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组蛋白去乙酰化I型酶选择性抑制剂与8-羟基鸟嘌呤苷酸酶抑制剂的设计合成及抗肿瘤活性评价 学位论文
广州生物院: 中国科学院大学, 2016
作者:  姚毅武
收藏  |  浏览/下载:25/0  |  提交时间:2018/12/25
吡唑[1,5-a]并吡啶-3-酰胺类新型抗结核药物的设计、合成及生物活性研究 学位论文
广州生物院: 中国科学院大学, 2016
作者:  汤健
收藏  |  浏览/下载:15/0  |  提交时间:2018/12/25
Design, synthesis, and in vitro biological evaluation of novel 6-methyl-7-substituted-7-deaza purine nucleoside analogs as anti-influenza A agents 期刊论文
ANTIVIRAL RESEARCH, 2016, 卷号: 129, 页码: 13-20
Lin, Cai; Sun, Chenghai; Liu, Xiao; Zhou, Yiqian; Hussain, Muzammal; Wan, Junting; Li, Minke; Li, Xue; Jin, Ruiliang; Tu, Zhengchao; Zhang, Jiancun
收藏  |  浏览/下载:41/0  |  提交时间:2016/12/16
Discovery of 2-(2-aminopyrimidin-5-yl)-4-morpholino-N-(pyridin-3-yl)quinazolin-7-amines as novel PI3K/mTOR inhibitors and anticancer agents 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 108, 页码: 644-654
作者:  Lu, Gui;  Liu, Quentin;  Long, Zi-Jie;  Tu, Zheng-Chao;  Peng, Wei
收藏  |  浏览/下载:15/0  |  提交时间:2018/12/13
Discovery of 2-(2-aminopyrimidin-5-yl)-4-morpholino-N-(pyridin-3-yl)quinazolin-7-amines as novel PI3K/mTOR inhibitors and anticancer agents 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 108, 页码: 644-654
Peng, Wei; Tu, Zheng-Chao; Long, Zi-Jie; Liu, Quentin; Lu, Gui
收藏  |  浏览/下载:19/0  |  提交时间:2016/12/16
Design, synthesis, and in vitro biological evaluation of novel 6-methyl-7-substituted-7-deaza purine nucleoside analogs as anti-influenza A agents 期刊论文
ANTIVIRAL RESEARCH, 2016, 卷号: 129, 页码: 13-20
作者:  Tu, Zhengchao;  Zhang, Jiancun;  Jin, Ruiliang;  Li, Xue;  Li, Minke
收藏  |  浏览/下载:29/0  |  提交时间:2018/12/13
Design, Synthesis, and Biological Evaluation of Pyrazolo[1,5-a]pyridine-3-carboxamides as Novel Antitubercular Agents 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 6, 期号: 7, 页码: 814-818
作者:  Ding, Ke;  Tang, Jian;  Wang, Bangxing;  Wu, Tian;  Wan, Junting
收藏  |  浏览/下载:29/0  |  提交时间:2018/12/13
Synthesis and Evaluation of Novel Erlotinib-NSAID Conjugates as More Comprehensive Anticancer Agents 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 6, 期号: 10, 页码: 1086-1090
Zhang, Yanmei; Tortorella, Micky D.; Liao, Jinxi; Qin, Xiaochu; Chen, Tingting; Luo, Jinfeng; Guan, Jiantong; Talley, John J.; Tu, Zhengchao
收藏  |  浏览/下载:33/0  |  提交时间:2016/12/16
Bacterial beta-Ketoacyl-Acyl Carrier Protein Synthase III (FabH) as a Target for Novel Antibacterial Agents Design 期刊论文
CURRENT MEDICINAL CHEMISTRY, 2015, 卷号: 22, 期号: 5, 页码: 651-667
Lu, X. Y.; Tang, J.; Zhang, Z.; Ding, K.
收藏  |  浏览/下载:12/0  |  提交时间:2016/12/16
The application of click chemistry in the synthesis of agents with anticancer activity 期刊论文
DRUG DESIGN DEVELOPMENT AND THERAPY, 2015, 卷号: 9, 页码: 1585-1599
Ma, Nan; Wang, Ying; Zhao, Bing-Xin; Ye, Wen-Cai; Jiang, Sheng
收藏  |  浏览/下载:31/0  |  提交时间:2016/12/16


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