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浏览/检索结果: 共5条，第1-5条 帮助 已选(0)清除 条数/页：5101520253035404550556065707580859095100   排序方式：请选择作者升序作者降序题名升序题名降序发表日期升序发表日期降序提交时间升序提交时间降序 Discovery of QCA570 as an Exceptionally Potent and Efficacious Proteolysis Targeting Chimera (PROTAC) Degrader of the Bromodomain and Extra-Terminal (BET) Proteins Capable of Inducing Complete and Durable Tumor Regression 期刊论文 JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 15, 页码: 6685-6704 作者:  Qin, Chong;  Hu, Yang;  Zhou, Bing;  Fernandez-Salas, Ester;  Yang, Chao-Yie 收藏  |  浏览/下载：45/0  |  提交时间：2019/01/08 Structure-Based Discovery of CF53 as a Potent and Orally Bioavailable Bromodomain and Extra-Terminal (BET) Bromodomain Inhibitor 期刊论文 JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 14, 页码: 6110-6120 作者:  Zhao, Yujun;  Zhou, Bing;  Bai, Longchuan;  Liu, Liu;  Yang, Chao-Yie 收藏  |  浏览/下载：49/0  |  提交时间：2019/01/08 Structure-Based Discovery of 4-(6-Methoxy-2-methyl-4-(quinolin-4-yl)-9H-pyrimido[4,5-b]indol-7-yl)-3,5-dimethylisoxazole (CD161) as a Potent and Orally Bioavailable BET Bromodomain Inhibitor 期刊论文 JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 9, 页码: 3887-3901 作者:  Zhao, Yujun;  Bai, Longchuan;  Liu, Liu;  McEachern, Donna;  Stuckey, Jeanne A. 收藏  |  浏览/下载：27/0  |  提交时间：2019/01/08 Discovery of a new class of highly potent small-molecule degraders of BET bromodomain proteins 会议论文 作者:  Xu, Fuming;  Hu, Jiantao;  Zhou, Bing;  Chen, Zhuo;  Lin, Mei 收藏  |  浏览/下载：27/0  |  提交时间：2019/01/08 Design of the First-in-Class, Highly Potent Irreversible Inhibitor Targeting the Menin-MLL Protein-Protein Interaction 期刊论文 Angewandte Chemie International Edition 作者:  Shaomeng Wang;  Shilin Xu;  Angelo Aguilar;  Tianfeng Xu;  Ke Zheng 收藏  |  浏览/下载：1/0  |  提交时间：2019/03/26 epigenetics  irreversible  inhibitors  Menin-MLL  protein-protein  interaction  MLL  leukemia