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Allosteric Modulation: Dynamics is Double-"E"dged 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 7, 页码: 3694-3696
作者:  Xiong, Bing
收藏  |  浏览/下载:15/0  |  提交时间:2021/06/11
The cross-talk between methylation and phosphorylation in lymphoid-specific helicase drives cancer stem-like properties 期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2020, 卷号: 5, 期号: 1, 页码: 14
作者:  Liu, Na;  Yang, Rui;  Shi, Ying;  Chen, Ling;  Liu, Yating
收藏  |  浏览/下载:33/0  |  提交时间:2020/12/21
Rational Design, synthesis and biological evaluation of novel triazole derivatives as potent and selective PRMT5 inhibitors with antitumor activity 期刊论文
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2019, 卷号: 33, 期号: 8, 页码: 775-785
作者:  Zhu, Kongkai;  Shao, Jingwei;  Tao, Hongrui;  Yan, Xue;  Luo, Cheng
收藏  |  浏览/下载:12/0  |  提交时间:2020/07/01
Discovery of Novel PRMT5 Inhibitors by Virtual Screening and Biological Evaluations 期刊论文
CHEMICAL & PHARMACEUTICAL BULLETIN, 2019, 卷号: 67, 期号: 4, 页码: 382-388
作者:  Tao, Hongrui;  Yan, Xue;  Zhu, Kongkai;  Zhang, Hua
收藏  |  浏览/下载:14/0  |  提交时间:2020/07/01
Discovery of 2-substituted-N-(3-(3,4-dihydroisoquinolin-2(1H)-yl)-2-hydroxypropyl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide as potent and selective protein arginine methyltransferases 5 inhibitors: Design, synthesis and biological evaluation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 164, 页码: 317-333
作者:  Shao, Jingwei;  Zhu, Kongkai;  Du, Daohai;  Zhang, Yuanyuan;  Tao, Hongrui
收藏  |  浏览/下载:35/0  |  提交时间:2020/07/01
A patent review of arginine methyltransferase inhibitors (2010-2018) 期刊论文
EXPERT OPINION ON THERAPEUTIC PATENTS, 2019, 卷号: 29, 期号: 2, 页码: 97-114
作者:  Li, Xiao;  Wang, Chen;  Jiang, Hao;  Luo, Cheng
收藏  |  浏览/下载:8/0  |  提交时间:2020/07/01
Low expression of PRMT5 in peripheral blood may serve as a potential independent risk factor in assessments of the risk of stable CAD and AMI 期刊论文
BMC CARDIOVASCULAR DISORDERS, 2019, 卷号: 19
作者:  Tan, Buchuan;  Liu, Qian;  Yang, Liping;  Yang, Yushuang;  Liu, Dongna
收藏  |  浏览/下载:21/0  |  提交时间:2019/12/05
PRMT5 enhances tumorigenicity and glycolysis in pancreatic cancer via the FBW7/cMyc axis 期刊论文
CELL COMMUNICATION AND SIGNALING, 2019, 卷号: 17
作者:  Qin, Yi;  Hu, Qiangsheng;  Xu, Jin;  Ji, Shunrong;  Dai, Weixing
收藏  |  浏览/下载:29/0  |  提交时间:2019/12/05
MiR-1266 suppresses the growth and metastasis of prostate cancer via targeting PRMT5 期刊论文
EUROPEAN REVIEW FOR MEDICAL AND PHARMACOLOGICAL SCIENCES, 2019, 卷号: 23, 期号: 15
作者:  Sun, C-M;  Zhang, G-M;  Qian, H-N;  Cheng, S-J;  Wang, M.
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/05
UHRF1 suppresses retrotransposons and cooperates with PRMT5 and PIWI proteins in male germ cells 期刊论文
NATURE COMMUNICATIONS, 2019, 卷号: 10
作者:  Dong, Juan;  Wang, Xiaoli;  Cao, Congcong;  Wen, Yujiao;  Sakashita, Akihiko
收藏  |  浏览/下载:45/0  |  提交时间:2019/12/05


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