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上海药物研究所 [7]
新疆天文台 [4]
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期刊论文 [37]
发表日期
2020 [37]
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天文学 [4]
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A Middle Eocene lowland humid subtropical "Shangri-La" ecosystem in central Tibet
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2020, 卷号: 117, 期号: 52, 页码: 32989-32995
作者:
Su, Tao
;
Spicer, Robert A.
;
Wu, Fei-Xiang
;
Farnsworth, Alexander
;
Huang, Jian
收藏
  |  
浏览/下载:56/0
  |  
提交时间:2021/09/17
biodiversity
fossil
monsoon
Tibetan Plateau
topography
Identification of SARS-CoV-2 entry inhibitors among already approved drugs
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 7
作者:
Yang, Li
;
Pei, Rong-juan
;
Li, Heng
;
Ma, Xin-na
;
Zhou, Yu
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  |  
浏览/下载:42/0
  |  
提交时间:2020/12/24
COVID-19
SARS-CoV-2
virus entry inhibitors
high throughput screening assay
approved drug library
histamine receptor antagonists
clemastine
Structure-based design, synthesis and bioactivity evaluation of macrocyclic inhibitors of mutant isocitrate dehydrogenase 2 (IDH2) displaying activity in acute myeloid leukemia cells
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 19
作者:
Che, Jinxin
;
Huang, Feng
;
Zhang, Mengmeng
;
Xu, Gaoya
;
Qu, Bingxue
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  |  
浏览/下载:21/0
  |  
提交时间:2020/12/21
Metabolic pathways
Isocitrate dehydrogenase 2
Conformational restriction
Macrocyclic derivatives
Inhibitors
Structure-based design, synthesis and bioactivity evaluation of macrocyclic inhibitors of mutant isocitrate dehydrogenase 2 (IDH2) displaying activity in acute myeloid leukemia cells
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 19
作者:
Che, Jinxin
;
Huang, Feng
;
Zhang, Mengmeng
;
Xu, Gaoya
;
Qu, Bingxue
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/12/21
Metabolic pathways
Isocitrate dehydrogenase 2
Conformational restriction
Macrocyclic derivatives
Inhibitors
Multi-feature weighting neighborhood density clustering
期刊论文
NEURAL COMPUTING & APPLICATIONS, 2020, 卷号: 32, 期号: 13, 页码: 9545-9565
作者:
Xu, Shuliang
;
Feng, Lin
;
Liu, Shenglan
;
Zhou, Jian
;
Qiao, Hong
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  |  
浏览/下载:13/0
  |  
提交时间:2020/08/03
Clustering analysis
Multi-feature
Neighborhood density
Rough set
Granular computing
DC591017, a phosphodiesterase-4 (PDE4) inhibitor with robust anti-inflammation through regulating PKA-CREB signaling
期刊论文
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 177, 页码: 15
作者:
Li, Heng
;
Li, Jian
;
Zhang, Xianglei
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  |  
浏览/下载:28/0
  |  
提交时间:2020/12/24
DC591017
PDE4
Inflammation
Macrophages
Dendritic cells
Psoriasis
DC591017, a phosphodiesterase-4 (PDE4) inhibitor with robust anti-inflammation through regulating PKA-CREB signaling
期刊论文
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 177, 页码: 15
作者:
Li, Heng
;
Li, Jian
;
Zhang, Xianglei
;
Feng, Chunlan
;
Fan, Chen
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  |  
浏览/下载:40/0
  |  
提交时间:2020/12/24
DC591017
PDE4
Inflammation
Macrophages
Dendritic cells
Psoriasis
Safety, Clinical Activity, and Pharmacokinetics of Al flutinib (AST2818) in Patients With Advanced NSCLC With EGFR T790M Mutation
期刊论文
JOURNAL OF THORACIC ONCOLOGY, 2020, 卷号: 15, 期号: 6, 页码: 1015-1026
作者:
Shi, Yuankai
;
Zhang, Shucai
;
Hu, Xingsheng
;
Feng, Jifeng
;
Ma, Zhiyong
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  |  
浏览/下载:37/0
  |  
提交时间:2020/12/24
Alflutinib
NSCLC
EGFR T790M mutation
Efficacy
Safety
Data processing and data products from 2017 to 2019 campaign of astronomical site testing at Ali, Daocheng and Muztagh-ata
期刊论文
RESEARCH IN ASTRONOMY AND ASTROPHYSICS, 2020, 卷号: 20, 期号: 6, 页码: 82
作者:
Cao, Zi-Huang
;
Hao, Jin-Xin
;
Feng, Lu
;
Jones, Hugh R. A.
;
Li, Jian
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  |  
浏览/下载:74/0
  |  
提交时间:2021/04/01
LOT
Site-selection
data processing
Site-testing at Muztagh-ata site I: ground meteorology and sky brightness
期刊论文
RESEARCH IN ASTRONOMY AND ASTROPHYSICS, 2020, 卷号: 20, 期号: 6, 页码: 86
作者:
Xu, Jing
;
Esamdin, Ali
;
Hao, Jin-Xin
;
Bai, Jin-Min
;
Yang, Ji
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  |  
浏览/下载:22/0
  |  
提交时间:2021/04/01
site-testing
meteorological condition
optical observing
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