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山东大学 [12]
上海药物研究所 [11]
长春应用化学研究所 [11]
化学研究所 [9]
重庆大学 [5]
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Identification of methyl (5-(6-((4-(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinopyrrolo[2,1-f][1,2,4]triazin-2-yl)-4-(trifluoromethyl)pyridin-2-yl)carbamate (CYH33) as an orally bioavailable, highly potent, PI3K alpha inhibitor for the treatment of advanced solid tumors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 209, 页码: 10
作者:
Xiang, Hao-Yue
;
Wang, Xiang
;
Chen, Yan-Hong
;
Zhang, Xi
;
Tan, Cun
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2021/05/24
PI3K
Pyrrolo[2,1-f][1,2,4]triazine
Anti-cancer
Target therapy
Synthesis and Cytotoxic Activity of Novel C-23-Modified Asiatic Acid Derivatives
期刊论文
MOLECULES, 2020, 卷号: 25, 期号: 16, 页码: 20
作者:
Lu, Yi-hong
;
Chen, Ming-cang
;
Liu, Fang
;
Xu, Zhou
;
Tian, Xiao-ting
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  |  
浏览/下载:13/0
  |  
提交时间:2020/12/24
asiatic acid
modification at C-23
intramolecular hydrogen bonding
cytotoxic activity
The iron chelator desferrioxamine synergizes with chemotherapy for cancer treatment
期刊论文
JOURNAL OF TRACE ELEMENTS IN MEDICINE AND BIOLOGY, 2019, 卷号: 56, 页码: 131-138
作者:
Wang, Lingjuan
;
Li, Xiaoqing
;
Mu, Yanxi
;
Lu, Chang
;
Tang, Shiqian
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  |  
浏览/下载:30/0
  |  
提交时间:2020/09/09
Ovarian cancer
DFO
CDDP
Cancer therapy
Discovery of 3,4,6-Trisubstituted Piperidine Derivatives as Orally Active, Low hERG Blocking Akt Inhibitors via Conformational Restriction and Structure-Based Design
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 15, 页码: 7264-7288
作者:
Dong, Xiaowu
;
Zhan, Wenhu
;
Zhao, Mengting
;
Che, Jinxin
;
Dai, Xiaoyang
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  |  
浏览/下载:30/0
  |  
提交时间:2020/07/01
Impact and underlying mechanisms of miR-1271 on cisplatin resistance in the human ovarian cancer cell line SKOV3/DDP
期刊论文
INTERNATIONAL JOURNAL OF CLINICAL AND EXPERIMENTAL MEDICINE, 2019, 卷号: 12, 期号: 2, 页码: 1577-1583
作者:
Lu, Jie[1]
;
Wang, Guangzhou[2]
;
Li, Jilin[3]
;
Wang, Jinfu[4]
;
Mao, Lingxiang[5]
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/12/24
miR-1271
XIAP
cisplatin resistance
ovarian cancer
SKOV3/DDP cells
Targeting slug-mediated non-canonical activation of c-Met to overcome chemo-resistance in metastatic ovarian cancer cells
期刊论文
ACTA PHARMACEUTICA SINICA B, 2019, 卷号: 9
-
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  |  
浏览/下载:5/0
  |  
提交时间:2020/10/26
EPITHELIAL-MESENCHYMAL TRANSITION
TUMOR-GROWTH
HETEROGENEITY
AMPLIFICATION
CONTRIBUTES
PROGRESSION
CARCINOMA
REVEALS
PATHWAY
SNAIL
Slug
c-Met
Drug resistance
Ovarian cancer
XL184
Robust anticancer efficacy of a biologically synthesized tumor acidity-responsive and autophagy-inducing functional beclin 1
期刊论文
Acs applied materials & interfaces, 2018, 卷号: 10, 期号: 6, 页码: 5227-5239
作者:
Ding, Guo-Bin
;
Sun, Junqing
;
Wu, Gengfeng
;
Li, Binchun
;
Yang, Peng
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  |  
浏览/下载:39/0
  |  
提交时间:2019/04/23
Functional beclin 1
Phlip
Biological synthesis
Autophagy induction
Anticancer efficacy
Design, synthesis, biological evaluation and cocrystal structures with tubulin of chiral beta-lactam bridged combretastatin A-4 analogues as potent antitumor agents
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 144, 页码: 817-842
作者:
Zhou, Pengfei
;
Liang, Yuru
;
Zhang, Hao
;
Jiang, Hao
;
Feng, Kechang
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
1,4-Diaryl-2-azetidinone
Combretastatin A-4
Tubulin polymerization
Antitumor
ER alpha and ER beta oppositely regulated plexin B1 expression and migration of ovarian cancer SKOV-3 cells
期刊论文
INTERNATIONAL JOURNAL OF CLINICAL AND EXPERIMENTAL MEDICINE, 2018, 卷号: 11, 期号: 4
作者:
Liu, Yang
;
Sun, Chunyi
;
Mo, Yuxia
;
Liu, Huijin
;
Zhai, Shujuan
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/12/04
Plexin B1
ER alpha
ER beta
ovarian cancer
cell migration
Effects of isoliquiritigenin on ovarian cancer cells.
期刊论文
Onco Targets Ther, 2018, 卷号: Vol.11, 页码: 1633-1642
作者:
Li N
;
Yang L
;
Deng X
;
Sun Y.
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  |  
浏览/下载:3/0
  |  
提交时间:2019/03/26
OVCAR3
PI3K/Akt/mTOR
pathway
SKOV3
apoptosis
isoliquiritigenin
(ILQ)
ovarian
cancer
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