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科研机构
海洋研究所 [7]
内容类型
期刊论文 [7]
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2021 [1]
2017 [2]
2016 [1]
2013 [2]
2012 [1]
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Pharmacolo... [2]
Chemistry,... [1]
Chemistry,... [1]
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Discovery of 5-(3-bromo-2-(2,3-dibromo-4,5-dimethoxybenzyl)-4,5-dimethoxybenzylidene)thiazolidine-2,4-dione as a novel potent protein tyrosine phosphatase 1B inhibitor with antidiabetic properties
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 108, 页码: 13
作者:
Jiang, Bo
;
Luo, Jiao
;
Guo, Shuju
;
Wang, Lijun
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2021/05/11
Type 2 diabetes mellitus
Protein tyrosine phosphatase 1B inhibitors
Thiazolidinedione
Insulin signaling
Anti-diabetic activities
Design, synthesis and biological evaluation of uncharged catechol derivatives as selective inhibitors of PTP1B
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 136, 页码: 348-359
作者:
Li, Xiang-Qian
;
Xu, Qi
;
Luo, Jiao
;
Wang, Li-Jun
;
Jiang, Bo
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2017/10/09
Type 2 Diabetes
Ptp1b Inhibition
Selectivity
Competitive
Cellular Activity
Discovery and evaluation of the hybrid of bromophenol and saccharide as potent and selective protein tyrosine phosphatase 1B inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 134, 页码: 24-33
作者:
Zhang, Renshuai
;
Yu, Rilei
;
Xu, Qi
;
Li, Xiangqian
;
Luo, Jiao
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  |  
浏览/下载:24/0
  |  
提交时间:2017/07/10
PTP1B
Bromophenol
Saccharide
Selectivity
Permeability
The design strategy of selective PTP1B inhibitors over TCPTP
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 16, 页码: 3343-3352
作者:
Li, XiangQian
;
Wang, LiJun
;
Shi, DaYong
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  |  
浏览/下载:11/0
  |  
提交时间:2016/12/05
Selectivity
PTP1B inhibitor
TCPTP
Diabetes
Design strategy
Discovery of novel bromophenol 3,4-dibromo-5-(2-bromo-3,4-dihydroxy-6-(isobutoxymethyl)benzyl)benzene-1,2-diol as protein tyrosine phosphatase 1B inhibitor and its anti-diabetic properties in C57BL/KsJ-db/db mice
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 64, 页码: 129-136
作者:
Jiang, Bo
;
Guo, Shuju
;
Shi, Dayong
;
Guo, Chao
;
Wang, Tao
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2014/07/17
Type 2 diabetes mellitus
Protein tyrosine phosphatase 1B
Bromophenol
Anti-diabetic activities
HPN, a Synthetic Analogue of Bromophenol from Red Alga Rhodomela confervoides: Synthesis and Anti-Diabetic Effects in C57BL/KsJ-db/db Mice
期刊论文
MARINE DRUGS, 2013, 卷号: 11, 期号: 2, 页码: 350-362
作者:
Shi, Dayong
;
Guo, Shuju
;
Jiang, Bo
;
Guo, Chao
;
Wang, Tao
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2014/07/17
bromophenol
protein tyrosine phosphatase 1B inhibitor
db/db mouse model
anti-diabetes properties
Bromophenols as inhibitors of protein tyrosine phosphatase 1B with antidiabetic properties
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 卷号: 22, 期号: 8, 页码: 2827-2832
作者:
Shi, Dayong
;
Li, Jing
;
Jiang, Bo
;
Guo, Shuju
;
Su, Hua
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  |  
浏览/下载:18/0
  |  
提交时间:2013/09/24
Bromophenol derivatives
Protein tyrosine phosphatase 1B
Diarylmethane
Antidiabetic activities
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