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Design, synthesis and antiproliferative activity evaluation of a series of pyrrolo [2,1-f] [1,2,4] triazine derivatives 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 12, 页码: 4
作者:  Xiang, Hao-Yue;  Chen, Yan-Hong;  Wang, Yi;  Zhang, Xi;  Ding, Jian
收藏  |  浏览/下载:37/0  |  提交时间:2020/07/01
Inhibiting PI3 kinase-γ in both myeloid and plasma cells remodels the suppressive tumor microenvironment in desmoplastic tumors 期刊论文
Journal of Controlled Release, 2019, 卷号: 309
作者:  Zhang, Xueqiong;  Shen, Limei;  Liu, Qi;  Hou, Lin;  Huang, Leaf
收藏  |  浏览/下载:13/0  |  提交时间:2019/12/05
Spautin-A41 Attenuates Cerulein-Induced Acute Pancreatitis through Inhibition of Dysregulated Autophagy 期刊论文
BIOLOGICAL & PHARMACEUTICAL BULLETIN, 2019, 卷号: 42, 期号: 11, 页码: 1789-1798
作者:  Dong, Kai;  Chen, Xia;  Xie, Liping;  Yu, Lanting;  Shen, Mengjun
收藏  |  浏览/下载:30/0  |  提交时间:2019/12/11
CKLF1 aggravates neointimal hyperplasia by inhibiting apoptosis of vascular smooth muscle cells through PI3K/AKT/NF-kappa B signaling 期刊论文
2019, 卷号: 117, 页码: 108986
作者:  Duan, Yanyu;  Zhang, Yongbao;  Qu, Chengjia;  Yu, Weidong;  Tana
收藏  |  浏览/下载:14/0  |  提交时间:2020/01/03
High-throughput screening campaigns against a PI3K alpha isoform bearing the H1047R mutation identified potential inhibitors with novel scaffolds 期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 11, 页码: 1816-1822
作者:  Wang, Jia;  Gong, Grace Qun;  Zhou, Yan;  Lee, Woo-Jeong;  Buchanan, Christina Maree
收藏  |  浏览/下载:84/0  |  提交时间:2019/01/08
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3K delta) inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 页码: 831-846
作者:  Liang, Xiaofei;  Li, Feng;  Chen, Cheng;  Jiang, Zongru;  Wang, Aoli
收藏  |  浏览/下载:11/0  |  提交时间:2019/12/10
High-throughput screening campaigns against a PI3K alpha isoform bearing the H1047R mutation identified potential inhibitors with novel scaffolds 期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 11
作者:  Wang, Jia;  Gong, Grace Qun;  Zhou, Yan;  Lee, Woo-Jeong;  Buchanan, Christina Maree
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/05
Anti-diabetic effect of three new norditerpenoid alkaloids in vitro and potential mechanism via PI3K/Akt signaling pathway 期刊论文
BIOMEDICINE & PHARMACOTHERAPY, 2017, 卷号: 87, 期号: 3, 页码: 145-152
作者:  Tang, D (Tang, Dan);  Chen, QB (Chen, Qi-Bin);  Xin, XL (Xin, Xue-Lei);  Aisa, HA (Aisa, Haji-Akber)
收藏  |  浏览/下载:16/0  |  提交时间:2017/04/05
Discovery of new BTK inhibitors with B cell suppression activity bearing a 4,6-substituted thieno[3,2-d] pyrimidine scaffold 期刊论文
RSC ADVANCES, 2017, 卷号: 7, 期号: 42, 页码: 26060-26069
作者:  Zhang, Qiumeng;  Zhang, Luyao;  Yu, Jie;  Li, Heng;  He, Shijun
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08
Graphene Enhances Cellular Proliferation through Activating the Epidermal Growth Factor Receptor 期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2016, 卷号: 64, 期号: 29, 页码: 5909-5918
作者:  Liu, Wei;  Sun, Cheng;  Liao, Chunyang;  Cui, Lin;  Li, Haishan
收藏  |  浏览/下载:54/0  |  提交时间:2017/03/27


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