CORC

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Identification of methyl (5-(6-((4-(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinopyrrolo[2,1-f][1,2,4]triazin-2-yl)-4-(trifluoromethyl)pyridin-2-yl)carbamate (CYH33) as an orally bioavailable, highly potent, PI3K alpha inhibitor for the treatment of advanced solid tumors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 209, 页码: 10
作者:  Xiang, Hao-Yue;  Wang, Xiang;  Chen, Yan-Hong;  Zhang, Xi;  Tan, Cun
收藏  |  浏览/下载:33/0  |  提交时间:2021/05/24
Synthesis and Cytotoxic Activity of Novel C-23-Modified Asiatic Acid Derivatives 期刊论文
MOLECULES, 2020, 卷号: 25, 期号: 16, 页码: 20
作者:  Lu, Yi-hong;  Chen, Ming-cang;  Liu, Fang;  Xu, Zhou;  Tian, Xiao-ting
收藏  |  浏览/下载:13/0  |  提交时间:2020/12/24
The iron chelator desferrioxamine synergizes with chemotherapy for cancer treatment 期刊论文
JOURNAL OF TRACE ELEMENTS IN MEDICINE AND BIOLOGY, 2019, 卷号: 56, 页码: 131-138
作者:  Wang, Lingjuan;  Li, Xiaoqing;  Mu, Yanxi;  Lu, Chang;  Tang, Shiqian
收藏  |  浏览/下载:30/0  |  提交时间:2020/09/09
Discovery of 3,4,6-Trisubstituted Piperidine Derivatives as Orally Active, Low hERG Blocking Akt Inhibitors via Conformational Restriction and Structure-Based Design 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 15, 页码: 7264-7288
作者:  Dong, Xiaowu;  Zhan, Wenhu;  Zhao, Mengting;  Che, Jinxin;  Dai, Xiaoyang
收藏  |  浏览/下载:30/0  |  提交时间:2020/07/01
Impact and underlying mechanisms of miR-1271 on cisplatin resistance in the human ovarian cancer cell line SKOV3/DDP 期刊论文
INTERNATIONAL JOURNAL OF CLINICAL AND EXPERIMENTAL MEDICINE, 2019, 卷号: 12, 期号: 2, 页码: 1577-1583
作者:  Lu, Jie[1];  Wang, Guangzhou[2];  Li, Jilin[3];  Wang, Jinfu[4];  Mao, Lingxiang[5]
收藏  |  浏览/下载:14/0  |  提交时间:2019/12/24
Targeting slug-mediated non-canonical activation of c-Met to overcome chemo-resistance in metastatic ovarian cancer cells 期刊论文
ACTA PHARMACEUTICA SINICA B, 2019, 卷号: 9
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收藏  |  浏览/下载:5/0  |  提交时间:2020/10/26
Robust anticancer efficacy of a biologically synthesized tumor acidity-responsive and autophagy-inducing functional beclin 1 期刊论文
Acs applied materials & interfaces, 2018, 卷号: 10, 期号: 6, 页码: 5227-5239
作者:  Ding, Guo-Bin;  Sun, Junqing;  Wu, Gengfeng;  Li, Binchun;  Yang, Peng
收藏  |  浏览/下载:39/0  |  提交时间:2019/04/23
Design, synthesis, biological evaluation and cocrystal structures with tubulin of chiral beta-lactam bridged combretastatin A-4 analogues as potent antitumor agents 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 144, 页码: 817-842
作者:  Zhou, Pengfei;  Liang, Yuru;  Zhang, Hao;  Jiang, Hao;  Feng, Kechang
收藏  |  浏览/下载:16/0  |  提交时间:2019/01/08
ER alpha and ER beta oppositely regulated plexin B1 expression and migration of ovarian cancer SKOV-3 cells 期刊论文
INTERNATIONAL JOURNAL OF CLINICAL AND EXPERIMENTAL MEDICINE, 2018, 卷号: 11, 期号: 4
作者:  Liu, Yang;  Sun, Chunyi;  Mo, Yuxia;  Liu, Huijin;  Zhai, Shujuan
收藏  |  浏览/下载:6/0  |  提交时间:2019/12/04
Effects of isoliquiritigenin on ovarian cancer cells. 期刊论文
Onco Targets Ther, 2018, 卷号: Vol.11, 页码: 1633-1642
作者:  Li N;  Yang L;  Deng X;  Sun Y.
收藏  |  浏览/下载:3/0  |  提交时间:2019/03/26


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