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科研机构
上海药物研究所 [43]
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期刊论文 [40]
会议论文 [2]
学位论文 [1]
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2021 [1]
2020 [5]
2019 [1]
2018 [1]
2017 [2]
2016 [1]
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Chemistry [3]
Biochemist... [1]
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A homogeneous time-resolved fluorometric energy transfer assay for the binding assessment of FcRn with IgG antibodies
期刊论文
JOURNAL OF IMMUNOLOGICAL METHODS, 2021, 卷号: 499, 页码: 6
作者:
Song, Yakai
;
Deng, Xiaojie
;
Shi, Wei
;
Tang, Feng
;
Huang, Wei
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2022/01/04
FcRn
TR-FRET
mAb
ADC
Pharmacokinetics
Structure-based drug optimization and biological evaluation of tetrahydroquinolin derivatives as selective and potent CBP bromodomain inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 22, 页码: 7
作者:
Bi, Xiaoyang
;
Chen, Yu
;
Sun, Zhongya
;
Lu, Wenchao
;
Xu, Pan
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2021/05/24
Drug design
CBP
Bromodomain
Inhibitor
Acute myeloid leukemia
Design, synthesis, and biological evaluation of tetrahydroquinolin derivatives as potent inhibitors of CBP bromodomain
期刊论文
BIOORGANIC CHEMISTRY, 2020, 卷号: 101, 页码: 11
作者:
Chen, Yu
;
Bi, Xiaoyang
;
Zhang, Fengcai
;
Sun, Zhongya
;
Xu, Pan
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2020/12/24
In silico screening
Drug design
CBP
Bromodomain
Inhibitor
Acute Myeloblastic Leukemia
An in vitro Fo''rster resonance energy transfer-based high-throughput screening assay identifies inhibitors of SUMOylation E2 Ubc9
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 10
作者:
Wang, Yu-zhe
;
Liu, Xiao
;
Way, George
;
Madarha, Vipul
;
Zhou, Qing-tong
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2020/07/01
SUMOylation inhibitor
WNN0605-F008
high-throughput screening
Ubc9
PIAS1
Fo''rster resonance energy transfer
surface plasmon resonance
Discovery of novel CBP bromodomain inhibitors through TR-FRET-based high-throughput screening
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 2, 页码: 286-292
作者:
Zhang, Feng-cai
;
Sun, Zhong-ya
;
Liao, Li-ping
;
Zuo, Yu
;
Zhang, Dan
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2020/07/01
CBP bromodomain
small-molecule inhibitor
high-throughput screening
TR-FRET
molecular modeling
human leukemia MV4-11 cells
discoveryofnovelcbpbromodomaininhibitorsthroughtrfretbasedhighthroughputscreening
期刊论文
actapharmacologicasinica, 2020, 卷号: 41, 期号: 2, 页码: 285
作者:
Zhang Fengcai
;
Sun Zhongya
;
Liao Liping
;
Zuo Yu
;
Zhang Dan
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2020/07/01
CBP bromodomain
small-molecule inhibitor
high-throughput screening
TR-FRET
molecular modeling
human leukemia MV4-11 cells
G-quadruplex and duplex DNA binding studies of novel Ruthenium(II) complexes containing ascididemin ligands
期刊论文
JOURNAL OF INORGANIC BIOCHEMISTRY, 2019, 卷号: 196, 页码: 10
作者:
Wumaier, Maierhaba
;
Shi, Jing-Jing
;
Yao, Tian-Ming
;
Hu, Xiao-Chun
;
Gao, Ru-Ru
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/07/01
Ruthenium complexes
G-quadruplex
Duplex DNA
Ascididemin
Structural basis for signal recognition and transduction by platelet-activating-factor receptor
期刊论文
NATURE STRUCTURAL & MOLECULAR BIOLOGY, 2018, 卷号: 25, 期号: 6, 页码: 488-+
作者:
Cao, Can
;
Tan, Qiuxiang
;
Xu, Chanjuan
;
He, Lingli
;
Yang, Linlin
收藏
  |  
浏览/下载:70/0
  |  
提交时间:2019/01/08
How Well Can Implicit Solvent Simulations Explore Folding Pathways? A Quantitative Analysis of alpha-Helix Bundle Proteins
期刊论文
JOURNAL OF CHEMICAL THEORY AND COMPUTATION, 2017, 卷号: 13, 期号: 12, 页码: 6177-6190
作者:
Shao, Qiang
;
Zhu, Weiliang
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
A Self-Assembled Ratiometric Polymeric Nanoprobe for Highly Selective Fluorescence Detection of Hydrogen Peroxide
期刊论文
LANGMUIR, 2017, 卷号: 33, 期号: 13, 页码: 3287-3295
作者:
Feng, Chongchong
;
Wang, Fengyang
;
Dang, Yijing
;
Xu, Zhiai
;
Yu, Haijun
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
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