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上海药物研究所 [6]
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期刊论文 [21]
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Architecture of the mycobacterial succinate dehydrogenase with a membrane-embedded Rieske FeS cluster
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118
作者:
Zhou, Xiaoting
;
Gao, Yan
;
Wang, Weiwei
;
Yang, Xiaolin
;
Yang, Xiuna
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2021/06/15
succinate dehydrogenase
Mycobacterium smegmatis
electron transport chain
cryoelectron microscopy
Pharmacokinetic Drug-drug Interaction of Antibiotics Used in Sepsis Care in China
期刊论文
CURRENT DRUG METABOLISM, 2021, 卷号: 22, 期号: 1, 页码: 5-23
作者:
Yu, Xuan
;
Chu, Zixuan
;
Li, Jian
;
He, Rongrong
;
Wang, Yaya
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  |  
浏览/下载:67/0
  |  
提交时间:2021/05/24
Pharmacokinetics
drug-drug interaction
antibiotic
sepsis
transporter
enzyme
Discovery of New and Potent InhA Inhibitors as Antituberculosis Agents: Structure-Based Virtual Screening Validated by Biological Assays and X-ray Crystallography
期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2020, 卷号: 60, 期号: 1, 页码: 226-234
作者:
Kamsri, Pharit
;
Hanwarinroj, Chayanin
;
Phusi, Naruedon
;
Pornprom, Thimpika
;
Chayajarus, Kampanart
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  |  
浏览/下载:23/0
  |  
提交时间:2020/07/01
Synthesis and Cdc25B/PTP1B Inhibitory Activity Evaluation of Novel Acylhydrazone Derivatives Containing Carbazole Moity
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 39, 期号: 2, 页码: 491-499
作者:
Li Yingjun
;
Wang Siyuan
;
Jin Kun
;
Gao Lixin
;
Sheng Li
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  |  
浏览/下载:17/0
  |  
提交时间:2020/07/01
acylhydrazone
carbazole
synthesis
Cdc25B and PTP1B inhibitor
molecular docking
synthesisandcdc25bptp1binhibitoryactivityevaluationofnovelacylhydrazonederivativescontainingcarbazolemoity
期刊论文
chinesejournaloforganicchemistry, 2019, 卷号: 39, 期号: 2, 页码: 491
作者:
Li YJ(李英俊)
;
Wang SY(王思远)
;
Jin K(靳焜)
;
Gao LX(高立信)
;
Sheng L(盛丽)
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  |  
浏览/下载:5/0
  |  
提交时间:2020/07/01
BIOLOGICAL EVALUATION
ANTITUBERCULOSIS ACTIVITY
PHOSPHATASE INHIBITORS
ANTIMICROBIAL ACTIVITY
DOCKING
OPTIMIZATION
MECHANISM
ANALOGS
DESIGN
AGENTS
acylhydrazone
carbazole
synthesis
Cdc25B and PTP1B inhibitor
molecular docking
A New Pentacyclic Ergosteroid from Fungus Aspergillus sp. SCSIO41211 Derived of Mangrove Sediment Sample
期刊论文
NATURAL PRODUCT COMMUNICATIONS, 2018, 卷号: 13, 期号: 12, 页码: 1629, 1631
作者:
Tao, Huaming
;
Li, Yunqiu
;
Lin, Xiuping
;
Zhou, Xuefeng
;
Dong, Junde
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  |  
浏览/下载:48/0
  |  
提交时间:2019/09/09
Marine-derived fungus
Aspergillus
Steroid
Mycotoxins
Antituberculosis compounds from a deep-sea-derived fungus Aspergillus sp SCSIO Ind09F01
期刊论文
NATURAL PRODUCT RESEARCH, 2017, 卷号: 31, 期号: 16, 页码: 1958-1962
作者:
Luo, XW
;
Zhou, XF
;
Lin, XP
;
Qin, XC
;
Zhang, TY
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  |  
浏览/下载:35/0
  |  
提交时间:2017/09/08
Deep sea fungi
Aspergillus sp
anti-tuberculosis
alkaloids
Enantioselective Total Syntheses of Various Amphilectane and Serrulatane Diterpenoids via Cope Rearrangements
期刊论文
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2016
Yu, Xuerong
;
Su, Fan
;
Liu, Chang
;
Yuan, Haosen
;
Zhao, Shan
;
Zhou, Zhiyao
;
Quan, Tianfei
;
Luo, Tuoping
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2017/12/03
WHIP PSEUDOPTEROGORGIA-ELISABETHAE
ENANTIOSPECIFIC TOTAL-SYNTHESIS
MARINE NATURAL-PRODUCTS
A-F AGLYCONE
SECO-PSEUDOPTEROSINS
GOLD(I)-CATALYZED CYCLIZATIONS
MYCOBACTERIUM-TUBERCULOSIS
ANTIMICROBIAL ACTIVITY
SEA
CATALYSIS
Identification of N-(2-Phenoxyethyl)imidazo[1,2-a]pyridine-3-carboxamides as New Antituberculosis Agents
期刊论文
2016, 卷号: 7, 期号: 12, 页码: 1130-1133
作者:
Wu, Zhaoyang
;
Lu, Yu
;
Li, Linhu
;
Zhao, Rui
;
Wang, Bin
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  |  
浏览/下载:3/0
  |  
提交时间:2020/01/04
Antitubercular agents
MTB H37Rv
multidrug resistant-MTB
N-(2-phenoxyethyl)imidazo[1
2-a]pyridine carboxamides
structure-activity relationship
Synthesis, spectral characterization, and antituberculosis activity of thiazino[3,2-A]benzimidazole derivatives
期刊论文
PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 2016, 卷号: 191, 期号: 7, 页码: 1036-1041
作者:
Gong, Jing-Xu
;
He, Ya
;
Cui, Zhen-Lin
;
Guo, Yue-Wei
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
Thiazino-benzimidazole derivatives
synthesis
crystal structure
anti-TB activity
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