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Identification of Betulinic Acid Derivatives as Potent TGR5 Agonists with Antidiabetic Effects via Humanized TGR5(H88Y) Mutant Mice 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12181-12199
作者:  Yun, Ying;  Zhang, Chenlu;  Guo, Shimeng;  Liang, Xiaoying;  Lan, Yuan
收藏  |  浏览/下载:40/0  |  提交时间:2021/11/04
Design of G-protein-coupled bile acid receptor 1 (GPBAR1, TGR5) soft drugs with reduced gallbladder-filling effects 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 12
作者:  Han, Fanghui;  Ning, Mengmeng;  Cao, Hua;  Ye, Yangliang;  Feng, Ying
收藏  |  浏览/下载:32/0  |  提交时间:2020/12/21
The G-protein-coupled bile acid receptor Gpbar1 (TGR5) protects against renal inflammation and renal cancer cell proliferation and migration through antagonizing NF-kappa B and STAT3 signaling pathways 期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 33, 页码: 54378-54387
作者:  Su Jia[1];  Zhang Qiqi[2];  Qi Hui[3];  Wu Linlin[4];  Li Yuanqiang[5]
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/23
Discovery and Structure-Activity Relationship Study of 4-Phenoxythiazol-5-carboxamides as Highly Potent TGR5 Agonists 期刊论文
CHEMICAL & PHARMACEUTICAL BULLETIN, 2016, 卷号: 64, 期号: 4, 页码: 326-339
作者:  Chen, Zhixiang;  Ning, Mengmeng;  Zou, Qingan;  Cao, Hua;  Ye, Yangliang
收藏  |  浏览/下载:9/0  |  提交时间:2019/01/08
TGR5, Not Only a Metabolic Regulator 期刊论文
FRONTIERS IN PHYSIOLOGY, 2016, 卷号: 7
作者:  Guo, Cong[1];  Chen, Wei-Dong[2];  Wang, Yan-Dong[3]
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/23
Aberrant DNA methylation of G-protein-coupled bile acid receptor Gpbar1 predicts prognosis of acute-on-chronic hepatitis B liver failure 期刊论文
Journal of viral hepatitis., 2015, 卷号: 22, 期号: 2, 页码: 112-119
作者:  Gao, S.;  Ji, X-F;  Li, F.;  Sun, F-K;  Zhao, J.
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/17
The G-Protein-Coupled Bile Acid Receptor Gpbar1 (TGR5) Inhibits Gastric Inflammation Through Antagonizing NF-kappa B Signaling Pathway 期刊论文
FRONTIERS IN PHARMACOLOGY, 2015, 卷号: 6, 页码: 287
作者:  Guo, Cong[1];  Qi, Hui[2];  Yu, Yingjie[3];  Zhang, Qiqi[4];  Su, Jia[5]
收藏  |  浏览/下载:5/0  |  提交时间:2019/12/23
The G-protein-coupled bile acid receptor Gpbar1 (TGR5) suppresses gastric cancer cell proliferation and migration through antagonizing STAT3 signaling pathway 期刊论文
ONCOTARGET, 2015, 卷号: 6, 期号: 33, 页码: 34402-34413
作者:  Guo, Cong[1];  Su, Jia[2];  Li, Zhijun[3];  Xiao, Rui[4];  Wen, Jianxun[5]
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/23
Aberrant DNA Methylation of G-protein-coupled Bile Acid Receptor Gpbar1 (TGR5) is a Potential Biomarker for Hepatitis B Virus Associated Hepatocellular Carcinoma 期刊论文
INTERNATIONAL JOURNAL OF MEDICAL SCIENCES, 2014, 卷号: 11, 期号: 2, 页码: 164-171
作者:  Han, Li-Yan;  Fan, Yu-Chen;  Mu, Nan-Nan;  Gao, Shuai;  Li, Feng
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/17
Deficiency of G-Protein-Coupled Bile Acid Receptor Gpbar1 (TGR5) Enhances Chemically Induced Liver Carcinogenesis (Retracted article. See vol. 58, pg. 1194, 2013) 期刊论文
HEPATOLOGY, 2013, 卷号: 57, 期号: 2, 页码: 656-666
作者:  Chen, Wei-Dong[1];  Yu, Donna[2];  Forman, Barry M.[3];  Huang, Wendong[4];  Wang, Yan-Dong[5]
收藏  |  浏览/下载:6/0  |  提交时间:2019/12/23


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