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科研机构
上海药物研究所 [12]
内容类型
期刊论文 [12]
发表日期
2021 [4]
2020 [1]
2019 [4]
2017 [3]
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Rosmarinic Acid Suppresses Abdominal Aortic Aneurysm Progression in Apolipoprotein E-deficient Mice
期刊论文
PLANTA MEDICA, 2021, 页码: 14
作者:
Bian, Huimiao
;
Wang, Yang
;
Wu, Peng
;
Han, Na
;
Wang, Linlin
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2021/12/16
abdominal aortic aneurysm
rosmarinic acid
salvianolic acid C
salvianolic acid B
Salvia miltiorrhiza Bunge
Labiatae
Solidification of volatile D-Limonene by cyclodextrin metal-organic framework for pulmonary delivery via dry powder inhalers: In vitro and in vivo evaluation
期刊论文
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2021, 卷号: 606, 页码: 9
作者:
Zhou, Yong
;
Zhang, Meijuan
;
Wang, Caifen
;
Ren, Xiaohong
;
Guo, Tao
收藏
  |  
浏览/下载:114/0
  |  
提交时间:2021/11/04
D-Limonene
gamma-cyclodextrin metal-organic framework
Dry powder inhaler
Solidification
Aerosolization
Bioavailability
Discovery of thalidomide-based PROTAC small molecules as the highly efficient SHP2 degraders
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 218, 页码: 14
作者:
Yang, Xiangbo
;
Wang, Zhijia
;
Pei, Yuan
;
Song, Ning
;
Xu, Lei
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2021/08/17
SHP2 degradation
Proteolysis targeting chimera (PROTAC)
Thalidomide-based heterobifunctional molecules
E3 ubiquitin ligase
CRBN
Divalent tranylcypromine derivative as lysine-specific demethylase 1 inhibitor
期刊论文
MEDICINAL CHEMISTRY RESEARCH, 2021, 页码: 8
作者:
Sun, Yin
;
Li, Na
;
Su, Mingbo
;
Wang, Xiaowen
;
Zhao, Dongmei
收藏
  |  
浏览/下载:59/0
  |  
提交时间:2021/05/24
Divalent tranylcypromine
LSD1 inhibitor
MV4-11 antiproliferative activity
CD86 mRNA expression
Linker
Selectivity
SOMCL-863, a novel, selective and orally bioavailable small-molecule c-Met inhibitor, exhibits antitumor activity both in vitro and in vivo (vol 351, pg 413, 2014)
期刊论文
CANCER LETTERS, 2020, 卷号: 486, 页码: 71-72
作者:
Wang, Lu
;
Ai, Jing
;
Shen, Yanyan
;
Zhang, Haotian
;
Peng, Xia
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2020/12/24
Nanoporous CD-MOF particles with uniform and inhalable size for pulmonary delivery of budesonide
期刊论文
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2019, 卷号: 564, 页码: 153-161
作者:
Hu, Xiaoxiao
;
Wang, Caifen
;
Wang, Lebing
;
Liu, Zhaoxin
;
Wua, Li
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/07/01
gamma-Cyclodextrin metal-organic framework
Dry powder inhalation
Budesonide
Cholesterol
In vivo fluorescence imaging
Overcoming Poor Tabletability of Bulky Absorption Enhancers by Spray Drying Technology
期刊论文
JOURNAL OF PHARMACEUTICAL SCIENCES, 2019, 卷号: 108, 期号: 6, 页码: 2128-2135
作者:
Fan, Weiwei
;
Wang, Aohua
;
Wu, Yue
;
Water, Jorrit J.
;
Buckley, Stephen T.
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2020/07/01
absorption enhancers
spray drying
compaction
physicochemical properties
amorphism
tableting
Tranylcypromine and 6-trifluoroethyl thienopyrimidine hybrid as LSD1 inhibitor
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 6, 页码: 844-847
作者:
Wang, Xiaowen
;
Su, Mingbo
;
Li, You
;
Liu, Tongchao
;
Wang, Yujie
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/07/01
LSD1 inhibitor
Tranylcypromine
Menin-MLL1 protei n-protein interaction inhibitor
MV4-11 antiproliferative activity
Structure activity relationship
Stereoselective N-glycosylation with N-4-acyl cytosines and efficient synthesis of gemcitabine
期刊论文
TETRAHEDRON, 2019, 卷号: 75, 期号: 9, 页码: 1203-1213
作者:
Liu, Tongchao
;
Tang, Jiadeng
;
Liang, Jianpeng
;
Chen, Yabin
;
Wang, Xiaowen
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2020/07/01
Stereoselective
N-glycosylation
N-4-acyl cytosine
Nucleoside
Gemcitabine
Novel Inhibitors of Staphyloxanthin Virulence Factor in Comparison with Linezolid and Vancomycin versus Methicillin-Resistant, Linezolid-Resistant, and Vancomycin-Intermediate Staphylococcus aureus Infections in Vivo
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 19, 页码: 8145-8159
作者:
Ni, Shuaishuai
;
Wei, Hanwen
;
Li, Baoli
;
Chen, Feifei
;
Liu, Yifu
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
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