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Enzalutamide-induced and PTH1R-mediated TGFBR2 degradation in osteoblasts confers resistance in prostate cancer bone metastases 期刊论文
CANCER LETTERS, 2022, 卷号: 525, 页码: 170-178
作者:  Su, Shang;  Cao, Jingchen;  Meng, Xiangqi;  Liu, Ruihua;  Vander Ark, Alexandra
收藏  |  浏览/下载:52/0  |  提交时间:2022/01/04
New Cembrane-Type Diterpenoids from the South China Sea Soft Coral Sinularia nanolobata 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2022, 卷号: 40, 期号: 1, 页码: 28-38
作者:  Lin, Na;  Li, Heng;  Wang, Jian-Rong;  Tang, Wei;  Zheng, Ming-Yue
收藏  |  浏览/下载:26/0  |  提交时间:2022/01/04
LS-106, a novel EGFR inhibitor targeting C797S, exhibits antitumor activities both in vitro and in vivo 期刊论文
CANCER SCIENCE, 2021, 页码: 12
作者:  Liu, Yingqiang;  Lai, Mengzhen;  Li, Shan;  Wang, Yanan;  Feng, Fang
收藏  |  浏览/下载:62/0  |  提交时间:2022/01/18
Discrete genetic loci in human gutBacteroides thetaiotaomicron confer pectin metabolism 期刊论文
CARBOHYDRATE POLYMERS, 2021, 卷号: 272, 页码: 13
作者:  Li, Meixia;  Li, Saijuan;  Guo, Xiaozhen;  Guo, Ciliang;  Wang, Yeqin
收藏  |  浏览/下载:62/0  |  提交时间:2021/11/04
Discovery and Development of a Potent, Selective, and Orally Bioavailable CHK1 Inhibitor Candidate: 5-((4-((3-Amino-3-methylbutyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino)picolinonitrile 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 20, 页码: 15069-15090
作者:  Jin, Tingting;  Xu, Lei;  Wang, Peipei;  Hu, Xiaobei;  Zhang, Runyuan
收藏  |  浏览/下载:23/0  |  提交时间:2022/01/04
Discovery of a subtype-selective, covalent inhibitor against palmitoylation pocket of TEAD3 期刊论文
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 10, 页码: 3206-3219
作者:  Lu, Tian;  Li, Yong;  Lu, Wenchao;  Spitters, Twgm;  Fang, Xueyu
收藏  |  浏览/下载:41/0  |  提交时间:2021/12/01
Discovery of a Potential Liver Fibrosis Inhibitor from a Mushroom Endophytic Fungus by Genome Mining of a Silent Biosynthetic Gene Cluster 期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2021, 卷号: 69, 期号: 38, 页码: 11303-11310
作者:  Cheng, Jin-Tao;  Wang, Han-Min;  Yu, Jia-Hui;  Sun, Chen-Fan;  Cao, Fei
收藏  |  浏览/下载:28/0  |  提交时间:2021/12/01
Structural characterization of two novel polysaccharides from Gastrodia elata and their effects on Akkermansia muciniphila 期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2021, 卷号: 186, 页码: 501-509
作者:  Huo, Jiangyan;  Lei, Min;  Zhou, Yang;  Zhong, Xianchun;  Liu, Yameng
收藏  |  浏览/下载:66/0  |  提交时间:2021/11/04
Discovery of Cyclic Peptidomimetic Ligands Targeting the Extracellular Domain of EGFR 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 15, 页码: 11219-11228
作者:  Zheng, Mengmeng;  Li, Chunpu;  Zhou, Mi;  Jia, Ru;  Cai, Gang
收藏  |  浏览/下载:65/0  |  提交时间:2021/11/04
Discovery of pyrrolo[2,3-d]pyrimidine derivatives as potent Axl inhibitors: Design, synthesis and biological evaluation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 220, 页码: 18
作者:  Xu, Dandan;  Sun, Deqiao;  Wang, Wei;  Peng, Xia;  Zhan, Zhengsheng
收藏  |  浏览/下载:46/0  |  提交时间:2021/08/17


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