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吉林大学白求恩第一... [14]
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Discovery and structure - activity relationship exploration of pyrazolo [1,5-a]pyrimidine derivatives as potent FLT3-ITD inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 48, 页码: 13
作者:
Chen, Yun
;
Bai, Gang
;
Li, Yan
;
Ning, Yi
;
Cao, Sufen
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2021/12/01
FLT3
FLT3-ITD
Acute myeloid leukemia
Structure-activity relationships
Pyrazolo[1, 5-a]pyrimidine
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:
Xue, Yu
;
Song, Peiran
;
Song, Zilan
;
Wang, Aoli
;
Tong, Linjiang
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2019/08/23
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:
Xue, Yu
;
Song, Peiran
;
Song, Zilan
;
Wang, Aoli
;
Tong, Linjiang
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2019/01/08
Pyrazolo[3,4-d]pyrimidine derivatives containing a Schiff base moiety as potential antiviral agents
期刊论文
2018, 卷号: 28, 期号: 17, 页码: 2979-2984
作者:
Wang, Yan-Yan
;
Xu, Fang-Zhou
;
Zhu, Yun-Ying
;
Song, Baoan
;
Liu, Dexia
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2020/01/05
c-Src regulates cell cycle proteins expression through protein kinase B/glycogen synthase kinase 3 beta and extracellular signal-regulated kinases 1/2 pathways in MCF-7 cells
期刊论文
acta biochimica et biophysica sinica, 2013
Liu, Xiang
;
Du, Liying
;
Feng, Renqing
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  |  
浏览/下载:3/0
  |  
提交时间:2015/11/13
breast cancer
cell cycle proteins
c-Src suppression
PP2
siRNAs
BREAST-CANCER CELLS
FAMILY KINASES
DEPENDENT KINASES
G(1) PHASE
P27(KIP1)
D1
PHOSPHORYLATION
PROGRESSION
INHIBITOR
RECEPTOR
An in silico exploration of the interaction mechanism of pyrazolo[1,5-a]pyrimidine type CDK2 inhibitors
期刊论文
molecular biosystems, 2013, 卷号: 9, 期号: 9, 页码: 2266-2281
作者:
Li, Yan
;
Gao, Weimin
;
Li, Feng
;
Wang, Jinghui
;
Zhang, Jingxiao
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  |  
浏览/下载:28/0
  |  
提交时间:2015/11/09
A facile and efficient one-pot three-step protocol for synthesis of 6-aryl-7-oxo-5-aryoxy/alkoxy-1-(p-tolyl)-6,7-dihydro-1H-pyrazolo[4,3-d] pyrimidine-3-carbonitrile
期刊论文
Arkivoc, 2012, 卷号: 2012, 期号: 6, 页码: 295-303
作者:
Wu, Ming-Hu*
;
Hu, Ji-Huan
;
Guo, Hai-Bing
;
Li, Yan
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  |  
浏览/下载:7/0
  |  
提交时间:2019/12/23
1H-pyrazolo[4
3-d]pyrimidin-7(6H)-one
Aza-Wittig reaction
Domino reaction
Nitrogen heterocycle
F-18-labeled Pyrazolo[1,5-a]pyrimidine Derivatives: Synthesis from 2,4-Dinitrobenzamide and Tosylate Precursors and Comparative Biological Evaluation for Tumor Imaging with Positron Emission Tomography
期刊论文
2012, 卷号: 17, 期号: 4, 页码: 3774-3793
作者:
Xu, Jingli
;
Liu, Hang
;
Li, Guixia
;
He, Yong
;
Ding, Rui
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2020/01/13
F-18-labeled
pyrazolo[1
5-a]pyrimidine derivatives
2
4-dinitrobenzamide and tosylate precursors
PET imaging agents
tumor detection
Efficient Synthesis of Fused Pyrimidine Derivatives with Biological Activity via Aza-Wittig Reaction
期刊论文
Current Organic Synthesis, 2011, 卷号: 8, 期号: 5, 页码: 752-763
作者:
Ren Qingyun
;
Tan Xiaosong
;
He Hongwu*
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/12/23
1,2,3-triazolo[4,5-d]pyrimidin-7-ones
1,2,4-triazolo[1,5-a]pyrimidin- 10(3H)-ones
3,4-dihydro-pyrido[4,3-d] pyrimidine-8-carbonitriles
Fused pyrimidine derivatives
aza-Wittig reaction
fungicidal activity
herbicidal activity
pharmaceutical activity
pyrazolo[3,4-b]pyrido[4,3-d]-pyrimidine-4-ones
pyrazolo[4',3':5,6] pyrano[2,3-d]pyrimidin-4 (3H)-ones
pyrido[4,3-d]pyrimidine-4(3H)-ones
synthesis
thiazolo[4,5-d] pyrimidin-4(3H)-ones
thieno[3',2'-5,6]pyrido [4,3-d]pyrimidin-4(3H)-ones
Synthesis and biological evaluation of novel F-18 labeled pyrazolo[1,5-a] pyrimidine derivatives: Potential PET imaging agents for tumor detection
期刊论文
2011, 卷号: 21, 期号: 16, 页码: 4736-4741
作者:
Xu, Jingli
;
Liu, Hang
;
Li, Guixia
;
He, Yong
;
Ding, Rui
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2020/01/13
F-18 labeled
Pyrazolo[1
5-a] pyrimidine derivatives
PET imaging agents
Tumor detection
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