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Repressing MYC by targeting BET synergizes with selective inhibition of PI3K alpha against B cell lymphoma 期刊论文
CANCER LETTERS, 2022, 卷号: 524, 页码: 206-218
作者:  Chen, Zi-qi;  Cao, Zhe-rui;  Wang, Yi;  Zhang, Xi;  Xu, Lan
收藏  |  浏览/下载:53/0  |  提交时间:2021/12/16
CYH33  MYC  P300  BET  B cell lymphoma  PI3K  
Structure-Guided Development of Small-Molecule PRC2 Inhibitors Targeting EZH2-EED Interaction 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 12, 页码: 8194-8207
作者:  Du, Daohai;  Xu, Dandan;  Zhu, Licheng;  Stazi, Giulia;  Zwergel, Clemens
收藏  |  浏览/下载:74/0  |  提交时间:2021/08/17
EZH2 inhibitors abrogate upregulation of trimethylation of H3K27 by CDK9 inhibitors and potentiate its activity against diffuse large B-cell lymphoma 期刊论文
HAEMATOLOGICA, 2020, 卷号: 105, 期号: 4, 页码: 1021-1031
作者:  Xie, Shao;  Wei, Fan;  Sun, Yi-ming;  Gao, Ying-lei;  Pan, Lu-lu
收藏  |  浏览/下载:38/0  |  提交时间:2020/07/01
AZD9291 inactivates the PRC2 complex to mediate tumor growth inhibition 期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 12, 页码: 1587-1595
作者:  Zhang, Kai-li;  Shen, Qian-qian;  Fang, Yan-fen;  Sun, Yi-ming;  Ding, Jian
收藏  |  浏览/下载:27/0  |  提交时间:2020/07/01
Integrated Proteogenomic Characterization of HBV-Related Hepatocellular Carcinoma 期刊论文
CELL, 2019, 卷号: 179, 期号: 2, 页码: 561-+
作者:  Gao, Qiang;  Zhu, Hongwen;  Dong, Liangqing;  Shi, Weiwei;  Chen, Ran
收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01
Targeting Epigenetic Crosstalk as a Therapeutic Strategy for EZH2-Aberrant Solid Tumors 期刊论文
CELL, 2018, 卷号: 175, 期号: 1, 页码: 186-+
作者:  Huang, Xun;  Yan, Juan;  Zhang, Min;  Wang, Yafang;  Chen, Yi
收藏  |  浏览/下载:77/0  |  提交时间:2019/01/08
Lower genomic stability of induced pluripotent stem cells reflects increased non-homologous end joining 期刊论文
CANCER COMMUNICATIONS, 2018, 卷号: 38
作者:  Zhang, Minjie;  Wang, Liu;  An, Ke;  Cai, Jun;  Li, Guochao
收藏  |  浏览/下载:60/0  |  提交时间:2019/01/08
Discovery of novel Ponatinib analogues for reducing KDR activity as potent FGFRs inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 126, 页码: 122-132
作者:  Liu, Yang;  Peng, Xia;  Guan, Xiaocong;  Lu, Dong;  Xi, Yong
收藏  |  浏览/下载:42/0  |  提交时间:2019/01/08
exploitinghistonedeacetylasesforcancertherapyfromhematologicalmalignanciestosolidtumors 期刊论文
sciencechinalifesciences, 2017, 卷号: 60, 期号: 1, 页码: 94
作者:  Huang Min;  Geng Meiyu
收藏  |  浏览/下载:4/0  |  提交时间:2020/07/01
Identification of novel candidate drivers connecting different dysfunctional levels for lung adenocarcinoma using protein-protein interactions and a shortest path approach 期刊论文
SCIENTIFIC REPORTS, 2016, 卷号: 6
作者:  Chen, Lei;  Huang, Tao;  Zhang, Yu-Hang;  Jiang, Yang;  Zheng, Mingyue
收藏  |  浏览/下载:12/0  |  提交时间:2019/01/08


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