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科研机构
山东大学 [19]
合肥物质科学研究院 [7]
中国水产科学院 [5]
安徽大学 [4]
西安交通大学 [3]
北京航空航天大学 [3]
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期刊论文 [68]
会议论文 [6]
发表日期
2018 [74]
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Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:
Liu, Xuesong
;
Wang, Beilei
;
Chen, Cheng
;
Jiang, Zongru
;
Hu, Chen
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/11
ABL kinase
Kinase inhibitor
ABL mutant
CML
Salviachinensines A-F, Antiproliferative Phenolic Derivatives from the Chinese Medicinal Plant Salvia chinensis
期刊论文
JOURNAL OF NATURAL PRODUCTS, 2018, 卷号: 81, 期号: 11, 页码: 2531-2538
作者:
Wang, Qi
;
Hu, Zhenquan
;
Li, Xixiang
;
Wang, Aoli
;
Wu, Hong
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2019/12/25
Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 896-916
作者:
Wang, Beilei
;
Wu, Jiaxin
;
Wu, Yun
;
Chen, Cheng
;
Zou, Fengming
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  |  
浏览/下载:65/0
  |  
提交时间:2019/12/25
CDK9
Kinase inhibitor
Structure-activity relationship
Leukemia
Multidecadally resolved polarity oscillations during a geomagnetic excursion
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2018, 卷号: 115, 期号: 36, 页码: 8913-8918
作者:
Zhao, Xiang
;
Shen, Chuan-Chou
;
Chou,Yu-Min
;
Jiang, Zhaoxia
;
Liu, Jianxing
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  |  
浏览/下载:50/0
  |  
提交时间:2018/09/30
Multidecadally Resolved Polarity Oscillations
Geomagnetic Excursion
Abrupt Reversal Transition
Asymmetrical Interhemispheric Polarity Drifts
Stalagmite U-th Dating
Multidecadally resolved polarity oscillations during a geomagnetic excursion
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2018, 卷号: 115, 期号: 36, 页码: 8913-8918
作者:
Chou, Yu-Min
;
Jiang, Xiuyang
;
Liu, Qingsong
;
Hu, Hsun-Ming
;
Wu, Chung-Che
收藏
  |  
浏览/下载:63/0
  |  
提交时间:2018/10/08
multidecadally resolved polarity oscillations
geomagnetic excursion
abrupt reversal transition
asymmetrical interhemispheric polarity drifts
stalagmite U-Th dating
Multidecadally resolved polarity oscillations during a geomagnetic excursion
期刊论文
Proceedings of the National Academy of Sciences of the United States of America, 2018, 卷号: 115, 期号: 36, 页码: 8913-8918
作者:
Chou; Yu-Min
;
Jiang, Xiuyang
;
Liu, Qingsong
;
Hu, Hsun-Ming
;
Wu, Chung-Che
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/04/01
Abrupt reversal transition
Asymmetrical interhemispheric polarity drifts
Geomagnetic excursion
Multidecadally resolved polarity oscillations
Stalagmite U-Th dating
Copolymers of Bis-Diketopyrrolopyrrole and Benzothiadiazole Derivatives for High-Performance Ambipolar Field-Effect Transistors on Flexible Substrates
期刊论文
ACS APPLIED MATERIALS & INTERFACES, 2018, 卷号: 10, 期号: 31, 页码: 25858-25865
作者:
Chen, Jinyang
;
Jiang, Yingying
;
Yang, Jie
;
Sun, Yunlong
;
Shi, Longxian
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  |  
浏览/下载:43/0
  |  
提交时间:2019/04/09
Bis-diketopyrrolopyrrole
"acceptor Dimerization" Strategy
Field-effect Transistor
Ambipolar Polymer
Flexible Substrate
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3K delta) inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 页码: 831-846
作者:
Liang, Xiaofei
;
Li, Feng
;
Chen, Cheng
;
Jiang, Zongru
;
Wang, Aoli
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/12/10
PI3K delta
Kinase inhibitor
Acute myeloid leukemia
Structure-activity relationship
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:
Xue, Yu
;
Song, Peiran
;
Song, Zilan
;
Wang, Aoli
;
Tong, Linjiang
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2019/08/23
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:
Xue, Yu
;
Song, Peiran
;
Song, Zilan
;
Wang, Aoli
;
Tong, Linjiang
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2019/01/08
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