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科研机构
上海药物研究所 [24]
中国科学院大学 [4]
厦门大学 [1]
昆明植物研究所 [1]
上海有机化学研究所 [1]
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期刊论文 [31]
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2018 [1]
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Identification of a novel selective small-molecule inhibitor of protein arginine methyltransferase 5 (PRMT5) by virtual screening, resynthesis and biological evaluations
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 9, 页码: 1476-1483
作者:
Zhu, Kongkai
;
Jiang, Chengshi
;
Tao, Hongrui
;
Liu, Jingqiu
;
Zhang, Hua
收藏
  |  
浏览/下载:59/0
  |  
提交时间:2019/01/08
PRMT5 inhibitor
Resynthesis
Virtual screening
Molecular docking
Molecular dynamics simulation
Application of chemical biology in target identification and drug discovery
期刊论文
ARCHIVES OF PHARMACAL RESEARCH, 2015, 卷号: 38, 期号: 9, 页码: 1642-1650
作者:
Zhu, Yue
;
Xiao, Ting
;
Lei, Saifei
;
Zhou, Fulai
;
Wang, Ming-Wei
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/01/08
Chemical biology
Genomics
Proteomics
Drug discovery
Target validation
High-throughput screening (HTS)
Novel small-molecule AMPK activator orally exerts beneficial effects on diabetic db/db mice
期刊论文
TOXICOLOGY AND APPLIED PHARMACOLOGY, 2013, 卷号: 273, 期号: 2, 页码: 325-334
作者:
Li, Yuan-Yuan
;
Yu, Li-Fang
;
Zhang, Li-Na
;
Qiu, Bei-Ying
;
Su, Ming-Bo
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
AMPK
Activator
Allosteric
Small-molecule
Orally effective
Metabolic syndrome
Novel Small-Molecule AMP-Activated Protein Kinase Allosteric Activator with Beneficial Effects in db/db Mice
期刊论文
PLOS ONE, 2013, 卷号: 8, 期号: 8
作者:
Zhang, Li-Na
;
Xu, Lei
;
Zhou, Hua-Yong
;
Wu, Ling-Yan
;
Li, Yuan-Yuan
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
Discovery of novel PDE10 inhibitors by a robust homogeneous screening assay
期刊论文
ACTA PHARMACOLOGICA SINICA, 2013, 卷号: 34, 期号: 8, 页码: 1116-1120
作者:
Li, Qun-yi
;
Xu, Ming-kai
;
Liu, Gang
;
Christoffersen, Claus Tornby
;
Wang, Ming-wei
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2019/01/08
phosphodiesterase 10 (PDE10)
papaverine
high-throughput screening
psychosis
A universal and multiplex kinase assay using gamma-[O-18(4)]-ATP
期刊论文
http://dx.doi.org/10.1039/c3cc38467e, 2013
Fu, Chuan
;
Zheng, Xueyun
;
Jiang, Yao
;
Liu, Yan
;
Xu, Pengxiang
;
Zeng, Zhiping
;
Liu, Rihe
;
Zhao, Yufen
;
刘艳
;
许鹏翔
;
曾志平
;
赵玉芬
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/07/22
DEPENDENT PROTEIN-KINASE
SCINTILLATION PROXIMITY ASSAY
ELECTROCHEMICAL DETECTION
MASS-SPECTROMETRY
PHOSPHORYLATION
FLUORESCENCE
CELLS
INHIBITORS
SUBSTRATE
PROBES
Emodin, an 11 beta-hydroxysteroid dehydrogenase type 1 inhibitor, regulates adipocyte function in vitro and exerts anti-diabetic effect in ob/ob mice
期刊论文
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 9, 页码: 1195-1203
作者:
Wang, Yue-jing
;
Huang, Su-ling
;
Feng, Ying
;
Ning, Meng-meng
;
Leng, Ying
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
emodin
11 beta-hydroxysteroid dehydrogenase type 1
adipocyte
glucocorticoid
type 2 diabetes
ob/ob mice
emodinan11hydroxysteroiddehydrogenasetype1inhibitorregulatesadipocytefunctioninvitroandexertsantidiabeticeffectinobobmice
期刊论文
actapharmacologicasinica, 2012, 卷号: 33, 期号: 9, 页码: 1195
作者:
Wang Yuejing
;
Huang Suling
;
Feng Ying
;
Ning Mengmeng
;
Leng Ying
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2020/07/01
emodin
11β-hydroxysteroid dehydrogenase type 1
adipocyte
glucocorticoid
type 2 diabetes
ob/ob mice
Emodin, an 11β-hydroxysteroid dehydrogenase type 1 inhibitor, regulates adipocyte function in vitro and exerts anti-diabetic effect in ob/ob mice
期刊论文
Acta Pharmacologica Sinica, 2012, 卷号: 33, 期号: 9, 页码: 1195
作者:
Wang Yuejing
;
Huang Suling
;
Feng Ying
;
Ning Mengmeng
;
Leng Ying
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2020/12/24
emodin
11β-hydroxysteroid dehydrogenase type 1
adipocyte
glucocorticoid
type 2 diabetes
ob/ob mice
Emodin, a natural product, selectively inhibits 11 beta-hydroxysteroid dehydrogenase type 1 and ameliorates metabolic disorder in diet-induced obese mice
期刊论文
BRITISH JOURNAL OF PHARMACOLOGY, 2010, 卷号: 161, 期号: 1, 页码: 113-126
作者:
Feng, Ying
;
Huang, Su-Ling
;
Dou, Wei
;
Zhang, Song
;
Chen, Jun-Hua
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/01/08
emodin
11 beta-hydroxysteroid dehydrogenase type 1
diet-induced obese mice
insulin resistance
metabolic syndrome
type 2 diabetes
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