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Identification of 5-benzylidene-2-phenylthiazolones as potent PRMT5 inhibitors by virtual screening, structural optimization and biological evaluations 期刊论文
BIOORGANIC CHEMISTRY, 2018, 卷号: 81, 页码: 289-298
作者:  Zhu, Kongkai;  Tao, Hongrui;  Song, Jia-Li;  Jin, Lu;  Zhang, Yuanyuan
收藏  |  浏览/下载:129/0  |  提交时间:2019/01/08
Design, synthesis and anti leukemia cells proliferation activities of pyrimidylaminoquinoline derivatives as DOT1L inhibitors 期刊论文
BIOORGANIC CHEMISTRY, 2018, 卷号: 80, 页码: 649-654
作者:  Zhang, Li;  Chen, Yantao;  Liu, Na;  Li, Linjuan;  Xiao, Senhao
收藏  |  浏览/下载:38/0  |  提交时间:2019/01/08
Small molecules capable of activating DNA methylation-repressed genes targeted by the p38 mitogen-activated protein kinase pathway 期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2018, 卷号: 293, 期号: 19, 页码: 7423-7436
作者:  Shao, Wei;  Wang, Hailin;  Zheng, Yong;  Li, Xiang;  Zhao, Zuodong
收藏  |  浏览/下载:26/0  |  提交时间:2019/06/20
Discovery of potent DOT1L inhibitors by AlphaLISA based High Throughput Screening assay 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1751-1758
作者:  Song, Yakai;  Li, Linjuan;  Chen, Yantao;  Liu, Jingqiu;  Xiao, Senhao
收藏  |  浏览/下载:42/0  |  提交时间:2019/01/08
Roles of the CSE1L-mediated nuclear import pathway in epigenetic silencing 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2018, 卷号: 115, 期号: 17, 页码: E4013-E4022
作者:  Liu, Baodong;  Shao, Wei;  Yuan, Gang;  Xu, Shaohua;  Wang, Cheng-Zhi
收藏  |  浏览/下载:35/0  |  提交时间:2019/06/20
Roles of the CSE1L-mediated nuclear import pathway in epigenetic silencing 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2018, 卷号: 115, 期号: 17, 页码: E4013-E4022
作者:  Dong, Qiang;  Li, Xiang;  Wang, Cheng-Zhi;  Xu, Shaohua;  Yuan, Gang
收藏  |  浏览/下载:42/0  |  提交时间:2019/04/09
Identification and Characterizations of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Scaffold Hopping- and 2D-Molecular Fingerprint-Based Similarity Search 期刊论文
MOLECULES, 2018, 卷号: 23, 期号: 3
作者:  Ding, Hong;  Lu, Wen Chao;  Hu, Jun Chi;  Liu, Yu-Chih;  Zhang, Chen Hua
收藏  |  浏览/下载:50/0  |  提交时间:2019/01/08
Epigenetic actions of environmental factors and promising drugs for cancer therapy (Review) 期刊论文
ONCOLOGY LETTERS, 2018, 卷号: 15, 页码: 2049-2056
作者:  
收藏  |  浏览/下载:30/0  |  提交时间:2018/05/31
Effects of adolescent social stress and antidepressant treatment on cognitive inflexibility and Bdnf epigenetic modifications in the mPFC of adult mice 期刊论文
PSYCHONEUROENDOCRINOLOGY, 2018, 卷号: 88, 页码: 92-101
作者:  Xu, Hang;  Wang, Jiesi;  Zhang, Ke;  Zhao, Mei;  Ellenbroek, Bart
收藏  |  浏览/下载:42/0  |  提交时间:2018/05/28


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