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科研机构
上海药物研究所 [9]
内容类型
期刊论文 [9]
发表日期
2018 [3]
2017 [3]
2015 [1]
2012 [1]
2008 [1]
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PBA2 exhibits potent anti-tumor activity via suppression of VEGFR2 mediated-cell proliferation and angiogenesis
期刊论文
BIOCHEMICAL PHARMACOLOGY, 2018, 卷号: 150, 页码: 131-140
作者:
Fang, Xiaona
;
Xie, Hua
;
Luo, Min
;
Chen, Zhen
;
Wang, Fang
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2019/01/08
Angiogenesis
And-tumor activity
Multi-tyrosine kinases inhibitor
PBA2
VEGFR2
SOMCL-085, a novel multi-targeted FGFR inhibitor, displays potent anticancer activity in FGFR-addicted human cancer models
期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 2, 页码: 243-250
作者:
Jiang, Xi-fei
;
Dai, Yang
;
Peng, Xia
;
Shen, Yan-yan
;
Su, Yi
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2019/01/08
human cancer
anticancer drug
SOMCL-085
receptor tyrosine kinase
FGFR
xenograft nude mouse model
somcl085anovelmultitargetedfgfrinhibitordisplayspotentanticanceractivityinfgfraddictedhumancancermodels
期刊论文
actapharmacologicasinica, 2018, 卷号: 39, 期号: 2, 页码: 243
作者:
Jiang Xifei
;
Dai Yang
;
Peng Xia
;
Shen Yanyan
;
Su Yi
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2020/07/01
human cancer
anticancer drug
SOMCL-085
receptor tyrosine kinase
FGFR
xenograft nude mouse model
Evaluation of in vitro and in vivo activity of a multityrosine kinase inhibitor, AL3810, against human thyroid cancer
期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1533-1542
作者:
Xie, Qin
;
Chen, Hui
;
Ai, Jing
;
Gao, Ying-lei
;
Geng, Mei-yu
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
thyroid cancer
AL3810
multi-tyrosine kinases inhibitor
angiogenesis
RET
Discovery of novel Ponatinib analogues for reducing KDR activity as potent FGFRs inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 126, 页码: 122-132
作者:
Liu, Yang
;
Peng, Xia
;
Guan, Xiaocong
;
Lu, Dong
;
Xi, Yong
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  |  
浏览/下载:42/0
  |  
提交时间:2019/01/08
FGFR
KDR
Inhibitor
Anticancer
Ponatinib
evaluationofinvitroandinvivoactivityofamultityrosinekinaseinhibitoral3810againsthumanthyroidcancer
期刊论文
actapharmacologicasinica, 2017, 卷号: 38, 期号: 11, 页码: 1533
作者:
Xie Qin
;
Chen Hui
;
Al Jing
;
Gao Yinglei
;
Geng Meiyu
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/07/01
TARGETED THERAPIES
RET
CARCINOMA
MODELS
GROWTH
TUMORS
CELLS
thyroid cancer
AL3810
multi-tyrosine kinases inhibitor
angiogenesis
RET
DCLAK11, a multi-tyrosine kinase inhibitor, exhibits potent antitumor and antiangiogenic activity in vitro
期刊论文
ACTA PHARMACOLOGICA SINICA, 2015, 卷号: 36, 期号: 10, 页码: 1266-1276
作者:
Guo, Xiao-bin
;
Zhu, Wei
;
Chen, Xian-jie
;
Tong, Lin-jiang
;
Peng, Xia
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2019/01/08
DCLAK11
substituted pyridin-3-amine derivatives
tyrosine kinase
EGFR
HER2
VEGFR2
anticancer
anti-angiogenesis
AL3810, a multi-tyrosine kinase inhibitor, exhibits potent anti-angiogenic and anti-tumour activity via targeting VEGFR, FGFR and PDGFR
期刊论文
JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, 2012, 卷号: 16, 期号: 10, 页码: 2321-2330
作者:
Zhou, Yuanfeng
;
Chen, Yi
;
Tong, Linjiang
;
Xie, Hua
;
Wen, Weiwei
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
multi-tyrosine kinases inhibitor
angiogenesis
anti-tumour activity
The Marine-Derived Oligosaccharide Sulfate (MdOS), a Novel Multiple Tyrosine Kinase Inhibitor, Combats Tumor Angiogenesis both In Vitro and In Vivo
期刊论文
PLOS ONE, 2008, 卷号: 3, 期号: 11
作者:
Ma, Jingui
;
Xin, Xianliang
;
Meng, Linghua
;
Tong, Linjiang
;
Lin, Liping
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
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