×
验证码:
换一张
忘记密码?
记住我
CORC
首页
科研机构
检索
知识图谱
申请加入
托管服务
登录
注册
在结果中检索
科研机构
上海药物研究所 [11]
昆明植物研究所 [2]
厦门大学 [1]
上海大学 [1]
上海中医药大学 [1]
昆明医科大学 [1]
更多...
内容类型
期刊论文 [17]
学位论文 [1]
发表日期
2021 [1]
2019 [3]
2018 [3]
2017 [3]
2016 [1]
2015 [1]
更多...
学科主题
Chemistry,... [1]
Pharmacolo... [1]
Plant Scie... [1]
×
知识图谱
CORC
开始提交
已提交作品
待认领作品
已认领作品
未提交全文
收藏管理
QQ客服
官方微博
反馈留言
浏览/检索结果:
共18条,第1-10条
帮助
已选(
0
)
清除
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
作者升序
作者降序
题名升序
题名降序
发表日期升序
发表日期降序
提交时间升序
提交时间降序
Targeting Protein Neddylation to Inactivate Cullin-RING Ligases by Gossypol: A Lucky Hit or a New Start?
期刊论文
DRUG DESIGN DEVELOPMENT AND THERAPY, 2021, 卷号: 15
作者:
Yu, Qing
;
Sun, Yi
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/03/15
anti-cancer drug
cullin-RING E3 ligases
natural product
high-throughput screen
neddylation
small-molecule inhibitors
Orthogonal assays for the identification of inhibitors of the single-stranded nucleic acid binding protein YB-1
期刊论文
ACTA PHARMACEUTICA SINICA B, 2019, 卷号: 9, 期号: 5, 页码: 997-1007
作者:
Trevarton, Alexander J.
;
Zhou, Yan
;
Yang, Dehua
;
Rewcastle, Gordon W.
;
Flanagan, Jack U.
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/07/01
Cancer
YB-1
Luciferase
AlphaScreen
Transcription factor
Single-stranded DNA
Discovery of trisubstituted nicotinonitrile derivatives as novel human GCN5 inhibitors through AlphaScreen-based high throughput screening
期刊论文
RSC ADVANCES, 2019, 卷号: 9, 期号: 9, 页码: 4917-4924
作者:
Tao, Hongru
;
Wang, Jun
;
Lu, Wenchao
;
Zhang, Rukang
;
Xie, Yiqian
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2020/07/01
Discovery of trisubstituted nicotinonitrile derivatives as novel human GCN5 inhibitors through AlphaScreen-based high throughput screening
期刊论文
RSC ADVANCES, 2019, 卷号: 9, 页码: 4917-4924
作者:
Tao, Hongru[1]
;
Wang, Jun[2]
;
Lu, Wenchao[3]
;
Zhang, Rukang[4]
;
Xie, Yiqian[5]
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/04/22
Identification of small molecule inhibitors targeting the SMARCA2 bromodomain from a high-throughput screening assay
期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 9, 页码: 1544-1552
作者:
Lu, Tian
;
Hu, Jun-chi
;
Lu, Wen-chao
;
Han, Jie
;
Ding, Hong
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2019/01/08
AlphaScreen
high-throughput screening
SMARCA2
bromodomain
small molecule inhibitor
Design, synthesis and biological evaluation of benzo[cd]indo1-2(1H)-ones derivatives as BRD4 inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 264-273
作者:
Feng, Yuxin
;
Xiao, Senhao
;
Chen, Yantao
;
Jiang, Hao
;
Liu, Na
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2019/01/08
Benzo[cd]indol-2(1H)-one
Sulfonamide
BRD4 inhibitor
Bromodomain and extra-terminal domain
Acetyl-lysine binding pocket
A Highly Sensitive Non-Radioactive Activity Assay for AMP-Activated Protein Kinase (AMPK)
期刊论文
Methods and protocols, 2018, 卷号: 1, 期号: 1
作者:
Yan, Yan
;
Gu, Xin
;
Xu, H Eric
;
Melcher, Karsten
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
Discovery of novel trimethoxy-ring BRD4 bromodomain inhibitors: AlphaScreen assay, crystallography and cell-based assay
期刊论文
MEDCHEMCOMM, 2017, 卷号: 8, 期号: 6, 页码: 1322-1331
作者:
Chen, Zhifeng
;
Zhang, Hao
;
Liu, Shien
;
Xie, Yiqian
;
Jiang, Hao
收藏
  |  
浏览/下载:90/0
  |  
提交时间:2019/01/08
Discovery of novel BRD4 inhibitors by high-throughput screening, crystallography, and cell-based assays
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 9, 页码: 2003-2009
作者:
Sun, Zhongya
;
Zhang, Hao
;
Chen, Zhifeng
;
Xie, Yiqian
;
Jiang, Hao
收藏
  |  
浏览/下载:89/0
  |  
提交时间:2019/01/08
BRD4 inhibitor
High-throughput screening
Crystallography
Discovery of novel trimethoxy-ring BRD4 bromodomain inhibitors: AlphaScreen assay, crystallography and cell-based assay
期刊论文
MEDCHEMCOMM, 2017, 卷号: 8, 期号: 6
作者:
Chen, Zhifeng
;
Zhang, Hao
;
Liu, Shien
;
Xie, Yiqian
;
Jiang, Hao
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/05
©版权所有 ©2017 CSpace - Powered by
CSpace