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科研机构
上海药物研究所 [7]
海洋研究所 [3]
上海大学 [2]
中国医学科学院 北京... [1]
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期刊论文 [13]
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2021 [1]
2020 [5]
2019 [2]
2018 [4]
2017 [1]
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Discovery of High-Affinity Inhibitors of the BPTF Bromodomain
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12075-12088
作者:
Lu, Tian
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浏览/下载:38/0
  |  
提交时间:2021/11/04
Chromosome-level genome assembly of Paralithodes platypus provides insights into evolution and adaptation of king crabs
期刊论文
MOLECULAR ECOLOGY RESOURCES, 2020, 页码: 15
作者:
Tang, Boping
;
Wang, Zhongkai
;
Liu, Qiuning
;
Wang, Zhengfei
;
Ren, Yandong
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  |  
浏览/下载:104/0
  |  
提交时间:2021/04/12
adaptation
blue king crab
evolution
genome
Discovery of 8-Methyl-pyrrolo[1,2-a]pyrazin-1(2H)-one Derivatives as Highly Potent and Selective Bromodomain and Extra-Terminal (BET) Bromodomain Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 8, 页码: 3956-3975
作者:
Li, Zizhou
;
Xiao, Senhao
;
Yang, Yaxi
;
Chen, Chao
;
Lu, Tian
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  |  
浏览/下载:28/0
  |  
提交时间:2020/07/01
High-Quality Genome Assembly of Eriocheir japonica sinensis Reveals Its Unique Genome Evolution
期刊论文
FRONTIERS IN GENETICS, 2020, 卷号: 10, 页码: 9
作者:
Tang, Boping
;
Wang, Zhongkai
;
Liu, Qiuning
;
Zhang, Huabin
;
Jiang, Senhao
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  |  
浏览/下载:81/0
  |  
提交时间:2020/09/21
Eriocheir japonica sinensis
evolution
nanopore
crab
genome assembly and annotation
Chromosome-level genome assembly reveals the unique genome evolution of the swimming crab (Portunus trituberculatus)
期刊论文
GIGASCIENCE, 2020, 卷号: 9, 期号: 1, 页码: 10
作者:
Tang, Boping
;
Zhang, Daizhen
;
Li, Haorong
;
Jiang, Senhao
;
Zhang, Huabin
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  |  
浏览/下载:90/0
  |  
提交时间:2020/09/23
Portunus trituberculatus
genome assembly
crab
chromosome
evolution
discoveryofnovelcbpbromodomaininhibitorsthroughtrfretbasedhighthroughputscreening
期刊论文
actapharmacologicasinica, 2020, 卷号: 41, 期号: 2, 页码: 285
作者:
Zhang Fengcai
;
Sun Zhongya
;
Liao Liping
;
Zuo Yu
;
Zhang Dan
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  |  
浏览/下载:35/0
  |  
提交时间:2020/07/01
CBP bromodomain
small-molecule inhibitor
high-throughput screening
TR-FRET
molecular modeling
human leukemia MV4-11 cells
Discovery of alkoxy benzamide derivatives as novel BPTF bromodomain inhibitors via structure-based virtual screening
期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 86, 页码: 494-500
作者:
Zhang, Dan
;
Han, Jie
;
Lu, Wenchao
;
Lian, Fulin
;
Wang, Jun
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  |  
浏览/下载:11/0
  |  
提交时间:2020/07/01
Lysine acetylation
Bromodomain
Virtual screening
BPTF inhibitor
Discovery of alkoxy benzamide derivatives as novel BPTF bromodomain inhibitors via structure-based virtual screening
期刊论文
Bioorganic chemistry, 2019, 卷号: 86, 页码: 494-500
作者:
Zhang Dan[1]
;
Han Jie[2]
;
Lu Wenchao[3]
;
Lian Fulin[4]
;
Wang Jun[5]
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  |  
浏览/下载:33/0
  |  
提交时间:2019/04/22
BPTF inhibitor
Bromodomain
Lysine acetylation
Virtual screening
Discovery and biological evaluation of thiobarbituric derivatives as potent p300/CBP inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 20, 页码: 5397-5407
作者:
Lu, Wenchao
;
Xiong, Huan
;
Chen, Yu
;
Wang, Chen
;
Zhang, Hao
收藏
  |  
浏览/下载:138/0
  |  
提交时间:2019/01/08
Drug discovery
Epigenetics
Histone acetyltransferase
P300/CBP
Design, synthesis and biological evaluation of benzo[cd]indo1-2(1H)-ones derivatives as BRD4 inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 264-273
作者:
Feng, Yuxin
;
Xiao, Senhao
;
Chen, Yantao
;
Jiang, Hao
;
Liu, Na
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2019/01/08
Benzo[cd]indol-2(1H)-one
Sulfonamide
BRD4 inhibitor
Bromodomain and extra-terminal domain
Acetyl-lysine binding pocket
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