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JC-010a, a novel selective SHP2 allosteric inhibitor, overcomes RTK/non-RTK-mediated drug resistance in multiple oncogene-addicted cancers 期刊论文
CANCER LETTERS, 2024, 卷号: 582, 页码: 15
作者:  Lu, Xuxiu;  Yu, Rilei;  Li, Zhen;  Yang, Mengke;  Dai, Jiajia
收藏  |  浏览/下载:2/0  |  提交时间:2024/04/07
Harnessing the targeting potential of differential radiobiological effects of photon versus particle radiation for cancer treatment 期刊论文
JOURNAL OF CELLULAR PHYSIOLOGY, 2020, 页码: 17
作者:  Zhang, Jinhua;  Si, Jing;  Gan, Lu;  Zhou, Rong;  Guo, Menghuan
收藏  |  浏览/下载:24/0  |  提交时间:2022/01/12
Design, Synthesis, and Biological Evaluation of HSP90 Inhibitor-SN38 Conjugates for Targeted Drug Accumulation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 10, 页码: 5421-5441
作者:  Zhu, Shulei;  Shen, Qianqian;  Gao, Yinglei;  Wang, Lei;  Fang, Yanfen
收藏  |  浏览/下载:8/0  |  提交时间:2020/12/24
DCZ5248, a novel dual inhibitor of Hsp90 and autophagy, exerts antitumor activity against colon cancer 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 10
作者:  Chen, Xiang-ling;  Liu, Peng;  Zhu, Wei-liang;  Lou, Li-guang
收藏  |  浏览/下载:49/0  |  提交时间:2020/07/01
Optimized HSP90 mediated fluorescent probes for cancer-specific bioimaging 期刊论文
JOURNAL OF MATERIALS CHEMISTRY B, 2020, 卷号: 8, 期号: 9, 页码: 1878-1896
作者:  Zhu, Shulei;  Li, Yalei;  Huang, Yushu;  Zhang, Minmin;  Gu, Xiaofan
收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01
Time course analysis of immunity-related gene expression in the sea cucumber Apostichopus japonicus during exposure to thermal and hypoxic stress 期刊论文
FISH & SHELLFISH IMMUNOLOGY, 2019, 卷号: 95, 页码: 383-390
作者:  Huo, Da;  Sun, Lina;  Zhang, Libin;  Yang, Hongsheng;  Liu, Shilin
收藏  |  浏览/下载:58/0  |  提交时间:2020/03/20
Design, Synthesis and Pharmacological Evaluation of Novel Hsp90N-terminal Inhibitors Without Induction of Heat Shock Response 期刊论文
CHEMISTRYOPEN, 2019, 卷号: 8, 期号: 3, 页码: 344-353
作者:  Liu, Peng;  Chen, Xiangling;  Zhu, Jianming;  Li, Bo;  Chen, Zhaoqiang
收藏  |  浏览/下载:33/0  |  提交时间:2020/07/01
Recent Advances in the Discovery of Novel HSP90 Inhibitors: An Update from 2014 期刊论文
Current drug targets, 2019
作者:  Xiao Yan;  Liu Yajun
收藏  |  浏览/下载:5/0  |  提交时间:2019/12/02
HSP90 inhibitor DPB induces autophagy and more effectively apoptosis in A549 cells combined with autophagy inhibitors 期刊论文
IN VITRO CELLULAR & DEVELOPMENTAL BIOLOGY-ANIMAL, 2019, 卷号: 55, 期号: 5, 页码: 349-354
作者:  Zhao, YanChun;  Li, Kunlun;  Zhao, BaoXiang;  Su, Le
收藏  |  浏览/下载:14/0  |  提交时间:2019/12/11
Discovery of Small-Molecule Inhibitors of the HSP90-Calcineurin-NFAT Pathway against Glioblastoma 期刊论文
CELL CHEMICAL BIOLOGY, 2019, 卷号: 26, 期号: 3, 页码: 352-3650000000
作者:  Liu, Zhenzhen;  Li, Hongli;  He, Lian;  Xiang, Yu;  Tian, Chengsen
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/11


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