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科研机构
上海药物研究所 [4]
高能物理研究所 [4]
复旦大学上海医学院 [4]
中国医学科学院 北京... [3]
清华大学 [2]
重庆大学 [2]
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期刊论文 [20]
会议论文 [4]
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Design, synthesis and antitumor study of a series of N-Cyclic sulfamoylaminoethyl substituted 1,2,5-oxadiazol-3-amines as new indoleamine 2, 3-dioxygenase 1 (IDO1) inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 179, 页码: 38-55
作者:
Chen, Shulun
;
Guo, Wei
;
Liu, Xiaohua
;
Sun, Pu
;
Wang, Yi
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/07/01
Indoleamine 2,3-dioxygenase
Immunotherapy
Oxadiazole
PD-1
Life span
Dose Optimization of Colistin Combinations against Carbapenem-Resistant Acinetobacter baumannii from Patients with Hospital-Acquired Pneumonia in China by Using an In Vitro Pharmacokinetic/Pharmacodynamic Model
期刊论文
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2019, 卷号: 63, 期号: 4
作者:
Liu, Xiaofen
;
Chen, Daijie
;
Li, Jian
;
Zhang, Jing
;
Bian, Xingchen
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/12/05
Acinetobacter baumannii
PK/PD modeling
carbapenem resistance
colistin
combination therapy
meropenem
Dose Optimization of Colistin Combinations against Carbapenem-Resistant Acinetobacter baumannii from Chinese Hospital-acquired Pneumonia Patients Using In Vitro PK/PD Model.
期刊论文
Antimicrobial agents and chemotherapy, 2019
作者:
Xingchen Bian
;
Xiaofen Liu
;
Yuancheng Chen
;
Daijie Chen
;
Jian Li
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2019/12/17
Pharmacokinetics-pharmacodynamics and tissue distribution analysis of Low Polar extract of Xiaoyao Powder combined with rat model of chronic unpredictable mild stress
期刊论文
2019, 卷号: 42, 期号: 7-8, 页码: 173-183
作者:
Gao, Xiaoxia
;
Wang, Peng
;
Wu, Li
;
Liu, Jiali
;
Fang, Yuan
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2020/01/03
Pharmacokinetics-pharmacodynamics (PK-PD)
low polar extract of Xiaoyao powder (XYP-A)
polyacetylene
Chronic Unpredictable Mild Stress (CUMS)
monoamine neurotransmitters
Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 896-916
作者:
Wang, Beilei
;
Wu, Jiaxin
;
Wu, Yun
;
Chen, Cheng
;
Zou, Fengming
收藏
  |  
浏览/下载:65/0
  |  
提交时间:2019/12/25
CDK9
Kinase inhibitor
Structure-activity relationship
Leukemia
In Vitro Anaerobic Pharmacokinetic/Pharmacodynamic Model to Simulate the Bactericidal Activity of Levornidazole Against Bacteroides fragilis
期刊论文
CLINICAL THERAPEUTICS, 2017, 卷号: 39, 期号: 4
作者:
Hu, Jiali
;
Zhang, Jing
;
Chen, Yuancheng
;
Liang, Wang
;
Wu, Shi
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/12/05
anaerobe
dynamic pharmacokinetic/pharmacodynamic model
in vitro
levornidazole
PK/PD target value
Population Pharmacokinetic/Pharmacodynamics Modeling of Ibutilide in Chinese Healthy Volunteers and Patients With Atrial Fibrillation (AF) and/or Atrial Flutter (AFL)
期刊论文
2017, 卷号: 39, 期号: 7, 页码: 1320-1335
作者:
Zeng, Zhijun
;
Wang, Li
;
Hua, Lu
;
Jiang, Juanjuan
;
Pang, Huimin
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/01/04
ibutilide
NONMEM
population PK and PK/PD model
QT interval prolongation
sigmoid E-max model
HER2-targeted antibody drug conjugates for ovarian cancer therapy
期刊论文
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2016, 卷号: 93, 页码: 274-286
作者:
Jiang, Jing
;
Dong, Lihou
;
Wang, Lei
;
Wang, Ling
;
Zhang, Jing
收藏
  |  
浏览/下载:52/0
  |  
提交时间:2019/01/08
Ovarian cancer
Antibody drug conjugates (ADCs)
HER2/ErbB2
Monomethyl auristatin E (MMAE)
Synergistic killing by meropenem and colistin combination of carbapenem-resistant Acinetobacter baumannii isolates from Chinese patients in an in vitro pharmacokinetic/pharmacodynamic model
期刊论文
INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS, 2016, 卷号: 48, 期号: 5
作者:
Liu, Xiaofen
;
Zhao, Miao
;
Chen, Yuancheng
;
Bian, Xingchen
;
Li, Yunfei
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/13
Carbapenem-resistant Acinetobacter baumannii
Meropenem
Colistin
Combination therapy
In vitro
PK/PD model
Antitumor effects of CPT-11 liposomes on HT-29 Xenograft and PK/PD correlation evaluation
期刊论文
Chinese Journal New Drugs, 2014, 卷号: 23, 期号: 6, 页码: 721-726
作者:
Li Ning
;
Zhang Qing
;
Jia Linchao
;
Zheng Qingmei
;
Yan Lei
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
CPT-11
CPT-11
liposome
antitumor
PK/PD correlation
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