×
验证码:
换一张
忘记密码?
记住我
CORC
首页
科研机构
检索
知识图谱
申请加入
托管服务
登录
注册
在结果中检索
科研机构
上海药物研究所 [8]
复旦大学上海医学院 [7]
上海生物化学与细胞生... [6]
四川大学 [5]
安徽大学 [3]
山东大学 [2]
更多...
内容类型
期刊论文 [46]
会议论文 [1]
发表日期
2018 [47]
学科主题
Biochemist... [1]
Cell Biolo... [1]
Plant Scie... [1]
×
知识图谱
CORC
开始提交
已提交作品
待认领作品
已认领作品
未提交全文
收藏管理
QQ客服
官方微博
反馈留言
浏览/检索结果:
共47条,第1-10条
帮助
限定条件
发表日期:2018
已选(
0
)
清除
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
发表日期升序
发表日期降序
提交时间升序
提交时间降序
题名升序
题名降序
作者升序
作者降序
Identification of 5-benzylidene-2-phenylthiazolones as potent PRMT5 inhibitors by virtual screening, structural optimization and biological evaluations
期刊论文
BIOORGANIC CHEMISTRY, 2018, 卷号: 81, 页码: 289-298
作者:
Zhu, Kongkai
;
Tao, Hongrui
;
Song, Jia-Li
;
Jin, Lu
;
Zhang, Yuanyuan
收藏
  |  
浏览/下载:129/0
  |  
提交时间:2019/01/08
PRMT5 inhibitor
Arginine methylation
Virtual screening
Molecular docking
Molecular dynamics simulation
Design, synthesis and anti leukemia cells proliferation activities of pyrimidylaminoquinoline derivatives as DOT1L inhibitors
期刊论文
BIOORGANIC CHEMISTRY, 2018, 卷号: 80, 页码: 649-654
作者:
Zhang, Li
;
Chen, Yantao
;
Liu, Na
;
Li, Linjuan
;
Xiao, Senhao
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2019/01/08
Pyrimidylaminoquinoline
Nonnucleoside DOT1L inhibitors
Amino side chains
Mixed-linage leukemia
Histone lysine methyltransferase
Small molecules capable of activating DNA methylation-repressed genes targeted by the p38 mitogen-activated protein kinase pathway
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2018, 卷号: 293, 期号: 19, 页码: 7423-7436
作者:
Shao, Wei
;
Wang, Hailin
;
Zheng, Yong
;
Li, Xiang
;
Zhao, Zuodong
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/06/20
DNA methylation
high-throughput screening (HTS)
p38
mitogen-activated protein kinase (MAPK)
gene regulation
gene activation
Discovery of potent DOT1L inhibitors by AlphaLISA based High Throughput Screening assay
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1751-1758
作者:
Song, Yakai
;
Li, Linjuan
;
Chen, Yantao
;
Liu, Jingqiu
;
Xiao, Senhao
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2019/01/08
DOT1L
MLL-rearranged leukemia
AlphaLISA
HTS
Novel inhibitors
Roles of the CSE1L-mediated nuclear import pathway in epigenetic silencing
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2018, 卷号: 115, 期号: 17, 页码: E4013-E4022
作者:
Liu, Baodong
;
Shao, Wei
;
Yuan, Gang
;
Xu, Shaohua
;
Wang, Cheng-Zhi
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2019/06/20
CSE1L
DNA methylation
gene silencing
nuclear import pathway
Roles of the CSE1L-mediated nuclear import pathway in epigenetic silencing
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2018, 卷号: 115, 期号: 17, 页码: E4013-E4022
作者:
Dong, Qiang
;
Li, Xiang
;
Wang, Cheng-Zhi
;
Xu, Shaohua
;
Yuan, Gang
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2019/04/09
Cse1l
Dna Methylation
Gene Silencing
Nuclear Import Pathway
Identification and Characterizations of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Scaffold Hopping- and 2D-Molecular Fingerprint-Based Similarity Search
期刊论文
MOLECULES, 2018, 卷号: 23, 期号: 3
作者:
Ding, Hong
;
Lu, Wen Chao
;
Hu, Jun Chi
;
Liu, Yu-Chih
;
Zhang, Chen Hua
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2019/01/08
SET7
inhibitor
similarity search
ligand-based drug design
chemical biology probe
Epigenetic actions of environmental factors and promising drugs for cancer therapy (Review)
期刊论文
ONCOLOGY LETTERS, 2018, 卷号: 15, 页码: 2049-2056
作者:
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2018/05/31
epigenetic modification
environmental factor
promising drug
cancer therapy
Effects of adolescent social stress and antidepressant treatment on cognitive inflexibility and Bdnf epigenetic modifications in the mPFC of adult mice
期刊论文
PSYCHONEUROENDOCRINOLOGY, 2018, 卷号: 88, 页码: 92-101
作者:
Xu, Hang
;
Wang, Jiesi
;
Zhang, Ke
;
Zhao, Mei
;
Ellenbroek, Bart
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2018/05/28
Adolescent
Social stress
Cognitive inflexibility
Brain-derived neurotrophic factor (BDNF)
Epigenetic mechanism
©版权所有 ©2017 CSpace - Powered by
CSpace