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Multi-omics characterization of WNT pathway reactivation to ameliorate BET inhibitor resistance in liver cancer cells 期刊论文
GENOMICS, 2021, 卷号: 113, 期号: 3, 页码: 1057-1069
作者:  Liu, Yuwei;  Xue, Mengzhu;  Cao, Danyan;  Qin, Lihuai;  Wang, Ying
收藏  |  浏览/下载:32/0  |  提交时间:2021/08/17
Metal-free quinolylation of the primary amino groups of amino acid derivatives and peptides with dihydrooxazolo[3,2-a]quinoliniums 期刊论文
GREEN CHEMISTRY, 2019, 卷号: 21, 期号: 15, 页码: 4231-4237
作者:  Liu, Peng;  Li, Bo;  Xi, Mengyu;  Chen, Zhaoqiang;  Sun, Haiguo
收藏  |  浏览/下载:9/0  |  提交时间:2020/07/01
One Pot and Metal-Free Approach to 3-(2-Hydroxybenzoyl)-1-aza-anthraquinones 期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 16, 页码: 12
作者:  Yuan, Jiaqi;  He, Qian;  Song, Shanshan;  Zhang, Xiaofei;  Miao, Zehong
收藏  |  浏览/下载:5/0  |  提交时间:2020/07/01
Inulin based glutathione-responsive delivery system for colon cancer treatment 期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2018, 卷号: 111, 页码: 1264-1272
作者:  Wang, Dongdong;  Sun, Feifei;  Lu, Chunbo;  Chen, Peng;  Wang, Zhaojie
收藏  |  浏览/下载:31/0  |  提交时间:2019/01/08
Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 页码: 156-175
作者:  Hu, Jianping;  Wang, Yingqing;  Li, Yanlian;  Cao, Danyan;  Xu, Lin
收藏  |  浏览/下载:34/0  |  提交时间:2019/01/08
Design and synthesis of 2-(4,5,6,7-tetrahydrothienopyridin-2-yl)-benzoimidazole carboxamides as novel orally efficacious Poly(ADP-ribose)polymerase (PARP) inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 145, 页码: 389-403
作者:  Chen, Xuxing;  Huan, Xiajuan;  Liu, Qiufeng;  Wang, Yuqin;  He, Qian
收藏  |  浏览/下载:31/0  |  提交时间:2019/01/08
Structural Modification of Natural Product Tanshinone I Leading to Discovery of Novel Nitrogen-Enriched Derivatives with Enhanced Anticancer Profile and Improved Drug-like Properties 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 3, 页码: 760-776
作者:  Ding, Chunyong;  Tian, Qianting;  Li, Jie;  Jiao, Mingkun;  Song, Shanshan
收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08
Discovery, mechanism and metabolism studies of 2,3-difluorophenyl-linker-containing PARP1 inhibitors with enhanced in vivo efficacy for cancer therapy 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138, 页码: 514-531
作者:  Chen, Wenhua;  Guo, Ne;  Qi, Minghui;  Dai, Haiying;  Hong, Minghuang
收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 137, 页码: 176-195
作者:  Hu, Jianping;  Wang, Yingqing;  Li, Yanlian;  Xu, Lin;  Cao, Danyan
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
discoveryofpotent24difluorolinkerpolyadpribosepolymerase1inhibitorswithenhancedwatersolubilityandinvivoanticancerefficacy 期刊论文
actapharmacologicasinica, 2017, 卷号: 38, 期号: 11, 页码: 1521
作者:  Chen Wenhua;  Song Shanshan;  Ql Minghui;  Huan Xiajuan;  Wang Yingqing
收藏  |  浏览/下载:5/0  |  提交时间:2020/07/01


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