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| Design, synthesis and biological evaluation of a series of novel 2-benzamide-4-(6-oxy-N-methyl-1-naphthamide)-pyridine derivatives as potent fibroblast growth factor receptor (FGFR) inhibitors 会议论文 作者: Zhang, Ao 收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08 |
| IDENTIFICATION OF NOVEL HUMAN PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9 (PCSK9) INHIBITORS USING A CELL-BASED HIGH-THROUGHPUT SCREENING ASSAY 会议论文 ATHEROSCLEROSIS, 2017-08-01 作者: Wang, Li; Hong, Bin; Wang, Xuelei 收藏  |  浏览/下载:3/0  |  提交时间:2020/01/04 |
| Synthesis and Biological Evaluation of Novel Berberine Derivatives as Potent Inhibitors against IFN-γ-induced IDO1 Expression 会议论文 第十三届全国抗生素学术会议, 中国福建福州, 2017-11-22 作者: Pang WQ(庞伟强); Wang YX(汪燕翔); Deng HB(邓洪斌) 收藏  |  浏览/下载:5/0  |  提交时间:2020/01/04
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| HDAC Inhibitors Lead to Significant Survival Benefit in a Novel Fusion Protein TBLR1-Rara Induced Murine Promyelocytic Leukemia Model 会议论文 BLOOD, 2016-12-02 作者: Li, Shouyun; Liu, Shuang; Chen, Shuying; Chen, Yirui; Wang, Ying 收藏  |  浏览/下载:5/0  |  提交时间:2020/01/04 |
| 丙酮酸脱氢酶激酶共价抑制剂JX06抗肿瘤活性和机制研究(英文) 会议论文 作者: 孙文怡; 谢作权; 刘逸夫; 赵丹; 武志翔 收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
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| JX06 selectively inhibits pyruvate dehydrogenase kinase 1 by covalently targeting a cysteine residue 会议论文 作者: Sun WY(孙文怡); Xie ZQ(谢作权); Liu YF(刘逸夫); Zhao D(赵丹); Wu ZX(武志翔) 收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08
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| Novel fatty acid binding protein 4 (FABP4) inhibitors: virtual screening, synthesis and crystal structure determination 会议论文 作者: Cai HY(蔡海燕); Chen KX(陈凯先); Ding HP(丁海鹏); Chen TT(陈甜甜); Yan GR(闫桂蕊) 收藏  |  浏览/下载:3/0  |  提交时间:2019/12/19
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| A novel accurate method of human protein tyrosine phosphatase 1B inhibitors high-throughput screening 会议论文 The 12th Meeting of the Asia Pacific Federation of Pharmacologists(第十二届亚洲太平洋地区药理学家联盟会议暨中国药理学会第十二次全国学术会议), 2013-07-09 - 收藏  |  浏览/下载:4/0  |  提交时间:2019/12/23
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| A novel accurate method of human protein tyroslne phosphatase 1B inhibitors highthroughput screening 会议论文 2013-07-05 作者: Xiao-bin PANG[1]; Xin-mei XIE[2]; Qing-hui ZHAO[3]; Shou-bao WANG[4]; Guan-hua DU[5] 收藏  |  浏览/下载:4/0  |  提交时间:2019/12/23
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| A novel anti-rheumatic drug,iguratimod for RA-an initial clinical trial 会议论文 作者: Feng XIAO; Ling-ling ZHANG; Wei WEI; Jian-hua XU; Xing-fu LI 收藏  |  浏览/下载:6/0  |  提交时间:2019/12/31
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