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上海药物研究所 [39]
西北高原生物研究所 [9]
昆明植物研究所 [1]
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华中师范大学 [1]
武汉理工大学 [1]
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期刊论文 [52]
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Multi-omics characterization of WNT pathway reactivation to ameliorate BET inhibitor resistance in liver cancer cells
期刊论文
GENOMICS, 2021, 卷号: 113, 期号: 3, 页码: 1057-1069
作者:
Liu, Yuwei
;
Xue, Mengzhu
;
Cao, Danyan
;
Qin, Lihuai
;
Wang, Ying
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2021/08/17
Multi-omics
BET inhibitor responses
WNT pathway
Liver cancer
Precise therapy
Metal-free quinolylation of the primary amino groups of amino acid derivatives and peptides with dihydrooxazolo[3,2-a]quinoliniums
期刊论文
GREEN CHEMISTRY, 2019, 卷号: 21, 期号: 15, 页码: 4231-4237
作者:
Liu, Peng
;
Li, Bo
;
Xi, Mengyu
;
Chen, Zhaoqiang
;
Sun, Haiguo
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/07/01
One Pot and Metal-Free Approach to 3-(2-Hydroxybenzoyl)-1-aza-anthraquinones
期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 16, 页码: 12
作者:
Yuan, Jiaqi
;
He, Qian
;
Song, Shanshan
;
Zhang, Xiaofei
;
Miao, Zehong
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  |  
浏览/下载:5/0
  |  
提交时间:2020/07/01
3-(2-hydroxybenzoyl)-1-aza-anthraquinones
chromones
anti-proliferation agent
Inulin based glutathione-responsive delivery system for colon cancer treatment
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2018, 卷号: 111, 页码: 1264-1272
作者:
Wang, Dongdong
;
Sun, Feifei
;
Lu, Chunbo
;
Chen, Peng
;
Wang, Zhaojie
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
Inulin
Lipoic add
Polymeric micelles
Colorectal cancer
Probiotic
Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 页码: 156-175
作者:
Hu, Jianping
;
Wang, Yingqing
;
Li, Yanlian
;
Cao, Danyan
;
Xu, Lin
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  |  
浏览/下载:34/0
  |  
提交时间:2019/01/08
BRD4
BI2536
Indoline
WPF binders
c-Myc
PD-L1
Design and synthesis of 2-(4,5,6,7-tetrahydrothienopyridin-2-yl)-benzoimidazole carboxamides as novel orally efficacious Poly(ADP-ribose)polymerase (PARP) inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 145, 页码: 389-403
作者:
Chen, Xuxing
;
Huan, Xiajuan
;
Liu, Qiufeng
;
Wang, Yuqin
;
He, Qian
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  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
PARP1/2 inhibitor
Benzimidazole
4,5,6,7-Tetrahydrothienopyridine
Co-crystal structure
Isothermal Titration Calorimetry
Structural Modification of Natural Product Tanshinone I Leading to Discovery of Novel Nitrogen-Enriched Derivatives with Enhanced Anticancer Profile and Improved Drug-like Properties
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 3, 页码: 760-776
作者:
Ding, Chunyong
;
Tian, Qianting
;
Li, Jie
;
Jiao, Mingkun
;
Song, Shanshan
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  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
Discovery, mechanism and metabolism studies of 2,3-difluorophenyl-linker-containing PARP1 inhibitors with enhanced in vivo efficacy for cancer therapy
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138, 页码: 514-531
作者:
Chen, Wenhua
;
Guo, Ne
;
Qi, Minghui
;
Dai, Haiying
;
Hong, Minghuang
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
Antitumor drug
BRCA1/2
PARP inhibitors
Molecular docking
Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 137, 页码: 176-195
作者:
Hu, Jianping
;
Wang, Yingqing
;
Li, Yanlian
;
Xu, Lin
;
Cao, Danyan
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2019/01/08
BRD4 inhibitor
Kinase
BI-2536
Dihydroquinoxalin-2(1H)-one
discoveryofpotent24difluorolinkerpolyadpribosepolymerase1inhibitorswithenhancedwatersolubilityandinvivoanticancerefficacy
期刊论文
actapharmacologicasinica, 2017, 卷号: 38, 期号: 11, 页码: 1521
作者:
Chen Wenhua
;
Song Shanshan
;
Ql Minghui
;
Huan Xiajuan
;
Wang Yingqing
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2020/07/01
PARP INHIBITORS
MEDICINAL CHEMISTRY
DRUG DISCOVERY
CANCER
THERAPY
DESIGN
FLUORINE
SUCCESS
PREDICT
METRICS
PARP-1 inhibitor
olaparib
breast cancer
BRCA-deficient tumors
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