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Targeting KRAS mutant cancers: from druggable therapy to drug resistance 期刊论文
MOLECULAR CANCER, 2022, 卷号: 21
作者:  Zhu, Chunxiao;  Guan, Xiaoqing;  Zhang, Xinuo;  Luan, Xin;  Song, Zhengbo
收藏  |  浏览/下载:22/0  |  提交时间:2022/12/23
A Peptide Binder of E3 Ligase Adaptor SPOP Disrupts Oncogenic SPOP-Protein Interactions in Kidney Cancer Cells 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2020, 页码: 274-280
作者:  Wang, Zhen;  Zhang, Hao;  Chen, Baoen;  Ouyang, Sisheng;  Zheng, Tong
收藏  |  浏览/下载:124/0  |  提交时间:2021/05/24
Discovery of an Inhibitor for the TREK-1 Channel Targeting an Intermediate Transition State of Channel Gating 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 19, 页码: 10972-10983
作者:  Ma, Yuqin;  Luo, Qichao;  Fu, Jie;  Che, Yanxin;  Guo, Fei
收藏  |  浏览/下载:11/0  |  提交时间:2021/05/24
Synthesis and biological investigation of triazolopyridinone derivatives as potential multireceptor atypical antipsychotics 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 8, 页码: 6
作者:  Shi, Wenqiang;  Wang, Yu;  Wu, Chunhui;  Yang, Feipu;  Zheng, Wei
收藏  |  浏览/下载:26/0  |  提交时间:2020/07/01
Selective activation of TWIK-related acid-sensitive K+ 3 subunit-containing channels is analgesic in rodent models 期刊论文
SCIENCE TRANSLATIONAL MEDICINE, 2019, 卷号: 11, 期号: 519, 页码: 12
作者:  Liao, Ping;  Qiu, Yunguang;  Mo, Yiqing;  Fu, Jie;  Song, Zhenpeng
收藏  |  浏览/下载:30/0  |  提交时间:2020/07/01
Small-Molecule Targeting of Oncogenic FTO Demethylase in Acute Myeloid Leukemia 期刊论文
CANCER CELL, 2019, 卷号: 35, 期号: 4, 页码: 677-+
作者:  Huang, Yue;  Su, Rui;  Sheng, Yue;  Dong, Lei;  Dong, Ze
收藏  |  浏览/下载:25/0  |  提交时间:2020/07/01
Bromodomain-Containing Protein 4: A Druggable Target. 期刊论文
Current drug targets, 2019
作者:  Shi Yingying;  Liu Jingwen;  Zhao Yuanyuan;  Cao Jiaoxian;  Li Yiming
收藏  |  浏览/下载:21/0  |  提交时间:2019/12/05
Allostery in Drug Development 期刊论文
PROTEIN ALLOSTERY IN DRUG DISCOVERY, 2019, 卷号: 1163, 页码: 1-23
作者:  Cheng, Xi;  Jiang, Hualiang
收藏  |  浏览/下载:14/0  |  提交时间:2020/07/01
Current Strategies and Applications for Precision Drug Design 期刊论文
FRONTIERS IN PHARMACOLOGY, 2018, 卷号: 9
作者:  Wang, Chen;  Xu, Pan;  Zhang, Luyu;  Huang, Jing;  Zhu, Kongkai
收藏  |  浏览/下载:47/0  |  提交时间:2019/01/08
Quinone skeleton as a new class of irreversible inhibitors against Staphylococcus aureus sortase A 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 10, 页码: 1864-1869
作者:  Hou, Xiaochen;  Wang, Meining;  Wen, Yi;  Ni, Tengfeng;  Guan, Xiangna
收藏  |  浏览/下载:33/0  |  提交时间:2019/01/08


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