEMICAL & PHARMACEUTICAL BULLETIN, 2018, 卷号: 66, 期号: 9, 页码: 885-886
作者:  Wang, Luo-Na;  Jiang, Hao-Wen;  Li, Jin-Long;  Li, Jing-Ya
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
Ligand-based pharmacophore model for the discovery of novel CXCR2 antagonists as anti-cancer metastatic agents 期刊论文
ROYAL SOCIETY OPEN SCIENCE, 2018, 卷号: 5, 期号: 7
作者:  Che, Jinxin;  Wang, Zhilong;  Sheng, Haichao;  Huang, Feng;  Dong, Xiaowu
收藏  |  浏览/下载:41/0  |  提交时间:2019/01/08
OsSND2, a NAC family transcription factor, is involved in secondary cell wall biosynthesis through regulating MYBs expression in rice 期刊论文
RICE, 2018, 卷号: 11, 期号: 无, 页码: 14
作者:  Ye, Yafeng;  Wu, Kun;  Chen, Jianfeng;  Liu, Qian;  Wu, Yuejin
收藏  |  浏览/下载:63/0  |  提交时间:2019/08/23
Identification of a novel selective small-molecule inhibitor of protein arginine methyltransferase 5 (PRMT5) by virtual screening, resynthesis and biological evaluations 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 9, 页码: 1476-1483
作者:  Zhu, Kongkai;  Jiang, Chengshi;  Tao, Hongrui;  Liu, Jingqiu;  Zhang, Hua
收藏  |  浏览/下载:59/0  |  提交时间:2019/01/08
Discovery of potent DOT1L inhibitors by AlphaLISA based High Throughput Screening assay 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1751-1758
作者:  Song, Yakai;  Li, Linjuan;  Chen, Yantao;  Liu, Jingqiu;  Xiao, Senhao
收藏  |  浏览/下载:42/0  |  提交时间:2019/01/08
Screening of neuraminidase inhibitory activities of some medicinal plants traditionally used in Lingnan Chinese medicines 期刊论文
BMC COMPLEMENTARY AND ALTERNATIVE MEDICINE, 2018, 卷号: 18
作者:  Liu, Jiawei;  Zu, Mian;  Chen, Kaotan;  Gao, Li;  Min, Huan
收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08


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