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Identification of a novel selective small-molecule inhibitor of protein arginine methyltransferase 5 (PRMT5) by virtual screening, resynthesis and biological evaluations 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 9, 页码: 1476-1483
作者:  Zhu, Kongkai;  Jiang, Chengshi;  Tao, Hongrui;  Liu, Jingqiu;  Zhang, Hua
收藏  |  浏览/下载:59/0  |  提交时间:2019/01/08
Application of chemical biology in target identification and drug discovery 期刊论文
ARCHIVES OF PHARMACAL RESEARCH, 2015, 卷号: 38, 期号: 9, 页码: 1642-1650
作者:  Zhu, Yue;  Xiao, Ting;  Lei, Saifei;  Zhou, Fulai;  Wang, Ming-Wei
收藏  |  浏览/下载:10/0  |  提交时间:2019/01/08
Novel small-molecule AMPK activator orally exerts beneficial effects on diabetic db/db mice 期刊论文
TOXICOLOGY AND APPLIED PHARMACOLOGY, 2013, 卷号: 273, 期号: 2, 页码: 325-334
作者:  Li, Yuan-Yuan;  Yu, Li-Fang;  Zhang, Li-Na;  Qiu, Bei-Ying;  Su, Ming-Bo
收藏  |  浏览/下载:12/0  |  提交时间:2019/01/08
Novel Small-Molecule AMP-Activated Protein Kinase Allosteric Activator with Beneficial Effects in db/db Mice 期刊论文
PLOS ONE, 2013, 卷号: 8, 期号: 8
作者:  Zhang, Li-Na;  Xu, Lei;  Zhou, Hua-Yong;  Wu, Ling-Yan;  Li, Yuan-Yuan
收藏  |  浏览/下载:12/0  |  提交时间:2019/01/08
Discovery of novel PDE10 inhibitors by a robust homogeneous screening assay 期刊论文
ACTA PHARMACOLOGICA SINICA, 2013, 卷号: 34, 期号: 8, 页码: 1116-1120
作者:  Li, Qun-yi;  Xu, Ming-kai;  Liu, Gang;  Christoffersen, Claus Tornby;  Wang, Ming-wei
收藏  |  浏览/下载:8/0  |  提交时间:2019/01/08
A universal and multiplex kinase assay using gamma-[O-18(4)]-ATP 期刊论文
http://dx.doi.org/10.1039/c3cc38467e, 2013
Fu, Chuan; Zheng, Xueyun; Jiang, Yao; Liu, Yan; Xu, Pengxiang; Zeng, Zhiping; Liu, Rihe; Zhao, Yufen; 刘艳; 许鹏翔; 曾志平; 赵玉芬
收藏  |  浏览/下载:3/0  |  提交时间:2015/07/22
Emodin, an 11 beta-hydroxysteroid dehydrogenase type 1 inhibitor, regulates adipocyte function in vitro and exerts anti-diabetic effect in ob/ob mice 期刊论文
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 9, 页码: 1195-1203
作者:  Wang, Yue-jing;  Huang, Su-ling;  Feng, Ying;  Ning, Meng-meng;  Leng, Ying
收藏  |  浏览/下载:16/0  |  提交时间:2019/01/08
emodinan11hydroxysteroiddehydrogenasetype1inhibitorregulatesadipocytefunctioninvitroandexertsantidiabeticeffectinobobmice 期刊论文
actapharmacologicasinica, 2012, 卷号: 33, 期号: 9, 页码: 1195
作者:  Wang Yuejing;  Huang Suling;  Feng Ying;  Ning Mengmeng;  Leng Ying
收藏  |  浏览/下载:8/0  |  提交时间:2020/07/01
Emodin, an 11β-hydroxysteroid dehydrogenase type 1 inhibitor, regulates adipocyte function in vitro and exerts anti-diabetic effect in ob/ob mice 期刊论文
Acta Pharmacologica Sinica, 2012, 卷号: 33, 期号: 9, 页码: 1195
作者:  Wang Yuejing;  Huang Suling;  Feng Ying;  Ning Mengmeng;  Leng Ying
收藏  |  浏览/下载:7/0  |  提交时间:2020/12/24
Emodin, a natural product, selectively inhibits 11 beta-hydroxysteroid dehydrogenase type 1 and ameliorates metabolic disorder in diet-induced obese mice 期刊论文
BRITISH JOURNAL OF PHARMACOLOGY, 2010, 卷号: 161, 期号: 1, 页码: 113-126
作者:  Feng, Ying;  Huang, Su-Ling;  Dou, Wei;  Zhang, Song;  Chen, Jun-Hua
收藏  |  浏览/下载:11/0  |  提交时间:2019/01/08


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