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Sublyratins A-O, Labdane-Type Diterpenoids from Croton sublyratus 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2021, 卷号: 84, 期号: 11, 页码: 2971-2980
作者:  Qi, Jing-Jing;  Zhou, Jun-Su;  Zhang, Yan;  Fan, Yao-Yue;  Zhou, Bin
收藏  |  浏览/下载:19/0  |  提交时间:2022/01/18
Molecular insights into differentiated ligand recognition of the human parathyroid hormone receptor 2 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 32, 页码: 8
作者:  Wang, Xi;  Cheng, Xi;  Zhao, Lihua;  Wang, Yuzhe;  Ye, Chenyu
收藏  |  浏览/下载:25/0  |  提交时间:2021/11/04
Activation pathway of a G protein-coupled receptor uncovers conformational intermediates as targets for allosteric drug design 期刊论文
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 15
作者:  Lu, Shaoyong;  He, Xinheng;  Yang, Zhao;  Chai, Zongtao;  Zhou, Shuhua
收藏  |  浏览/下载:35/0  |  提交时间:2021/11/04
Metabolically controlled histone H4K5 acylation/acetylation ratio drives BRD4 genomic distribution 期刊论文
CELL REPORTS, 2021, 卷号: 36, 期号: 4, 页码: 22
作者:  Gao, Mengqing;  Wang, Jin;  Rousseaux, Sophie;  Tan, Minjia;  Pan, Lulu
收藏  |  浏览/下载:67/0  |  提交时间:2021/11/04
Discovery of SARS-CoV-2-E channel inhibitors as antiviral candidates 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 7
作者:  Wang, Yi;  Fang, Sui;  Wu, Yan;  Cheng, Xi;  Zhang, Lei-ke
收藏  |  浏览/下载:103/0  |  提交时间:2021/08/17
Global identification of phospho-dependent SCF substrates reveals a FBXO22 phosphodegron and an ERK-FBXO22-BAG3 axis in tumorigenesis 期刊论文
CELL DEATH AND DIFFERENTIATION, 2021, 页码: 13
作者:  Liu, Ping;  Cong, Xiaoji;  Liao, Shengjie;  Jia, Xinglong;  Wang, Xiaomin
收藏  |  浏览/下载:79/0  |  提交时间:2021/08/17
Structure-Guided Development of Small-Molecule PRC2 Inhibitors Targeting EZH2-EED Interaction 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 12, 页码: 8194-8207
作者:  Du, Daohai;  Xu, Dandan;  Zhu, Licheng;  Stazi, Giulia;  Zwergel, Clemens
收藏  |  浏览/下载:74/0  |  提交时间:2021/08/17
SAF-248, a novel PI3K delta-selective inhibitor, potently suppresses the growth of diffuse large B-cell lymphoma 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:  Zhang, Xi;  Duan, Yu-ting;  Wang, Yi;  Zhao, Xing-dong;  Sun, Yi-ming
收藏  |  浏览/下载:37/0  |  提交时间:2021/05/24
A 36-week multicenter, randomized, double-blind, placebo-controlled, parallel-group, phase 3 clinical trial of sodium oligomannate for mild-to-moderate Alzheimer’s dementia 期刊论文
Alzheimer's Research & Therapy, 2021, 卷号: 13, 期号: 1
作者:  Xiao,Shifu;  Chan,Piu;  Wang,Tao;  Hong,Zhen;  Wang,Shuzhen
收藏  |  浏览/下载:148/0  |  提交时间:2021/05/24
Discovery of 5-Benzylidene-2-phenyl-1,3-dioxane-4,6-diones as Highly Potent and Selective SIRT1 Inhibitors 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 12, 期号: 3, 页码: 397-403
作者:  Li, Chunpu;  Hu, Sha-Sha;  Yang, Lisheng;  Wang, Min;  Long, Jian-Dong
收藏  |  浏览/下载:57/0  |  提交时间:2021/05/24


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