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科研机构
北京大学 [5]
内容类型
期刊论文 [5]
发表日期
2017 [1]
2016 [1]
2015 [1]
2013 [2]
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专题:北京大学
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Discovery of 2-((3-Acrylamido-4-methylphenyl)amino)-N-(2-methyl5-(3,4,5-trimethoxyben zamido)phenyI)-4-(methylamino)pyrimidine-5-carboxamide (CHMFL-BMX-078) as a Highly Potent and Selective Type II Irreversible Bone Marrow Kinase in the X Chro
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017
Liang, Xiaofei
;
Lv, Fengchao
;
Wang, Beilei
;
Yu, Kailin
;
Wu, Hong
;
Qi, Ziping
;
Jiang, Zongru
;
Chen, Cheng
;
Wang, Aoli
;
Miao, Weili
;
Wang, Wenchao
;
Hu, Zhenquan
;
Liu, Juan
;
Liu, Xiaochuan
;
Zhao, Zheng
;
Wang, Li
;
Zhang, Shanchuan
;
Ye, Zi
;
Wang, Chu
;
Ren, Tao
;
Wang, Yinsheng
;
Liu, Qingsong
;
Liu, Jing
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
GROWTH-FACTOR RECEPTOR
TYROSINE KINASE
COVALENT
ETK/BMX
FAMILY
CELLS
GENE
BTK
ACTIVATION
EXPRESSION
Ibrutinib targets mutant-EGFR kinase with a distinct binding conformation
期刊论文
ONCOTARGET, 2016
Wang, Aoli
;
Yan, Xiao-E
;
Wu, Hong
;
Wang, Wenchao
;
Hu, Chen
;
Chen, Cheng
;
Zhao, Zheng
;
Zhao, Peng
;
Li, Xixiang
;
Wang, Li
;
Wang, Beilei
;
Ye, Zi
;
Wang, Jinhua
;
Wang, Chu
;
Zhang, Wei
;
Gray, Nathanael S.
;
Weisberg, Ellen L.
;
Chen, Liang
;
Liu, Jing
;
Yun, Cai-Hong
;
Liu, Qingsong
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2017/12/04
Ibrutinib
EGFR kinase
DFG-in/c-Helix-out
inactive conformation
NSCLC
BRUTONS TYROSINE KINASE
MANTLE-CELL LYMPHOMA
CHRONIC LYMPHOCYTIC-LEUKEMIA
GROWTH-FACTOR RECEPTOR
INHIBITORS
BTK
SYSTEM
CRYSTALLOGRAPHY
ACTIVATION
RESISTANCE
Ibrutinib selectively and irreversibly targets EGFR (L858R, Del19) mutant but is moderately resistant to EGFR (T790M) mutant NSCLC Cells
期刊论文
ONCOTARGET, 2015
Wu, Hong
;
Wang, Aoli
;
Zhang, Wei
;
Wang, Beilei
;
Chen, Cheng
;
Wang, Wenchao
;
Hu, Chen
;
Ye, Zi
;
Zhao, Zheng
;
Wang, Li
;
Li, Xixiang
;
Yu, Kailin
;
Liu, Juan
;
Wu, Jiaxin
;
Yan, Xiao-E
;
Zhao, Peng
;
Wang, Jinhua
;
Wang, Chu
;
Weisberg, Ellen L.
;
Gray, Nathanael S.
;
Yun, Cai-Hong
;
Liu, Jing
;
Chen, Liang
;
Liu, Qingsong
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
ibrutinib
NSCLC
EGFR mutation
drug resistance
drug combination
GROWTH-FACTOR RECEPTOR
BRUTONS TYROSINE KINASE
CHRONIC LYMPHOCYTIC-LEUKEMIA
LUNG-CANCER
ACQUIRED-RESISTANCE
INHIBITORS
BTK
MUTATION
GEFITINIB
LYMPHOMA
The production of phytolith-occluded carbon in China's forests: implications to biogeochemical carbon sequestration
期刊论文
全球变化生物学, 2013
Song, Zhaoliang
;
Liu, Hongyan
;
Li, Beilei
;
Yang, Xiaomin
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/11/10
bamboo
biogeochemical carbon sequestration
carbon sink
China
forest
phytolith-occluded carbon (PhytOC)
PLANT-IMPACT
SILICON
STORAGE
BAMBOO
CYCLE
CO2
The production and accumulation of phytolith-occluded carbon in Baiyangdian reed wetland of China
期刊论文
applied geochemistry, 2013
Li, Zimin
;
Song, Zhaoliang
;
Li, Beilei
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2015/11/11
BIOGENETIC OPAL
SILICON
SEQUESTRATION
SOILS
WHEAT
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