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Discovery and structure - activity relationship exploration of pyrazolo [1,5-a]pyrimidine derivatives as potent FLT3-ITD inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 48, 页码: 13
作者:  Chen, Yun;  Bai, Gang;  Li, Yan;  Ning, Yi;  Cao, Sufen
收藏  |  浏览/下载:32/0  |  提交时间:2021/12/01
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:  Xue, Yu;  Song, Peiran;  Song, Zilan;  Wang, Aoli;  Tong, Linjiang
收藏  |  浏览/下载:32/0  |  提交时间:2019/08/23
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:  Xue, Yu;  Song, Peiran;  Song, Zilan;  Wang, Aoli;  Tong, Linjiang
收藏  |  浏览/下载:36/0  |  提交时间:2019/01/08
Pyrazolo[3,4-d]pyrimidine derivatives containing a Schiff base moiety as potential antiviral agents 期刊论文
2018, 卷号: 28, 期号: 17, 页码: 2979-2984
作者:  Wang, Yan-Yan;  Xu, Fang-Zhou;  Zhu, Yun-Ying;  Song, Baoan;  Liu, Dexia
收藏  |  浏览/下载:1/0  |  提交时间:2020/01/05
c-Src regulates cell cycle proteins expression through protein kinase B/glycogen synthase kinase 3 beta and extracellular signal-regulated kinases 1/2 pathways in MCF-7 cells 期刊论文
acta biochimica et biophysica sinica, 2013
Liu, Xiang; Du, Liying; Feng, Renqing
收藏  |  浏览/下载:3/0  |  提交时间:2015/11/13
An in silico exploration of the interaction mechanism of pyrazolo[1,5-a]pyrimidine type CDK2 inhibitors 期刊论文
molecular biosystems, 2013, 卷号: 9, 期号: 9, 页码: 2266-2281
作者:  Li, Yan;  Gao, Weimin;  Li, Feng;  Wang, Jinghui;  Zhang, Jingxiao
收藏  |  浏览/下载:28/0  |  提交时间:2015/11/09
A facile and efficient one-pot three-step protocol for synthesis of 6-aryl-7-oxo-5-aryoxy/alkoxy-1-(p-tolyl)-6,7-dihydro-1H-pyrazolo[4,3-d] pyrimidine-3-carbonitrile 期刊论文
Arkivoc, 2012, 卷号: 2012, 期号: 6, 页码: 295-303
作者:  Wu, Ming-Hu*;  Hu, Ji-Huan;  Guo, Hai-Bing;  Li, Yan
收藏  |  浏览/下载:7/0  |  提交时间:2019/12/23
F-18-labeled Pyrazolo[1,5-a]pyrimidine Derivatives: Synthesis from 2,4-Dinitrobenzamide and Tosylate Precursors and Comparative Biological Evaluation for Tumor Imaging with Positron Emission Tomography 期刊论文
2012, 卷号: 17, 期号: 4, 页码: 3774-3793
作者:  Xu, Jingli;  Liu, Hang;  Li, Guixia;  He, Yong;  Ding, Rui
收藏  |  浏览/下载:2/0  |  提交时间:2020/01/13
Efficient Synthesis of Fused Pyrimidine Derivatives with Biological Activity via Aza-Wittig Reaction 期刊论文
Current Organic Synthesis, 2011, 卷号: 8, 期号: 5, 页码: 752-763
作者:  Ren Qingyun;  Tan Xiaosong;  He Hongwu*
收藏  |  浏览/下载:9/0  |  提交时间:2019/12/23
Synthesis and biological evaluation of novel F-18 labeled pyrazolo[1,5-a] pyrimidine derivatives: Potential PET imaging agents for tumor detection 期刊论文
2011, 卷号: 21, 期号: 16, 页码: 4736-4741
作者:  Xu, Jingli;  Liu, Hang;  Li, Guixia;  He, Yong;  Ding, Rui
收藏  |  浏览/下载:1/0  |  提交时间:2020/01/13


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