QQ客服 官方微博 反馈留言

浏览/检索结果: 共11条，第1-10条 帮助 限定条件 发表日期：2019     已选(0)清除 条数/页：5101520253035404550556065707580859095100   排序方式：请选择作者升序作者降序题名升序题名降序发表日期升序发表日期降序提交时间升序提交时间降序 Designing of novel ERR gamma inverse agonists by molecular modeling studies of docking and 3D-QSAR on hydroxytamoxifen derivatives 期刊论文 MEDICINAL CHEMISTRY RESEARCH, 2019, 卷号: 28, 期号: 10, 页码: 1661-1673 作者:  Li, Rui;  Du, Yongli;  Shen, Jingkang 收藏  |  浏览/下载：7/0  |  提交时间：2020/07/01 ERR gamma inverse agonist  Molecular docking  3D-QSAR  CoMFA  CoMSIA   Structure-Based Discovery and Development of a Series of Potent and Selective Bromodomain and Extra-Terminal Protein Inhibitors 期刊论文 JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 18, 页码: 8642-8663 作者:  Hu, Jianping;  Tian, Chang-Qing;  Damaneh, Mohammadali Soleimani;  Li, Yanlian;  Cao, Danyan 收藏  |  浏览/下载：11/0  |  提交时间：2020/07/01 Design and Synthesis of Potent, Selective Inhibitors of Protein Arginine Methyltransferase 4 against Acute Myeloid Leukemia 期刊论文 JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 11, 页码: 5414-5433 作者:  Guo, Zuhao;  Zhang, Zhuqing;  Yang, Hong;  Cao, Danyan;  Xu, Xiaowei 收藏  |  浏览/下载：16/0  |  提交时间：2020/07/01 Tranylcypromine and 6-trifluoroethyl thienopyrimidine hybrid as LSD1 inhibitor 期刊论文 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 6, 页码: 844-847 作者:  Wang, Xiaowen;  Su, Mingbo;  Li, You;  Liu, Tongchao;  Wang, Yujie 收藏  |  浏览/下载：11/0  |  提交时间：2020/07/01 LSD1 inhibitor  Tranylcypromine  Menin-MLL1 protei n-protein interaction inhibitor  MV4-11 antiproliferative activity  Structure activity relationship   Stereoselective N-glycosylation with N-4-acyl cytosines and efficient synthesis of gemcitabine 期刊论文 TETRAHEDRON, 2019, 卷号: 75, 期号: 9, 页码: 1203-1213 作者:  Liu, Tongchao;  Tang, Jiadeng;  Liang, Jianpeng;  Chen, Yabin;  Wang, Xiaowen 收藏  |  浏览/下载：41/0  |  提交时间：2020/07/01 Stereoselective  N-glycosylation  N-4-acyl cytosine  Nucleoside  Gemcitabine   Discovery of a series of dimethoxybenzene FGFR inhibitors with 5H-pyrrolo[2,3-b]pyrazine scaffold: structure-activity relationship, crystal structural characterization and and in vivo study 期刊论文 ACTA PHARMACEUTICA SINICA B, 2019, 卷号: 9, 期号: 2, 页码: 351-368 作者:  Wei, Peng;  Liu, Bo;  Wang, Ruifeng;  Gao, Yinglei;  Li, Lanlan 收藏  |  浏览/下载：103/0  |  提交时间：2020/07/01 Fibroblast growth factor  Tyrosine kinase receptor  Structure-based  Crystallography  Selectivity  Hybrid  5-Hydrosulfonyl-5H- pyrrolo[2.3-b]pyrazine  Inhibitor   Fragment-based drug discovery of triazole inhibitors to block PDE delta-RAS protein-protein interaction 期刊论文 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 163, 页码: 597-609 作者:  Chen, Danqi;  Chen, Yuehong;  Lian, Fulin;  Chen, Liu;  Li, Yanlian 收藏  |  浏览/下载：17/0  |  提交时间：2020/07/01 PDE delta-RAS  Fragment-based  Inhibitor  Protein-protein interaction   SCN9A Epileptic Encephalopathy Mutations Display a Gain-of-function Phenotype and Distinct Sensitivity to Oxcarbazepine. 期刊论文 Neuroscience bulletin, 2019 作者:  Zhu Yudan;  Zhang Shuzhang;  Zhang Zhiping;  Shen Yuan;  Du Kun 收藏  |  浏览/下载：4/0  |  提交时间：2019/12/05 Electrophysiological function  Epilepsy  Oxcarbazepine  SCN9A  Sensitivity  Voltage-gated sodium channel   Overview to the Hard X-ray Modulation Telescope (Insight-HXMT) Satellite 期刊论文 arXiv e-prints, 2019 作者:  Zhang, ShuangNan;  Li, TiPei;  Lu, FangJun;  Song, LiMing;  Xu, YuPeng 收藏  |  浏览/下载：164/0  |  提交时间：2019/11/18 The Structure of MT189-Tubulin Complex Provides Insights into Drug Design 期刊论文 LETTERS IN DRUG DESIGN & DISCOVERY, 2019, 卷号: 16, 期号: 9, 页码: 1069-1073 作者:  Li, Zhongping;  Ma, Lingling;  Wu, Chengyong;  Meng, Tao;  Ma, Lanping 收藏  |  浏览/下载：7/0  |  提交时间：2020/07/01 Crystal structure  tubulin  colchicine binding site  inhibitor  MT189  drug design