CORC

浏览/检索结果: 共59条,第1-10条 帮助

限定条件    
已选(0)清除 条数/页:   排序方式:
Discovery of Potent Irreversible Pan-Fibroblast Growth Factor Receptor (FGFR) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 20, 页码: 9085-9104
作者:  Wang, Yuming;  Li, Lijun;  Fan, Jun;  Dai, Yang;  Jiang, Alan
收藏  |  浏览/下载:30/0  |  提交时间:2019/01/08
Pyrazolo[4,3-b]pyrimido[4,5-e][1,4]diazepine derivatives as new multi-targeted inhibitors of Aurora A/B and KDR 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 428-441
作者:  Zhang, Qiumeng;  Shen, Qianqian;  Gao, Lixin;  Tong, Linjiang;  Li, Jia
收藏  |  浏览/下载:34/0  |  提交时间:2019/01/08
Stable Cocrystals and Salts of the Antineoplastic Drug Apatinib with Improved Solubility in Aqueous Solution 期刊论文
CRYSTAL GROWTH & DESIGN, 2018, 卷号: 18, 期号: 8, 页码: 4701-4714
作者:  Zhu, Bin;  Wang, Jian-Rong;  Zhang, Qi;  Li, Meiqi;  Guo, Chunyang
收藏  |  浏览/下载:71/0  |  提交时间:2019/01/08
Design, synthesis and biological evaluation of a series of novel 2-benzamide-4-(6-oxy-N-methyl-l-naphthamide)-pyridine derivatives as potent fibroblast growth factor receptor (FGFR) inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 154, 页码: 9-28
作者:  Wei, Manman;  Peng, Xia;  Xing, Li;  Dai, Yang;  Huang, Ruimin
收藏  |  浏览/下载:63/0  |  提交时间:2019/01/08
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:  Wang, Qiang;  Liu, Feiyang;  Qi, Shuang;  Qi, Ziping;  Yan, Xiao-E.
收藏  |  浏览/下载:63/0  |  提交时间:2019/06/10
PBA2 exhibits potent anti-tumor activity via suppression of VEGFR2 mediated-cell proliferation and angiogenesis 期刊论文
BIOCHEMICAL PHARMACOLOGY, 2018, 卷号: 150, 页码: 131-140
作者:  Fang, Xiaona;  Xie, Hua;  Luo, Min;  Chen, Zhen;  Wang, Fang
收藏  |  浏览/下载:34/0  |  提交时间:2019/01/08
Preclinical characterization of anlotinib, a highly potent and selective vascular endothelial growth factor receptor-2 inhibitor 期刊论文
CANCER SCIENCE, 2018, 卷号: 109, 期号: 4, 页码: 1207-1219
作者:  Xie, Chengying;  Wan, Xiaozhe;  Quan, Haitian;  Zheng, Mingyue;  Fu, Li
收藏  |  浏览/下载:43/0  |  提交时间:2019/01/08
Ph-triggered peptide self-assembly for targeting imaging and therapy toward angiogenesis with enhanced signals 期刊论文
Acs applied materials & interfaces, 2018, 卷号: 10, 期号: 9, 页码: 7871-7881
作者:  Qian, Yixia;  Wang, Weizhi;  Wang, Zihua;  Jia, Xiangqian;  Han, Qiuju
收藏  |  浏览/下载:41/0  |  提交时间:2019/04/23
New microtubulin inhibitor MT189 suppresses angiogenesis via the JNK-VEGF/VEGFR2 signaling axis 期刊论文
CANCER LETTERS, 2018, 卷号: 416, 页码: 57-65
作者:  Xu, Lin;  Wang, Wei;  Meng, Tao;  Ma, Lan-Ping;  Tong, Lin-Jiang
收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
SOMCL-085, a novel multi-targeted FGFR inhibitor, displays potent anticancer activity in FGFR-addicted human cancer models 期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 2, 页码: 243-250
作者:  Jiang, Xi-fei;  Dai, Yang;  Peng, Xia;  Shen, Yan-yan;  Su, Yi
收藏  |  浏览/下载:54/0  |  提交时间:2019/01/08


©版权所有 ©2017 CSpace - Powered by CSpace