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Design, synthesis, in vitro evaluation of a new pyrrolo[1,2-a]thiazolo[5,4-d]pyrimidinone derivatives as cholinesterase inhibitors against Alzheimer's disease 期刊论文
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2022, 卷号: 59, 期号: 6, 页码: 1086-1101
作者:  Zeng, Y (Zeng, Yan) [1] , [2];  Nie, LF (Nie, Lifei) [1];  Liu, L (Liu, Liu) [1];  Niu, C (Niu, Chao) [1] , [2];  Li, Y (Li, Yi) [1] , [2]
收藏  |  浏览/下载:19/0  |  提交时间:2022/06/21
Hollow urchin-shaped manganese dioxide microspheres immobilized acetylcholinesterase for rapid screening inhibitors from traditional herbal medicines 期刊论文
Journal of Chromatography A, 2022, 期号: 1665, 页码: 462824
作者:  Liu J(刘佳);  Ha W(哈伟);  Zhang HX(张海霞);  Shi YP(师彦平)
收藏  |  浏览/下载:2/0  |  提交时间:2022/11/15
Kinetics-Driven Drug Design Strategy for Next-Generation Acetylcholinesterase Inhibitors to Clinical Candidate 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 4, 页码: 1844-1855
作者:  Zhou, Yu;  Fu, Yan;  Yin, Wanchao;  Li, Jian;  Wang, Wei
收藏  |  浏览/下载:21/0  |  提交时间:2021/05/24
[1,5]-Hydride Shift-Cyclization versus C(sp(2))-H Functionalization in the Knoevenagel-Cyclization Domino Reactions of 1,4-and 1,5-Benzoxazepines 期刊论文
MOLECULES, 2020, 卷号: 25, 期号: 6, 页码: 19
作者:  Vargane, Dora Szaloki;  Toth, Laszlo;  Buglyo, Balazs;  Kiss-Szikszai, Attila;  Mandi, Attila
收藏  |  浏览/下载:37/0  |  提交时间:2020/07/01
Discovery and Biological Evaluation of New Selective Acetylcholinesterase Inhibitors with Anti-A beta Aggregation Activity through Molecular Docking-Based Virtual Screening 期刊论文
CHEMICAL & PHARMACEUTICAL BULLETIN, 2020, 卷号: 68, 期号: 2, 页码: 161-166
作者:  Liu, Guangpu;  Jiao, Yang;  Lin, Yongqiang;  Hao, Haifang;  Dou, Yanli
收藏  |  浏览/下载:53/0  |  提交时间:2020/07/01
Design, synthesis and biological evaluation of novel copper-chelating acetylcholinesterase inhibitors with pyridine and N-benzylpiperidine fragments 期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 93, 页码: 13
作者:  Zhou, Yeheng;  Sun, Wei;  Peng, Jiale;  Yan, Hui;  Zhang, Li
收藏  |  浏览/下载:14/0  |  提交时间:2020/03/18
Donepezil, a drug for Alzheimer's disease, promotes oligodendrocyte generation and remyelination 期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 11, 页码: 1386-1393
作者:  Cui, Xue;  Guo, Yu-e;  Fang, Jia-hui;  Shi, Chang-jie;  Suo, Na
收藏  |  浏览/下载:68/0  |  提交时间:2020/07/01
Quantitative visualization and detection of acetylcholinesterase activity and its inhibitor based on the oxidation character of ultrathin MnO2 nanosheets. Analytical Methods, Analytical Methods, 2019, 期刊论文
Analytical Methods, 2019, 卷号: 11, 期号: -, 页码: 4931–4938
作者:  Cai-Hong Li;  Jun-Li Yang;  Wei-Feng Wang;  Won Keun Oh;  Dang Lan Huong
收藏  |  浏览/下载:55/0  |  提交时间:2019/11/11
Discovery of New Selective Butyrylcholinesterase (BChE) Inhibitors with Anti-A beta Aggregation Activity: Structure-Based Virtual Screening, Hit Optimization and Biological Evaluation 期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 14, 页码: 21
作者:  Jiang, Cheng-Shi;  Ge, Yong-Xi;  Cheng, Zhi-Qiang;  Wang, Yin-Yin;  Tao, Hong-Rui
收藏  |  浏览/下载:13/0  |  提交时间:2020/07/01
Surface modification with highly-homogeneous porous silica layer for enzyme immobilization in capillary enzyme microreactors 期刊论文
TALANTA, 2019, 卷号: 197, 页码: 539-547
作者:  Liu, Xin;  Zhu, Xudong;  Camara, Mohamed Amara;  Qu, Qishu;  Shan, Yichu
收藏  |  浏览/下载:174/0  |  提交时间:2019/06/20


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