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科研机构
上海药物研究所 [11]
内容类型
期刊论文 [11]
发表日期
2020 [11]
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发表日期:2020
专题:上海药物研究所
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Identify potent SARS-CoV-2 main protease inhibitors via accelerated free energy perturbation-based virtual screening of existing drugs
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2020, 卷号: 117, 期号: 44, 页码: 27381-27387
作者:
Li, Zhe
;
Li, Xin
;
Huang, Yi-You
;
Wu, Yaoxing
;
Liu, Runduo
收藏
  |  
浏览/下载:75/0
  |  
提交时间:2020/12/24
virtual screening
SARS-CoV-2
drug repurposing
free energy perturbation
main protease
Light-induced primary amines and o-nitrobenzyl alcohols cyclization as a versatile photoclick reaction for modular conjugation
期刊论文
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 13
作者:
Guo, An-Di
;
Wei, Dan
;
Nie, Hui-Jun
;
Hu, Hao
;
Peng, Chengyuan
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2020/12/24
Supramolecular Assembly of TPE-Based Glycoclusters with Dicyanomethylene-4H-pyran (DM) Fluorescent Probes Improve Their Properties for Peroxynitrite Sensing and Cell Imaging
期刊论文
CHEMISTRY-A EUROPEAN JOURNAL, 2020, 页码: 9
作者:
Dong, Lei
;
Fu, Mengqi
;
Liu, Lifang
;
Han, Hai-Hao
;
Zang, Yi
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2020/12/21
cell imaging
glycoclusters
peroxynitrite detection
self-assembly
tetraphenylethylene
Selective Inhibition of STRN3-Containing PP2A Phosphatase Restores Hippo Tumor-Suppressor Activity in Gastric Cancer
期刊论文
CANCER CELL, 2020, 卷号: 38, 期号: 1, 页码: 115-+
作者:
Tang, Yang
;
Fang, Gemin
;
Guo, Fenghua
;
Zhang, Hui
;
Chen, Xiaoxu
收藏
  |  
浏览/下载:95/0
  |  
提交时间:2020/12/24
Active constituents and mechanisms of Respiratory Detox Shot, a traditional Chinese medicine prescription, for COVID-19 control and prevention: Network -molecular docking-LC-MSE analysis
期刊论文
JOURNAL OF INTEGRATIVE MEDICINE-JIM, 2020, 卷号: 18, 期号: 3, 页码: 229-241
作者:
Zhang, Zi-jia
;
Wu, Wen-yong
;
Hou, Jin-jun
;
Zhang, Lin-lin
;
Li, Fei-fei
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2020/07/01
Lung-toxin Dispelling Formula No. 1
COVID-19
3C-like protease
Network pharmacology
Molecular docking
Meridian tropism
Quantitative analysis of fourteen bufadienolides in Venenum Bufonis crude drug and its Chinese patent medicines by ultra-high performance liquid chromatography coupled with tandem mass spectrometry
期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2020, 卷号: 251, 页码: 8
作者:
Wei, Wen-long
;
An, Ya-ling
;
Zhang, Yan-zhi
;
Li, Zhen-wei
;
Zhou, Yang
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/07/01
Venenum Bufonis
Multi-component quantification
Quality evaluation
UHPLC-QqQ-MS/MS
An unexpected reaction of cinobufagin analogues in the presence of PPh3/I-2
期刊论文
MONATSHEFTE FUR CHEMIE, 2020, 卷号: 151, 期号: 4, 页码: 617-623
作者:
Zhou, Yang
;
Zhang, Yanzhi
;
Chen, Xubing
;
Hou, Jinjun
;
Long, Huali
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  |  
浏览/下载:22/0
  |  
提交时间:2020/07/01
Cinobufagin
Bufalene
PPh3/I-2
Cyclopenta-1
3-Diene
Natural product
An integrated strategy for holistic quality identification of Chinese patent medicine:Liuwei Dihuang Pillsas a case study
期刊论文
PHYTOCHEMICAL ANALYSIS, 2020, 页码: 15
作者:
Wang, Xia
;
Wu, Wenyong
;
Zhang, Jianqing
;
Gao, Lei
;
Zhang, Linlin
收藏
  |  
浏览/下载:64/0
  |  
提交时间:2020/12/24
characteristic compound
holistic identification
LC-MS
LWDHP
multivariate statistical analysis
A new recombinant MS-superoxide dismutase alleviates 5-fluorouracil-induced intestinal mucositis in mice
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 3, 页码: 348-357
作者:
Yan, Xiao-xia
;
Li, Hai-long
;
Zhang, Yi-ting
;
Wu, Shou-yan
;
Lu, Heng-lei
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2020/07/01
manganese superoxide dismutase
5-fluorouracil
chemotherapy
intestinal mucositis
diarrhea
oxidative stress
cytokines
intestinal microbes
Structural basis of ligand recognition and self-activation of orphan GPR52
期刊论文
NATURE, 2020, 页码: 21
作者:
Lin, Xi
;
Li, Mingyue
;
Wang, Niandong
;
Wu, Yiran
;
Luo, Zhipu
收藏
  |  
浏览/下载:169/0
  |  
提交时间:2020/07/01
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