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Discovery of new [1,4]dioxino[2,3-f]quinazoline-based inhibitors of EGFR including the T790M/L858R mutant 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 13, 页码: 2871-2881
Qin, Xuemei; Li, Zhipeng; Yang, Leifu; Liu, Peng; Hu, Liming; Zeng, Chengchu; Pan, Zhiyong
收藏  |  浏览/下载:59/0  |  提交时间:2016/12/16
Novel morpholin-3-one fused quinazoline derivatives as EGFR tyrosine kinase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 6, 页码: 1571-1575
作者:  Lv, Yongjuan;  Qin, Xuemei;  Liu, Peng;  Li, Zhipeng;  Hu, Liming
收藏  |  浏览/下载:40/0  |  提交时间:2018/12/13
Novel morpholin-3-one fused quinazoline derivatives as EGFR tyrosine kinase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 6, 页码: 1571-1575
Qin, Xuemei; Lv, Yongjuan; Liu, Peng; Li, Zhipeng; Hu, Liming; Zeng, Chengchu; Yang, Leifu
收藏  |  浏览/下载:50/0  |  提交时间:2016/12/16
Discovery of new [1,4]dioxino[2,3-f]quinazoline-based inhibitors of EGFR including the T790M/L858R mutant 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 13, 页码: 2871-2881
作者:  Pan, Zhiyong;  Li, Zhipeng;  Yang, Leifu;  Liu, Peng;  Hu, Liming
收藏  |  浏览/下载:36/0  |  提交时间:2018/12/13
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M) 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
Chan, Shingpan; Han, Kun; Qu, Rong; Tong, Linjiang; Li, Yingjun; Zhang, Zhang; Cheng, Huimin; Lu, Xiaoyun; Patterson, Adam; Smaill, Jeff; Ren, Xiaomei; Ding, Jian; Xie, Hua; Ding, Ke
收藏  |  浏览/下载:246/0  |  提交时间:2016/12/16
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M) 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
作者:  Smaill, Jeff;  Lu, Xiaoyun;  Cheng, Huimin;  Zhang, Zhang;  Li, Yingjun
收藏  |  浏览/下载:48/0  |  提交时间:2018/12/13
Pyrimido[4,5-d]pyrimidin-4(1H)-one Derivatives as Selective Inhibitors of EGFR Threonine(790) to Methionine(790) (T790M) Mutants 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2013, 卷号: 52, 期号: 32
作者:  Zhang, Lianwen;  Ding, Ke;  Wang, Shaomeng;  Ren, Xiaomei;  Li, Honglin
收藏  |  浏览/下载:39/0  |  提交时间:2018/12/13
Pyrimido[4,5-d]pyrimidin-4(1H)-one Derivatives as Selective Inhibitors of EGFR Threonine(790) to Methionine(790) (T790M) Mutants 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2013, 卷号: 52, 期号: 32
Xu, Tianfeng; Zhang, Lianwen; Xu, Shilin; Yang, Chao-Yie; Luo, Jinfeng; Ding, Fang; Lu, Xiaoyun; Liu, Yingxue; Tu, Zhengchao; Li, Shiliang; Pei, Duanqing; Cai, Qian; Li, Honglin; Ren, Xiaomei; Wang, Shaomeng; Ding, Ke
收藏  |  浏览/下载:50/0  |  提交时间:2016/12/16


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