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GPR84 signaling promotes intestinal mucosal inflammation via enhancing NLRP3 inflammasome activation in macrophages 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:  Zhang, Qing;  Chen, Lin-hai;  Yang, Hui;  Fang, You-chen;  Wang, Si-wei
收藏  |  浏览/下载:44/0  |  提交时间:2022/01/18
Pharmacodynamic, pharmacokinetic, and phase 1a study of bisthianostat, a novel histone deacetylase inhibitor, for the treatment of relapsed or refractory multiple myeloma 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:  Zhou, Yu-bo;  Zhang, Yang-ming;  Huang, Hong-hui;  Shen, Li-jing;  Han, Xiao-feng
收藏  |  浏览/下载:90/0  |  提交时间:2021/11/04
Synthesis and Structure-Activity Relationships of Ring-Opened Bengamide Analogues against Methicillin-Resistant Staphylococcus aureus(dagger) 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2021, 卷号: 39, 期号: 3, 页码: 671-676
作者:  Yu, Chen-Xi;  Wei, Bing-Yan;  Kong, Xue-Qing;  Yang, Cai-Guang;  Nan, Fa-Jun
收藏  |  浏览/下载:41/0  |  提交时间:2021/05/24
Modulation of the G-Protein-Coupled Receptor 84 (GPR84) by Agonists and Antagonists 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 24, 页码: 15399-15409
作者:  Chen, Lin-Hai;  Zhang, Qing;  Xie, Xin;  Nan, Fa-Jun
收藏  |  浏览/下载:15/0  |  提交时间:2021/05/24
Pyrazolone derivative C29 protects against HFD-induced obesity in mice via activation of AMPK in adipose tissue 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:  Li, Bo-han;  Zhang, Mei;  Duan, Ya-nan;  Shuai, Lin;  Jiang, Hao-wen
收藏  |  浏览/下载:50/0  |  提交时间:2020/12/21
AMPK activator C24 inhibits hepatic lipogenesis and ameliorates dyslipidemia in HFHC diet-induced animal models 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 8
作者:  Sun, Shui-mei;  Xie, Zhi-fu;  Zhang, Yang-ming;  Zhang, Xin-wen;  Zhou, Chen-dong
收藏  |  浏览/下载:24/0  |  提交时间:2020/12/24
Design, Synthesis and Biological Evaluation of Bengamide Analogues as ClpP Activators 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2020, 页码: 5
作者:  Kong, Xue-Qing;  Wei, Bing-Yan;  Yu, Chen-Xi;  Guan, Xiang-Na;  Ma, Wei-Ping
收藏  |  浏览/下载:12/0  |  提交时间:2020/12/24
Discovery of aryl sulfonamide-selective Nav1.7 inhibitors with a highly hydrophobic ethanoanthracene core 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 3, 页码: 293-302
作者:  Wang, Jin-tao;  Zheng, Yue-ming;  Chen, Yue-ting;  Gu, Min;  Gao, Zhao-bing
收藏  |  浏览/下载:44/0  |  提交时间:2020/07/01
Synthesis and in Vitro and in Vivo Biological Evaluation of Tissue-Specific Bisthiazole Histone Deacetylase (HDAC) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 2, 页码: 804-815
作者:  Zhang, Shu-Wei;  Gong, Chao-Jun;  Su, Ming-Bo;  Chen, Fei;  He, Ting
收藏  |  浏览/下载:10/0  |  提交时间:2020/07/01
Berberine derivatives with a long alkyl chain branched by hydroxyl group and methoxycarbonyl group at 9-position show improved anti-proliferation activity and membrane permeability in A549 cells 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 12
作者:  Liu, Yi;  Zhu, Ke-xin;  Cao, Lei;  Xie, Zhi-fu;  Gu, Min
收藏  |  浏览/下载:15/0  |  提交时间:2020/07/01


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