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期刊论文 [31]
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Facile and Cost-Effective Route for the Synthesis of Simmerafil
期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 11, 页码: 2432-2437
作者:
Odilov, Abdullajon
;
Liu, Yin
;
Hu, Tianwen
;
Jiang, Xiangrui
;
Suo, Jin
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2022/01/18
simmerafil
PDE5 inhibitor
salicylamide
synthesis
Design and development of an oral remdesivir derivative VV116 against SARS-CoV-2
期刊论文
CELL RESEARCH, 2021, 页码: 3
作者:
Xie, Yuanchao
;
Yin, Wanchao
;
Zhang, Yumin
;
Shang, Weijuan
;
Wang, Zhen
收藏
  |  
浏览/下载:108/0
  |  
提交时间:2021/11/04
Weinreb Amide Approach to the Practical Synthesis of a Key Remdesivir Intermediate
期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 7, 页码: 5065-5072
作者:
Xie, Yuanchao
;
Hu, Tianwen
;
Zhang, Yan
;
Wei, Daibao
;
Zheng, Wei
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/08/17
A Phase I Study to Evaluate the Safety, Tolerability, and Pharmacokinetics of TPN171H, a Novel Phosphodiesterase Type 5 Inhibitor, in Healthy Subjects
期刊论文
DRUG DESIGN DEVELOPMENT AND THERAPY, 2021, 卷号: 15, 页码: 2947-2959
作者:
Qian, Hongjie
;
Chen, Qian
;
Lang, Liyu
;
Zou, Yang
;
Pu, Huahua
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2021/08/17
TPN171H
PDE5 inhibitor
safety
pharmacokinetics
food effect
healthy subjects
Weinreb Amide Approach to the Practical Synthesis of a Key Remdesivir Intermediate
期刊论文
The Journal of organic chemistry, 2021, 卷号: 86, 期号: 7, 页码: 5065-5072
作者:
Xie, Yuanchao
;
Hu, Tianwen
;
Zhang, Yan
;
Wei, Daibao
;
Zheng, Wei
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/05/06
Structural basis for inhibition of the RNA-dependent RNA polymerase from SARS-CoV-2 by remdesivir
期刊论文
SCIENCE, 2020, 卷号: 368, 期号: 6498, 页码: 1499-+
作者:
Yin, Wanchao
;
Mao, Chunyou
;
Luan, Xiaodong
;
Shen, Dan-Dan
;
Shen, Qingya
收藏
  |  
浏览/下载:56/0
  |  
提交时间:2020/12/24
Improved Synthesis of 6-Chloro-5-methylpyridin-2-amine: A Key Intermediate for Making Lumacaftor
期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2020, 卷号: 24, 期号: 6, 页码: 1175-1179
作者:
Zhang, Junchi
;
Zhu, Fuqiang
;
Tian, Guanghui
;
Jiang, Xiangrui
;
Shen, Jingshan
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/12/24
6-chloro-5-methylpyridin-2-amine
lumacaftor
methylation
safe
Effect of irrigation methods on root growth, root-shoot ratio and yield components of cotton by regulating the growth redundancy of root and shoot
期刊论文
AGRICULTURAL WATER MANAGEMENT, 2020, 卷号: 234
作者:
Wang, Jiangtao
;
Du, Gangfeng
;
Tian, Jingshan
;
Zhang, Yali
;
Jiang, Chuangdao
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/03/01
Mulched drip irrigation
Cotton
Root growth
Root-shoot ratio
Growth redundancy
Pharmacokinetics-Driven Optimization of 4(3H)-Pyrimidinones as Phosphodiesterase Type 5 Inhibitors Leading to TPN171, a Clinical Candidate for the Treatment of Pulmonary Arterial Hypertension
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 10, 页码: 4979-4990
作者:
Wang, Zhen
;
Jiang, Xiangrui
;
Zhang, Xianglei
;
Tian, Guanghui
;
Yang, Rulei
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2020/07/01
Continuation of structure-activity relationship study of novel benzamide derivatives as potential antipsychotics
期刊论文
ARCHIV DER PHARMAZIE, 2019, 卷号: 352, 期号: 4, 页码: 13
作者:
Xu, Mingshuo
;
Guo, Shuang
;
Yang, Feipu
;
Wang, Yu
;
Wu, Chunhui
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2020/07/01
5-HT1A
5-HT2A
catalepsy
D-2
PCP-induced hyperactivity
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