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Discovery of potent 2,4-difluoro-linker poly(ADP-ribose) polymerase 1 inhibitors with enhanced water solubility and in vivo anticancer efficacy 期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1521-1532
作者:  Chen, Wen-hua;  Song, Shan-shan;  Qi, Ming-hui;  Huan, Xia-juan;  Wang, Ying-qing
收藏  |  浏览/下载:26/0  |  提交时间:2019/01/08
Discovery, mechanism and metabolism studies of 2,3-difluorophenyl-linker-containing PARP1 inhibitors with enhanced in vivo efficacy for cancer therapy 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138, 页码: 514-531
作者:  Chen, Wenhua;  Guo, Ne;  Qi, Minghui;  Dai, Haiying;  Hong, Minghuang
收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
Combining 53BP1 with BRCA1 as a biomarker to predict the sensitivity of poly(ADP-ribose) polymerase (PARP) inhibitors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 7, 页码: 1038-1047
作者:  Yang, Zhong-min;  Liao, Xue-mei;  Chen, Yi;  Shen, Yan-yan;  Yang, Xin-ying
收藏  |  浏览/下载:25/0  |  提交时间:2019/01/08
AsperflavipineA: A Cytochalasan Heterotetramer Uniquely Defined by a Highly Complex Tetradecacyclic Ring System from Aspergillus flavipes QCS12 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2017, 卷号: 56, 期号: 19, 页码: 5242-5246
作者:  Zhu, Hucheng;  Chen, Chunmei;  Tong, Qingyi;  Yang, Jing;  Wei, Guangzheng
收藏  |  浏览/下载:38/0  |  提交时间:2017/06/30
A novel cycloartane triterpenoid from Cimicifuga induces apoptotic and autophagic cell death in human colon cancer HT-29 cells 期刊论文
ONCOLOGY REPORTS, 2017, 卷号: 37, 期号: 4, 页码: 2079-2086
作者:  Dai, Xiaoli;  Liu, Jing;  Nian, Yin;  Qiu, Ming-Hua;  Luo, Ying
收藏  |  浏览/下载:30/0  |  提交时间:2017/06/01
Phosphoglycerate mutase 1 regulates dNTP pool and promotes homologous recombination repair in cancer cells 期刊论文
JOURNAL OF CELL BIOLOGY, 2017, 卷号: 216, 期号: 2, 页码: 409-424
作者:  Qu, Jia;  Sun, Wenyi;  Zhong, Jie;  Lv, Hao;  Zhu, Mingrui
收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08
Poly(ADP-ribose)polymerase (PARP) inhibition and anticancer activity of simmiparib, a new inhibitor undergoing clinical trials 期刊论文
CANCER LETTERS, 2017, 卷号: 386, 页码: 47-56
作者:  Yuan, Bo;  Ye, Na;  Song, Shan-Shan;  Wang, Yu-Ting;  Song, Zilan
收藏  |  浏览/下载:43/0  |  提交时间:2019/01/08
Novel PARP1/2 inhibitor mefuparib hydrochloride elicits potent in vitro and in vivo anticancer activity, characteristic of high tissue distribution 期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 3, 页码: 4156-4168
作者:  He, Jin-Xue;  Wang, Meng;  Huan, Xia-Juan;  Chen, Chuan-Huizi;  Song, Shan-Shan
收藏  |  浏览/下载:35/0  |  提交时间:2019/01/08
Enhanced Radiotherapy using Bismuth Sulfide Nanoagents Combined with Photo-thermal Treatment 期刊论文
THERANOSTICS, 2017, 卷号: 7, 期号: 17, 页码: 4087-4098
作者:  Yong, Y;  Yang, G;  Dai, YH;  Song, X;  Pan, Y
收藏  |  浏览/下载:18/0  |  提交时间:2019/08/27


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