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北京大学 [4]
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复旦大学上海医学院 [2]
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期刊论文 [12]
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Targeting Protein Neddylation to Inactivate Cullin-RING Ligases by Gossypol: A Lucky Hit or a New Start?
期刊论文
DRUG DESIGN DEVELOPMENT AND THERAPY, 2021, 卷号: 15
作者:
Yu, Qing
;
Sun, Yi
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2021/03/15
anti-cancer drug
cullin-RING E3 ligases
natural product
high-throughput screen
neddylation
small-molecule inhibitors
A first-in-class inhibitor, MLN4924 (pevonedistat), induces cell-cycle arrest, senescence, and apoptosis in human renal cell carcinoma by suppressing UBE2M-dependent neddylation modification
期刊论文
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2018, 卷号: 81, 期号: 6
作者:
Xu, Bo
;
Deng, Yuyou
;
Bi, Ran
;
Guo, Haoran
;
Shu, Chang
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/12/05
MLN4924 (pevonedistat)
Renal cell carcinoma
Neddylation
Cullin-RING E3 ligases
NEDD8
Hiv-1 vpr increases hcv replication through vprbp in cell culture
期刊论文
Virus research, 2016, 卷号: 223, 页码: 153-160
作者:
Yan, Yanling
;
Huang, Fang
;
Yuan, Ting
;
Sun, Binlian
;
Yang, Rongge
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2019/05/09
Hiv-1
Hcv
Vpr
Vprbp
Cullin ring e3 ligases
DWD HYPERSENSITIVE TO UV-B 1 is negatively involved in UV-B mediated cellular responses in Arabidopsis
期刊论文
植物分子生物学, 2014
Kim, Sang-Hoon
;
Kim, Hani
;
Seo, Kyoung-In
;
Kim, Soon-Hee
;
Chung, Sunglan
;
Huang, Xi
;
Yang, Panyu
;
Deng, Xing Wang
;
Lee, Jae-Hoon
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/11/11
CRL4
UV-B
DHU1
Arabidopsis
SYNTHASE GENE-EXPRESSION
E3 UBIQUITIN LIGASES
TRANSCRIPTION FACTOR
SIGNAL-TRANSDUCTION
INDUCED PHOTOMORPHOGENESIS
CIRCADIAN CLOCK
FEEDBACK-REGULATION
STRESS ACCLIMATION
DEFENSE RESPONSES
BINDING PROTEINS
The covalent modifier Nedd8 is critical for the activation of Smurf1 ubiquitin ligase in tumorigenesis
期刊论文
http://dx.doi.org/10.1038/ncomms4733, 2014
Xie, Ping
;
Zhang, Minghua
;
He, Shan
;
Lu, Kefeng
;
Chen, Yuhan
;
Xing, Guichun
;
Lu, Yiming
;
Liu, Ping
;
Li, Yang
;
Wang, Shaoxia
;
Chai, Nan
;
Wu, Jiawei
;
Deng, Haiteng
;
Wang, Hong-Rui
;
Cao, Yu
;
Zhao, Fei
;
Cui, Yu
;
Wang, Jian
;
He, Fuchu
;
Zhang, Lingqiang
;
王洪睿
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2015/07/22
NEDD8-ACTIVATING ENZYME-INHIBITOR
E2 CONJUGATING ENZYMES
E3 LIGASE
HECT DOMAIN
FUNCTIONAL DIVERSITY
CULLIN NEDDYLATION
CELL POLARITY
DEGRADATION
PROTEIN
PATHWAY
Inositol hexakisphosphate kinase-1 mediates assembly/disassembly of the crl4-signalosome complex to regulate DNA repair and cell death
期刊论文
Proceedings of the National Academy of Sciences of the United States of America, 2014, 卷号: 111, 期号: 45
作者:
Rao, Feng/24465697600[0]
;
Xu, Jing/55584800265[1]
;
Khan, A. Basit/55902479300[2]
;
Gadalla, Moataz M./34976532700[3]
;
Cha, Jiyoung/56067617700[4]
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/19
Cullin ring E3 ligases
DNA repair
Inositol phosphates
Signalosome
UV radiation
Ubiquitin E3 ligase CRL4CDT2/DCAF2 as a potential chemotherapeutic target for ovarian surface epithelial cancer
期刊论文
http://dx.doi.org/10.1074/jbc.M113.495069, 2013
Pan, Wei-Wei
;
Zhou, Jian-Jie
;
Yu, Chao
;
Xu, Ying
;
Guo, Lian-Jun
;
Zhang, Hai-Yi
;
Zhou, Dawang
;
Song, Fang-Zhou
;
Fan, Heng-Yu
;
周大旺
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/07/22
Cell death
Chemical activation
Enzymes
Histology
Tumors
Conversion from CUL4-based COP1-SPA E3 apparatus to UVR8-COP1-SPA complexes underlies a distinct biochemical function of COP1 under UV-B
期刊论文
proceedings of the national academy of sciences of the united states of america, 2013
Huang, Xi
;
Ouyang, Xinhao
;
Yang, Panyu
;
Lau, On Sun
;
Chen, Liangbi
;
Wei, Ning
;
Deng, Xing Wang
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/11/10
light signaling
protein complex
posttranscriptional regulation
CONSTITUTIVELY PHOTOMORPHOGENIC1
LIGHT CONTROL
ARABIDOPSIS
PROTEINS
HY5
TRANSCRIPTION
SUPPRESSION
PERCEPTION
INTERACTS
GROWTH
Ubiquitin E3 Ligase CRL4(CDT2/DCAF2) as a Potential Chemotherapeutic Target for Ovarian Surface Epithelial Cancer
期刊论文
http://dx.doi.org/10.1074/jbc.M113.495069, 2013
Pan, Wei-Wei
;
Zhou, Jian-Jie
;
Yu, Chao
;
Xu, Ying
;
Guo, Lian-Jun
;
Zhang, Hai-Yi
;
Zhou, Dawang
;
Song, Fang-Zhou
;
Fan, Heng-Yu
;
周大旺
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2015/07/22
MLN4924 INDUCES AUTOPHAGY
CULLIN-RING LIGASES
NEDD8-ACTIVATING ENZYME
MOUSE EMBRYOGENESIS
INHIBITORY PROTEIN
ANTICANCER TARGETS
CELL-SURVIVAL
GROWTH
DDB1
REPLICATION
Targeting Cullin-RING ligases by MLN4924 induces autophagy via modulating the HIF1-REDD1-TSC1-mTORC1-DEPTOR axis
期刊论文
CELL DEATH & DISEASE, 2012, 卷号: 3
作者:
Zhao, Y.
;
Xiong, X.
;
Jia, L.
;
Sun, Y.
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/19
autophagy
Cullin neddylation
DEPTOR
HIF1 alpha
mTOR
CRL E3 ligases
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