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Design and synthesis of novel desfluoroquinolone-aminopyrimidine hybrids as potent anti-MRSA agents with low hERG activity 期刊论文
BIOORGANIC CHEMISTRY, 2020, 卷号: 103, 页码: 10
作者:  Song, Runzhe;  Wang, Yue;  Wang, Minghui;  Gao, Ruixuan;  Yang, Teng
收藏  |  浏览/下载:22/0  |  提交时间:2020/12/24
Aggregation-Induced Emission: Lighting Up hERG Potassium Channel 期刊论文
FRONTIERS IN CHEMISTRY, 2019, 卷号: 7
作者:  Zhang, Xiaomeng;  Liu, Tingting;  Li, Qi;  Li, Minyong;  Du, Lupei
收藏  |  浏览/下载:7/0  |  提交时间:2019/12/11
hERG optimizations of IMB1603, discovery of alternative benzothiazinones as new antitubercular agents 期刊论文
2019, 卷号: 179, 页码: 208-217
作者:  Lv Kai;  Wang Apeng;  Tao Zeyu;  Fu Lei;  Liu Hongtao
收藏  |  浏览/下载:12/0  |  提交时间:2020/01/03
康普瑞丁磷酸二钠对豚鼠心室肌细胞动作电位和hERG通道电流的影响 期刊论文
2019, 卷号: 34, 期号: 5, 页码: 1269-1273
作者:  管晓媛;  华潞;  孟红旭
收藏  |  浏览/下载:3/0  |  提交时间:2020/01/03
Design, synthesis and antimycobacterial activity of less lipophilic Q203 derivatives containing alkaline fused ring moieties 期刊论文
2019, 卷号: 27, 期号: 5, 页码: 813-821
作者:  Wang, Apeng;  Wang, Hongjian;  Geng, Yunhe;  Fu, Lei;  Gu, Jian
收藏  |  浏览/下载:22/0  |  提交时间:2020/01/03
Discovery of Potent Benzocycloalkane Derived Diapophytoene Desaturase Inhibitors with an Enhanced Safety Profile for the Treatment of MRSA, VISA, and LRSA Infections 期刊论文
ACS INFECTIOUS DISEASES, 2018, 卷号: 4, 期号: 3, 页码: 208-217
作者:  Li, Baoli;  Ni, Shuaishuai;  Chen, Feifei;  Mao, Fei;  Wei, Hanwen
收藏  |  浏览/下载:48/0  |  提交时间:2019/01/08
F463L increases the potential of dofetilide on human ether-a-go-go-related gene (hERG) channels 期刊论文
MICROSCOPY RESEARCH AND TECHNIQUE, 2018, 卷号: 81, 页码: 663-668
作者:  Cheng, Gong;  Wu, Jine;  Han, Wenqi;  Sun, Chaofeng
收藏  |  浏览/下载:3/0  |  提交时间:2019/11/19
A trafficking-deficient KCNQ1 mutation, T587M, causes a severe phenotype of long QT syndrome by interfering with intracellular hERG transport. 期刊论文
Journal of cardiology, 2018
作者:  Wu Jie;  Sakaguchi Tomoko;  Takenaka Kotoe;  Toyoda Futoshi;  Tsuji Keiko
收藏  |  浏览/下载:5/0  |  提交时间:2019/11/26
NS1643 enhances ionic currents in a G604S-WT hERG co-expression system associated with long QT syndrome 2 期刊论文
CLINICAL AND EXPERIMENTAL PHARMACOLOGY AND PHYSIOLOGY, 2017, 卷号: 44, 页码: 1125-1133
作者:  Huo, JianHua;  Guo, Xueyan;  Lu, Qun;  Qiang, Hua;  Liu, Ping
收藏  |  浏览/下载:3/0  |  提交时间:2019/11/26
Clenbuterol Attenuates hERG Channel by Promoting the Mature Channel Degradation 期刊论文
INTERNATIONAL JOURNAL OF TOXICOLOGY, 2017, 卷号: 36, 页码: 314-324
作者:  Luo, Ling;  Hu, Peijing;  Miao, Changqing;  Ma, Aiqun;  Wang, Tingzhong
收藏  |  浏览/下载:4/0  |  提交时间:2019/11/26


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