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A proteomic and phosphoproteomic landscape of KRAS mutant cancers identifies combination therapies 期刊论文
MOLECULAR CELL, 2021, 卷号: 81, 期号: 19, 页码: 4076-+
作者:  Liu, Zhiwei;  Liu, Yingluo;  Qian, Lili;  Jiang, Shangwen;  Gai, Xiameng
收藏  |  浏览/下载:24/0  |  提交时间:2021/12/01
Design, synthesis and pharmacological evaluation of bicyclic and tetracyclic pyridopyrimidinone analogues as new KRAS(G12C) inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 213, 页码: 17
作者:  Xiao, Xuanzheng;  Lai, Mengzhen;  Song, Zilan;  Geng, Meiyu;  Ding, Jian
收藏  |  浏览/下载:47/0  |  提交时间:2021/05/24
Simultaneous inhibition of PI3K alpha and CDK4/6 synergistically suppresses Kras-mutated non-small cell lung cancer 期刊论文
MOLECULAR CANCER RESEARCH, 2020, 卷号: 18, 期号: 10, 页码: 44-45
作者:  Wang, Yu-xiang;  Li, Xian;  Liu, Xue-ling;  Wang, Bo-bo;  Chen, Yi
收藏  |  浏览/下载:12/0  |  提交时间:2020/07/01
EPHA2 feedback activation limits the response to PDE delta inhibition in KRAS-dependent cancer cells 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 2, 页码: 270-277
作者:  Chen, Yue-hong;  Lv, Hao;  Shen, Ning;  Wang, Xiao-min;  Tang, Shuai
收藏  |  浏览/下载:33/0  |  提交时间:2020/07/01
Identification of a new inhibitor of KRAS-PDE delta interaction targeting KRAS mutant nonsmall cell lung cancer 期刊论文
INTERNATIONAL JOURNAL OF CANCER, 2019, 卷号: 145, 期号: 5, 页码: 1334-1345
作者:  Leung, Elaine Lai-Han;  Luo, Lian Xiang;  Li, Ying;  Liu, Zhong-Qiu;  Li, Lan Lan
收藏  |  浏览/下载:14/0  |  提交时间:2020/07/01
Fragment-based drug discovery of triazole inhibitors to block PDE delta-RAS protein-protein interaction 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 163, 页码: 597-609
作者:  Chen, Danqi;  Chen, Yuehong;  Lian, Fulin;  Chen, Liu;  Li, Yanlian
收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
MiR-1205 functions as a tumor suppressor by disconnecting the synergy between KRAS and MDM4/E2F1 in non-small cell lung cancer 期刊论文
AMERICAN JOURNAL OF CANCER RESEARCH, 2019, 卷号: 9, 期号: 2, 页码: 312-+
作者:  Yan, Hong;  Chen, Xiaoying;  Li, Yu;  Fan, Lei;  Tai, Yusi
收藏  |  浏览/下载:4/0  |  提交时间:2020/07/01
Simultaneous inhibition of PI3Kα and CDK4/6 synergistically suppresses KRAS-mutated non-small cell lung cancer 期刊论文
Cancer Biology and Medicine, 2019, 卷号: 16, 期号: 1, 页码: 66
作者:  Wang Yuxiang;  Li Xian;  Liu Xueling;  Chen Yi;  Yang Chunhao
收藏  |  浏览/下载:13/0  |  提交时间:2020/12/24
PI3Kα  CDK4/6  KRAS  NSCLC  CYH33  
simultaneousinhibitionofpi3kandcdk46synergisticallysuppresseskrasmutatednonsmallcelllungcancer 期刊论文
癌症生物学与医学英文版, 2019, 卷号: 016, 期号: 001, 页码: 66
作者:  Yuxiang Wang;  Xian Li;  Xueling Liu;  Yi Chen;  Chunhao Yang
收藏  |  浏览/下载:12/0  |  提交时间:2020/07/01
PI3Kα  CDK4/6  KRAS  NSCLC  CYH33  
Inhibition of KRAS-dependent lung cancer cell growth by deltarasin: blockage of autophagy increases its cytotoxicity 期刊论文
CELL DEATH & DISEASE, 2018, 卷号: 9
作者:  Leung, Elaine Lai Han;  Luo, Lian Xiang;  Liu, Zhong Qiu;  Wong, Vincent Kam Wai;  Lu, Lin Lin
收藏  |  浏览/下载:24/0  |  提交时间:2019/01/08


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