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科研机构
上海药物研究所 [135]
内容类型
期刊论文 [134]
会议论文 [1]
发表日期
2021 [7]
2020 [7]
2019 [6]
2018 [11]
2017 [5]
2016 [14]
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Chemistry [4]
Biochemist... [2]
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Enones as Alkenyl Reagents via Ligand-Promoted C-C Bond Activation
期刊论文
ACS CATALYSIS, 2021, 页码: 82-88
作者:
Li, Hanyuan
;
Wang, Mei-Ling
;
Liu, Yu-Wen
;
Li, Ling-Jun
;
Xu, Hui
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2022/01/18
C-C bond activation
enone
olefination
Pd-catalyzed
late-stage diversification
Effects of Food on the Pharmacokinetic Properties and Mass Balance of Henagliflozin in Healthy Male Volunteers
期刊论文
CLINICAL THERAPEUTICS, 2021, 卷号: 43, 期号: 9, 页码: E264-E273
作者:
Chen, Zhen-dong
;
Chen, Qian
;
Zhu, Yun-ting
;
Zhang, Yi-fan
;
Zhan, Yan
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2022/01/04
henagliflozin
food effects
mass balance
pharmacokinetics
SGLT-2 inhibitor
DFT Mechanism of Cu Catalyzed Coupling Reaction to Alkyl Aryl Ethers
期刊论文
ACTA CHIMICA SINICA, 2021, 卷号: 79, 期号: 7, 页码: 948-952
作者:
Man, Qingmin
;
Fu, Zunyun
;
Liu, Tiantian
;
Zheng, Mingyue
;
Jiang, Hualiang
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2021/11/04
density functional theory
Cu catalyzed
Ullmann C=O coupling
tert-butoxide
Targeting sorting nexin 10 improves mouse colitis via inhibiting PIKfyve-mediated TBK1/c-Rel signaling activation
期刊论文
PHARMACOLOGICAL RESEARCH, 2021, 卷号: 169, 页码: 11
作者:
Bao, Weilian
;
Liu, Xiaohong
;
You, Yan
;
Hou, Hui
;
Wang, Xu
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2021/11/16
SNX10
IBD
Macrophage
PIKfyve
TBK1
PPI inhibitor
Rhodium-Catalyzed C-H Activation/Annulation Cascade of Aryl Oximes and Propargyl Alcohols to Isoquinoline N-Oxides
期刊论文
ADVANCED SYNTHESIS & CATALYSIS, 2021, 页码: 7
作者:
Li, Yuan
;
Fang, Feifei
;
Zhou, Jianhui
;
Li, Jiyuan
;
Wang, Run
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2021/08/17
Isoquinoline N-oxides
beta-hydroxy elimination
Rhodium
Secondary propargyl alcohols
Exploration of tissue distribution of ginsenoside Rg1 by LC-MS/MS and nanospray desorption electrospray ionization mass spectrometry
期刊论文
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2021, 卷号: 198, 页码: 7
作者:
Wei, Wenlong
;
Li, Zhenwei
;
Li, Haojv
;
An, Yaling
;
Qu, Hua
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2021/05/24
Ginsenoside Rg1
Nanospray desorption electrospray ionization
Tissue distribution
Spatial distribution
Tumor-permeated bioinspired theranostic nanovehicle remodels tumor immunosuppression for cancer therapy
期刊论文
BIOMATERIALS, 2021, 卷号: 269, 页码: 15
作者:
Wang, Hong
;
Li, Jie
;
Wang, Zhiwan
;
Wang, Yuqi
;
Xu, Xiaoxuan
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2021/05/24
Melittin
Gemcitabine
Photodynamic therapy
Nanoparticle
Immunosuppression
Pharmacokinetics, mass balance, and metabolism of [C-14]vicagrel, a novel irreversible P2Y(12) inhibitor in humans
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 12
作者:
Zheng, Yuan-dong
;
Zhang, Hua
;
Zhan, Yan
;
Bian, Yi-cong
;
Ma, Sheng
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2021/05/24
vicagrel
[C-14]vicagrel
vicagrel pharmacokinetics
vicagrel metabolism
mass balance
P2Y(12) receptor inhibitor
Clinical application of pyrrole-hemoglobin adducts as a biomarker of pyrrolizidine alkaloid exposure in humans
期刊论文
ARCHIVES OF TOXICOLOGY, 2020, 页码: 7
作者:
Ma, Jiang
;
Zhang, Wei
;
He, Yisheng
;
Zhu, Lin
;
Zhang, Chunyuan
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2020/12/24
Pyrrolizidine alkaloids
Liver injury
Diagnostic biomarkers
Pyrrole-hemoglobin adducts
Pyrrole-plasma protein adducts
Transformations of Aryl Ketones via Ligand-Promoted C-C Bond Activation
期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2020, 页码: 7
作者:
Li, Hanyuan
;
Ma, Biao
;
Liu, Qi-Sheng
;
Wang, Mei-Ling
;
Wang, Zhen-Yu
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2020/12/24
aryl ketones
borylation
C-C bond activation
Pd catalysis
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