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广州生物医药与健康... [12]
湖南大学 [4]
重庆大学 [1]
暨南大学 [1]
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期刊论文 [18]
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2019 [4]
2016 [5]
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浏览/检索结果:
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Design, synthesis and biological evaluation of novel human monoamine oxidase B inhibitors based on a fragment in an X-ray crystal structure.
期刊论文
Bioorganic & medicinal chemistry letters, 2019
作者:
Kai Cheng
;
Shiyu Li
;
Xiao Lv
;
Yongbin Tian
;
Haiyan Kong
收藏
  |  
浏览/下载:71/0
  |  
提交时间:2019/12/13
Fragment-based drug design
Isatin
Isoform selectivity
Structure activity relationship
hMAO-B
Discovery of novel 2,3-dihydro-1H-inden-1-amine derivatives as selective monoamine oxidase B inhibitors
期刊论文
Bioorganic & Medicinal Chemistry Letters, 2019
作者:
Shiyu Li
;
Xiao Lv
;
Kai Cheng
;
Yongbing Tian
;
Xufeng Huang
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/12/13
Monoamine oxidase B
Selectivity
2,3-dihydro-1H-inden-1-amine
Structure activity relationship
Discovery of novel 2,3-dihydro-1H-inden-1-amine derivatives as selective monoamine oxidase B inhibitors.
期刊论文
Bioorganic & medicinal chemistry letters, 2019
作者:
Shiyu Li
;
Xiao Lv
;
Kai Cheng
;
Yongbing Tian
;
Xufeng Huang
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/12/13
2,3-Dihydro-1H-inden-1-amine
Monoamine oxidase B
Selectivity
Structure activity relationship
Design, synthesis and biological evaluation of novel human monoamine oxidase B inhibitors based on a fragment in an X-ray crystal structure
期刊论文
Bioorganic & Medicinal Chemistry Letters, 2019
作者:
Kai Cheng
;
Shiyu Li
;
Xiao Lv
;
Yongbin Tian
;
Haiyan Kong
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/12/17
hMAO-B
isatin
isoform
selectivity
fragment-based
drug
design
structure
activity
relationship
Selective Histone Deacetylase Inhibitors with Anticancer Activity
期刊论文
2016, 卷号: 16, 期号: [db:dc_citation_issue], 页码: 415
作者:
Ma, Nan[1,2,3]
;
Luo, Ying[4]
;
Wang, Ying[2]
;
Liao, Chenzhong[4]
;
Ye, Wen-Cai[2,3]
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/03
Selective Histone Deacetylase Inhibitors with Anticancer Activity
期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2016, 卷号: 16, 期号: 4, 页码: 415-426
作者:
Luo, Ying
;
Ma, Nan
;
Ye, Wen-Cai
;
Liao, Chenzhong
;
Wang, Ying
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2018/12/13
Structure-Based Design of Potent Nicotinamide Phosphoribosyltransferase Inhibitors with Promising in Vitro and in Vivo Antitumor Activities
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5766-5779
作者:
Jiang, Sheng
;
Li, Zheng
;
Qin, Dongguang
;
Qiu, Yatao
;
Chen, Jiaxuan
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2018/12/13
Selective Histone Deacetylase Inhibitors with Anticancer Activity
期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2016, 卷号: 16, 期号: 4, 页码: 415-426
Ma, Nan
;
Luo, Ying
;
Wang, Ying
;
Liao, Chenzhong
;
Ye, Wen-Cai
;
Jiang, Sheng
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2016/12/16
Structure-Based Design of Potent Nicotinamide Phosphoribosyltransferase Inhibitors with Promising in Vitro and in Vivo Antitumor Activities
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5766-5779
Bai, Jinhong
;
Liao, Chenzhong
;
Liu, Yanghan
;
Qin, Xiaochu
;
Chen, Jiaxuan
;
Qiu, Yatao
;
Qin, Dongguang
;
Li, Zheng
;
Tu, Zheng-Chao
;
Jiang, Sheng
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2016/12/16
Discovery of Novel Class I Histone Deacetylase Inhibitors with Promising in Vitro and in Vivo Antitumor Activities
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 19, 页码: 7672-7680
作者:
Li, Zheng
;
Jiang, Sheng
;
Li, Shang
;
Wang, Zhen
;
Liao, Chenzhong
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2018/12/13
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