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A general strategy to the intracellular sensing of glycosidases using AIE-based glycoclusters 期刊论文
CHEMICAL SCIENCE, 2021, 卷号: 13, 期号: 1, 页码: 247-256
作者:  Dong, Lei;  Zhang, Min-Yu;  Han, Hai-Hao;  Zang, Yi;  Chen, Guo-Rong
收藏  |  浏览/下载:27/0  |  提交时间:2022/01/18
Theoretical study and application of 2-phenyl-1,3,4-thiadiazole derivatives with optical and inhibitory activity against SHP1 期刊论文
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2021, 页码: 14
作者:  Zhang, Chun;  Sun, Yi-Tao;  Gao, Li-Xin;  Feng, Bo;  Yan, Xue
收藏  |  浏览/下载:16/0  |  提交时间:2022/01/18
NIR-II imaging of hepatocellular carcinoma based on a humanized anti-GPC3 antibody 期刊论文
RSC MEDICINAL CHEMISTRY, 2021, 页码: 8
作者:  Shi, Hui;  Huttad, Lakshmi Vageesh;  Tan, Mingdian;  Liu, Hongguang;  Chua, Mei-Sze
收藏  |  浏览/下载:20/0  |  提交时间:2022/01/04
Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site 期刊论文
ACS CHEMICAL BIOLOGY, 2021, 卷号: 16, 期号: 11, 页码: 2444-2452
作者:  Wang, Jiang;  Yang, Dehua;  Cheng, Xi;  Yang, Linlin;  Wang, Zhaohui
收藏  |  浏览/下载:23/0  |  提交时间:2022/01/04
The Novel RET Inhibitor SYHA1815 Inhibits RET-Driven Cancers and Overcomes Gatekeeper Mutations by Inducing G1 Cell-Cycle Arrest through c-Myc Downregulation 期刊论文
MOLECULAR CANCER THERAPEUTICS, 2021, 卷号: 20, 期号: 11, 页码: 2198-2206
作者:  Jiang, Yuchen;  Peng, Xia;  Ji, Yinchun;  Dai, Yang;  Fang, Yanfen
收藏  |  浏览/下载:28/0  |  提交时间:2021/12/16
Enhancing the Potential of Miniature-Scale DNA-Compatible Radical Reactions via an Electron Donor-Acceptor Complex and a Reversible Adsorption to Solid Support Strategy 期刊论文
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 19, 页码: 7381-7385
作者:  Lin, Bizhen;  Lu, Weiwei;  Chen, Zhen-yu;  Zhang, Yue;  Duan, Yin-zhe
收藏  |  浏览/下载:12/0  |  提交时间:2021/12/01
The inhibitory effect of 225 frequently-used traditional Chinese medicines for CYP3A4 metabolic enzyme by isoform-specific probe 期刊论文
FITOTERAPIA, 2021, 卷号: 152, 页码: 5
作者:  Wei, Wenlong;  Li, Zhenwei;  Li, Hao-jv;  An, Yaling;  Qu, Hua
收藏  |  浏览/下载:31/0  |  提交时间:2021/08/17
Bufalin exerts antitumor effects in neuroblastoma via the induction of reactive oxygen species-mediated apoptosis by targeting the electron transport chain 期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR MEDICINE, 2020, 卷号: 46, 期号: 6, 页码: 2137-2149
作者:  Pan, Lijia;  Nie, Litong;  Yao, Sheng;  Bi, Aiwei;  Ye, Yang
收藏  |  浏览/下载:26/0  |  提交时间:2020/12/24
Structure-based drug optimization and biological evaluation of tetrahydroquinolin derivatives as selective and potent CBP bromodomain inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 22, 页码: 7
作者:  Bi, Xiaoyang;  Chen, Yu;  Sun, Zhongya;  Lu, Wenchao;  Xu, Pan
收藏  |  浏览/下载:20/0  |  提交时间:2021/05/24
Unveiling conformational dynamics changes of H-Ras induced by mutations based on accelerated molecular dynamics 期刊论文
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2020, 卷号: 22, 期号: 37, 页码: 21238-21250
作者:  Chen, Jianzhong;  Wang, Wei;  Pang, Laixue;  Zhu, Weiliang
收藏  |  浏览/下载:26/0  |  提交时间:2020/12/21


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