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Twin drug design, synthesis and evaluation of diosgenin derivatives as multitargeted agents for the treatment of vascular dementia 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 37, 页码: 16
作者:  Yang, Gui-Xiang;  Sun, Jia-Min;  Zheng, Lu-Lu;  Zhang, Li;  Li, Jie
收藏  |  浏览/下载:68/0  |  提交时间:2021/06/11
Discovery of new multifunctional selective acetylcholinesterase inhibitors: structure-based virtual screening and biological evaluation 期刊论文
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2019, 卷号: 33, 期号: 5, 页码: 521-530
作者:  Jiang, Cheng-Shi;  Ge, Yong-Xi;  Cheng, Zhi-Qiang;  Song, Jia-Li;  Wang, Yin-Yin
收藏  |  浏览/下载:11/0  |  提交时间:2020/07/01
New 4-N-phenylaminoquinoline derivatives as antioxidant, metal chelating and cholinesterase inhibitors for Alzheimer's disease. 期刊论文
Bioorganic chemistry, 2019, 卷号: Vol.93, 页码: 103328
作者:  Rong Cai;  Li-Ning Wang;  Jing-Jing Fan;  Shang-Qi Geng;  Yu-Ming Liu
收藏  |  浏览/下载:9/0  |  提交时间:2019/11/21
Molecular-docking-guided design and synthesis of new IAA-tacrine hybrids as multifunctional AChE/BChE inhibitors 期刊论文
Bioorganic chemistry, 2018, 卷号: 83, 页码: 277-288
作者:  Cheng, Zhi-Qiang;  Zhu, Kong-Kai;  Zhang, Juan;  Song, Jia-Li;  Muehlmann, Luis Alexandre
收藏  |  浏览/下载:48/0  |  提交时间:2019/01/08
Evaluation of Novel Dual Acetyl- and Butyrylcholinesterase Inhibitors as Potential Anti-Alzheimer's Disease Agents Using Pharmacophore, 3D-QSAR and Molecular Docking Approaches 期刊论文
2017, 卷号: 22, 期号: 8
作者:  Pang, Xiaocong;  Fu, Hui;  Yang, Shilun;  Wang, Lin;  Liu, Ai-Lin
收藏  |  浏览/下载:10/0  |  提交时间:2020/01/04
The discovery of new acetylcholinesterase inhibitors derived from pharmacophore modeling, virtual screening, docking simulation and bioassays 期刊论文
MOLECULAR BIOSYSTEMS, 2016, 卷号: 12, 期号: 12, 页码: 3734-3742
作者:  Zhang, Yunqin;  Zhang, Shuqun;  Xu, Guowei;  Yan, Hui;  Pua, Yinglan
收藏  |  浏览/下载:29/0  |  提交时间:2017/02/14
Design, synthesis and evaluation of novel 7-aminoalkyl-substituted flavonoid derivatives with improved cholinesterase inhibitory activities 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 4, 页码: 672-680
作者:  Luo, Wen[1];  Chen, Ying[2];  Wang, Ting[3];  Hong, Chen[4];  Chang, Li-Ping[5]
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/23
Design, synthesis and evaluation of 4-dimethylamine flavonoid derivatives as potential multifunctional anti-Alzheimer agents 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 122, 页码: 17-26
作者:  Luo Wen[1];  Wang Ting[2];  Hong Chen[3];  Yang Ya-Chen[4];  Chen Ying[5]
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/23
Cholinesterase and Human Lung Cancer Cells (A-549) Inhibitory Activity of the Cassava Peel of Euphorbiaceae in Vitro 会议论文
Joint International Conference on Social Science and Environmental Science (SSES) / International Conference on Food Science and Engineering (ICFSE ), Guangzhou, PEOPLES R CHINA
作者:  Chen, Xiao-Ming;  Zhang, Zhi-Jun;  Liu, Ai-Lin;  Lv, Fei-Jie;  Li, Shu-Fang
收藏  |  浏览/下载:4/0  |  提交时间:2020/01/04
Cholinesterase and Human Lung Cancer Cells (A-549) Inhibitory Activity of the Cassava Peel of Euphorbiaceae in Vitro 会议论文
JOINT 2016 INTERNATIONAL CONFERENCE ON SOCIAL SCIENCE AND ENVIRONMENTAL SCIENCE (SSES 2016) AND INTERNATIONAL CONFERENCE ON FOOD SCIENCE AND ENGINEERING (ICFSE 2016), 2016-01-01
作者:  Chen, Xiao-Ming;  Zhang, Zhi-Jun;  Liu, Ai-Lin;  Lv, Fei-Jie;  Li, Shu-Fang
收藏  |  浏览/下载:7/0  |  提交时间:2020/01/04


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