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Discovery of pyrrolo[2,3-d]pyrimidine derivatives as potent Axl inhibitors: Design, synthesis and biological evaluation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 220, 页码: 18
作者:  Xu, Dandan;  Sun, Deqiao;  Wang, Wei;  Peng, Xia;  Zhan, Zhengsheng
收藏  |  浏览/下载:45/0  |  提交时间:2021/08/17
Synthesis of triazolotriazine derivatives as c-Met inhibitors 期刊论文
MOLECULAR DIVERSITY, 2020, 页码: 8
作者:  Guo, Yuting;  Peng, Xia;  Ji, Yinchun;  Zhang, Yitong;  Ding, Jian
收藏  |  浏览/下载:37/0  |  提交时间:2020/12/24
Evaluation of Deuterium-Labeled JNJ38877605: Pharmacokinetic, Metabolic, and in Vivo Antitumor Profiles 期刊论文
CHEMICAL RESEARCH IN TOXICOLOGY, 2018, 卷号: 31, 期号: 11, 页码: 1213-1218
作者:  Zhan, Zhengsheng;  Peng, Xia;  Sun, Yiming;  Ai, Jing;  Duan, Wenhu
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
Discovery of 6-(difluoro(6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b] [1,2,4]triazin-3-yl)methyl)quinoline as a highly potent and selective c-Met inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 239-251
作者:  Zhan, Zhengsheng;  Peng, Xia;  Liu, Qiufeng;  Chen, Fang;  Ji, Yinchun
收藏  |  浏览/下载:48/0  |  提交时间:2019/01/08
Simm530, a novel and highly selective c-Met inhibitor, blocks c-Met-stimulated signaling and neoplastic activities 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 25, 页码: 38091-38104
作者:  Wang, Ying;  Zhan, Zhengsheng;  Jiang, Xifei;  Peng, Xia;  Shen, Yanyan
收藏  |  浏览/下载:51/0  |  提交时间:2019/01/08
Simm530, a novel and highly selective c-Met inhibitor, blocks c-Met-stimulated signaling and neoplastic activities 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 25
作者:  Wang, Ying;  Zhan, Zhengsheng;  Jiang, Xifei;  Peng, Xia;  Shen, Yanyan
收藏  |  浏览/下载:13/0  |  提交时间:2019/12/06
Discovery of Anilinopyrimidines as Dual Inhibitors of c-Met and VEGFR-2: Synthesis, SAR, and Cellular Activity 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 5, 期号: 6, 页码: 673-678
作者:  Zhan, Zhengsheng;  Ai, Jing;  Liu, Qiufeng;  Ji, Yinchun;  Chen, Tiantian
收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08
A novel, potent, highly selective inhibitor of c-Met kinase, Simm559, inhibits c-Met-dependent neoplastic phenotypes in vitro and in vivo. 会议论文
作者:  Ai, Jing;  Zhan, ZhengSheng;  Wang, Ying;  Chen, Fang;  Peng, Xia
收藏  |  浏览/下载:45/0  |  提交时间:2019/01/08
O-Linked Triazolotriazines: Potent and Selective c-Met Inhibitors 期刊论文
CHEMMEDCHEM, 2012, 卷号: 7, 期号: 7, 页码: 1276-1285
作者:  Chen, Fang;  Wang, Ying;  Ai, Jing;  Zhan, Zhengsheng;  Lv, Yongcong
收藏  |  浏览/下载:8/0  |  提交时间:2019/01/08


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