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Design, Synthesis, and Biological Evaluation of 3-(Imidazo[1,2-a]pyrazin-3-ylethynyl)-4-isopropyl-N-(3-((4-methylpiperazin-1-yl)methyl)-5-(trifluoromethyl)phenyl)benzamide as a Dual Inhibitor of Discoidin Domain Receptors 1 and 2 期刊论文
2018, 卷号: 61, 期号: 17, 页码: 7977
作者:  Wang, Zhen[1,2];  Zhang, Yali[3];  Pinkas, Daniel M.[7];  Fox, Alice E.[7];  Luo, Jinfeng[2]
收藏  |  浏览/下载:27/0  |  提交时间:2019/12/17
Inhibition of Discoidin Domain Receptor 1 Reduces Collagen-mediated Tumorigenicity in Pancreatic Ductal Adenocarcinoma 期刊论文
2017, 卷号: 16, 期号: [db:dc_citation_issue], 页码: 2473
作者:  Aguilera, Kristina Y.[1,2];  Huang, Huocong[1,2];  Du, Wenting[1,2];  Hagopian, Moriah M.[1,2];  Wang, Zhen[3]
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/03
Tetrahydroisoquinoline-7-carboxamide Derivatives as New Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
2017, 卷号: 8, 期号: 3, 页码: 327
作者:  Wang, Zhen[1,2];  Zhang, Yali[3];  Bartual, Sergio G.[5];  Luo, Jinfeng[2];  Xu, Tingting[4]
收藏  |  浏览/下载:22/0  |  提交时间:2019/12/06
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
2016, 卷号: 59, 期号: [db:dc_citation_issue], 页码: 5911
作者:  Wang, Zhen[1,2];  Bian, Huan[4];  Bartual, Sergio G.[5];  Du, Wenting[6,7];  Luo, Jinfeng[1]
收藏  |  浏览/下载:5/0  |  提交时间:2019/12/03
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
Wang, Zhen; Bian, Huan; Bartual, Sergio G.; Du, Wenting; Luo, Jinfeng; Zhao, Hu; Zhang, Shasha; Mo, Cheng; Zhou, Yang; Xu, Yong; Tu, Zhengchao; Ren, Xiaomei; Lu, Xiaoyun; Brekken, Rolf A.; Yao, Libo; Bullock, Alex N.; Su, Jin; Ding, Ke
收藏  |  浏览/下载:50/0  |  提交时间:2016/12/16
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
作者:  Yao, Libo;  Ding, Ke;  Su, Jin;  Bullock, Alex N.;  Brekken, Rolf A.
收藏  |  浏览/下载:32/0  |  提交时间:2018/12/13
CXCL1 promotes tumor growth through VEGF pathway activation and is associated with inferior survival in gastric cancer 期刊论文
CANCER LETTERS, 2015, 卷号: 359, 页码: 335-343
作者:  Wei, Zhe-Wei[1,2];  Xia, Guang-Kai[1,2];  Wu, Ying[1,2];  Chen, Wei[1,2];  Xiang, Zhen[1,2]
收藏  |  浏览/下载:3/0  |  提交时间:2019/04/25


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