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上海药物研究所 [6]
西安交通大学 [3]
山东大学 [2]
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湖南大学 [2]
厦门大学 [1]
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期刊论文 [24]
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Nosiheptide analogues as potential antibacterial agents via dehydroalanine region modifications: Semi-synthesis, antimicrobial activity and molecular docking study
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 31, 页码: 10
作者:
Fan, Yafei
;
Chen, Hangfei
;
Mu, Ning
;
Wang, Wengui
;
Zhu, Kongkai
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2021/05/24
Nosiheptide analogues
Semi-synthesis
Antimicrobial activity
Molecular docking
TSL-1502, a glucuronide prodrug of a poly (ADP-ribose) polymerase (PARP) inhibitor, exhibits potent anti-tumor activity in preclinical models
期刊论文
AMERICAN JOURNAL OF CANCER RESEARCH, 2021, 卷号: 11, 期号: 4, 页码: 1632-1645
作者:
Wang, Lei
;
Zhu, Xi
;
Li, Lili
;
Li, Lin
;
Fu, Li
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  |  
浏览/下载:74/0
  |  
提交时间:2021/06/11
PARP
DNA damage
hematologic toxicity
beta-glucuronidase
tumor selectivity
Mutant p53 in cancer therapy-the barrier or the path
期刊论文
JOURNAL OF MOLECULAR CELL BIOLOGY, 2019, 卷号: 11, 期号: 4
作者:
Zhou, Xiang
;
Hao, Qian
;
Lu, Hua
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  |  
浏览/下载:4/0
  |  
提交时间:2019/12/05
mutant p53
gain-of-function
cancer therapy
chemoresistance
synthetic lethality
Identification of synthetic lethality based on a functional network by using machine learning algorithms
期刊论文
JOURNAL OF CELLULAR BIOCHEMISTRY, 2019, 卷号: 120, 页码: 405-416
作者:
Li, JiaRui[1]
;
Lu, Lin[2]
;
Zhang, Yu-Hang[3]
;
Liu, Min[4]
;
Chen, Lei[5]
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  |  
浏览/下载:22/0
  |  
提交时间:2019/04/22
maximum relevance and minimum redundancy (mRMR)
random forest (RF)
synthetic lethality
Identification of synthetic lethality based on a functional network by using machine learning algorithms
期刊论文
JOURNAL OF CELLULAR BIOCHEMISTRY, 2019, 卷号: Vol.120 No.1, 页码: 405-416
作者:
Li, JiaRui
;
Lu, Lin
;
Zhang, Yu-Hang
;
Liu, Min
;
Chen, Lei
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/12/17
maximum relevance and minimum redundancy (mRMR)
random forest (RF)
synthetic lethality
Lipid-Based Liquid Crystalline Nanoparticles Facilitate Cytosolic Delivery of siRNA via Structural Transformation
期刊论文
NANO LETTERS, 2018, 卷号: 18, 期号: 4, 页码: 2411-2419
作者:
He, Shufang
;
Fan, Weiwei
;
Wu, Na
;
Zhu, Jingjing
;
Miao, Yunqiu
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
Lipids
liquid crystalline nanoparticles
siRNA delivery
endosomal escape
synthetic lethality
Facilitating Anti-Cancer Combinatorial Drug Discovery by Targeting Epistatic Disease Genes
期刊论文
Molecules (Basel, Switzerland), 2018, 卷号: 23, 期号: 4
作者:
Quan, Yuan
;
Liu, Meng-Yuan
;
Liu, Ye-Mao
;
Zhu, Li-Da
;
Wu, Yu-Shan
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  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
Targeting death receptors for drug-resistant cancer therapy: Codelivery of pTRAIL and monensin using dual-targeting and stimuli-responsive self-assembling nanocomposites
期刊论文
BIOMATERIALS, 2018, 卷号: 158, 页码: 56-73
作者:
Xu, Fan
;
Zhong, Huihai
;
Chang, Ya
;
Li, Dongdong
;
Jin, Hongyue
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  |  
浏览/下载:49/0
  |  
提交时间:2019/01/08
TRAIL
Gene delivery
Monensin
Poly-gamma-glutamic acid
Death receptor
Drug resistance
Compound F779-0434 causes synthetic lethality in BRCA2-deficient cancer cells by disrupting RAD52–ssDNA association
期刊论文
RSC Advances, 2018, 卷号: Vol.8 No.34, 页码: 18859-18869
作者:
Li, J
;
Yang, QY
;
Zhang, Y
;
Huang, KJ
;
Sun, R
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/02/28
Novel PARP1/2 inhibitor mefuparib hydrochloride elicits potent in vitro and in vivo anticancer activity, characteristic of high tissue distribution
期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 3, 页码: 4156-4168
作者:
He, Jin-Xue
;
Wang, Meng
;
Huan, Xia-Juan
;
Chen, Chuan-Huizi
;
Song, Shan-Shan
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  |  
浏览/下载:35/0
  |  
提交时间:2019/01/08
MPH
PARP inhibitor
homologous recombination
antitumor activity
synthetic lethality
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