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LS-106, a novel EGFR inhibitor targeting C797S, exhibits antitumor activities both in vitro and in vivo 期刊论文
CANCER SCIENCE, 2021, 页码: 12
作者:  Liu, Yingqiang;  Lai, Mengzhen;  Li, Shan;  Wang, Yanan;  Feng, Fang
收藏  |  浏览/下载:61/0  |  提交时间:2022/01/18
Electron-ion collider in China 期刊论文
FRONTIERS OF PHYSICS, 2021, 卷号: 16, 期号: 6, 页码: 78
作者:  Anderle, Daniele P.;  Bertone, Valerio;  Cao, Xu;  Chang, Lei;  Chang, Ningbo
收藏  |  浏览/下载:82/0  |  提交时间:2021/12/08
Electron-ion collider in China 期刊论文
FRONTIERS OF PHYSICS, 2021, 卷号: 16, 期号: 6
作者:  Anderle, Daniele P.;  Bertone, Valerio;  Cao, Xu;  Chang, Lei;  Chang, Ningbo
收藏  |  浏览/下载:30/0  |  提交时间:2021/10/14
TANK-binding kinase 1 (TBK1): An emerging therapeutic target for drug discovery 期刊论文
DRUG DISCOVERY TODAY, 2021, 卷号: 26, 期号: 10, 页码: 2445-2455
作者:  Xiang, Shuang;  Song, Shukai;  Tang, Haotian;  Smaill, Jeff B.;  Wang, Aiqun
收藏  |  浏览/下载:23/0  |  提交时间:2021/12/01
NGPF2 triggers synaptic scaling up through ALK-LIMK-cofilin-mediated mechanisms 期刊论文
CELL REPORTS, 2021, 卷号: 36, 期号: 7, 页码: 20
作者:  Zhou, Zikai;  He, Guiqin;  Zhang, Xiaoyun;  Lv, Xin;  Zhang, Xiaolin
收藏  |  浏览/下载:65/0  |  提交时间:2021/11/04
Initial years' neutron-induced cross-section measurements at the CSNS Back-n white neutron source * 期刊论文
CHINESE PHYSICS C, 2021, 卷号: 45, 期号: 6, 页码: 14
作者:  Tang, Jingyu;  Liu, Rong;  Zhang, Guohui;  Ruan, Xichao;  Wu, Xiaoguang
收藏  |  浏览/下载:62/0  |  提交时间:2021/12/09
Integrative Proteomic Characterization of Human Lung Adenocarcinoma 期刊论文
CELL, 2020, 卷号: 182, 期号: 1, 页码: 245-+
作者:  Xu, Jun-Yu;  Zhang, Chunchao;  Wang, Xiang;  Zhai, Linhui;  Ma, Yiming
收藏  |  浏览/下载:51/0  |  提交时间:2020/12/24
2-Oxo-3,4-dihydropyrimido[4,5-d] pyrimidines as new reversible inhibitors of EGFR C797S (Cys797 to Ser797) mutant 期刊论文
CHINESE CHEMICAL LETTERS, 2020, 卷号: 31, 期号: 5, 页码: 1281-1287
作者:  Hu, Xianglong;  Xun, Qiuju;  Zhang, Tao;  Zhu, Su-Jie;  Li, Qian
收藏  |  浏览/下载:45/0  |  提交时间:2020/07/01
Design and synthesis of selective degraders of EGFR(L858R/T790M) mutant 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 192, 页码: 14
作者:  Zhang, Xin;  Xu, Fang;  Tong, Linjiang;  Zhang, Tao;  Xie, Hua
收藏  |  浏览/下载:80/0  |  提交时间:2020/07/01
Structure-Based Design of 5-Methylpyrimidopyridone Derivatives as New Wild-Type Sparing Inhibitors of the Epidermal Growth Factor Receptor Triple Mutant (EGFR(L858R/T790M/C797S)) 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 15, 页码: 7302-7308
作者:  Shen, Jiayi;  Zhang, Tao;  Zhu, Su-Jie;  Sun, Min;  Tong, Linjiang
收藏  |  浏览/下载:30/0  |  提交时间:2020/07/01


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