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科研机构
北京大学 [6]
上海药物研究所 [4]
西安交通大学 [1]
大连化学物理研究所 [1]
暨南大学 [1]
复旦大学上海医学院 [1]
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期刊论文 [14]
其他 [1]
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2021 [1]
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Design, synthesis and pharmacological evaluation of tricyclic derivatives as selective RXFP4 agonists
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 110, 页码: 17
作者:
Lin, Lin
;
Lin, Guangyao
;
Zhou, Qingtong
;
Bathgate, Ross A. D.
;
Gong, Grace Qun
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/08/17
Synthesis
Structure-activity relationship
Relaxin family peptide receptor 4
Selective agonist
Molecular docking
High-throughput screening campaign identifies a small molecule agonist of the relaxin family peptide receptor 4
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9
作者:
Lin, Guang-yao
;
Lin, Lin
;
Cai, Xiao-qing
;
Dai, An-tao
;
Zhu, Yue
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2020/07/01
RXFP4
INSL5
high-throughput screening
agonist
JK1
Serelaxin, recombinant human relaxin-2, for heart failure patients A systematic review and meta-analysis
期刊论文
2018, 卷号: 97, 期号: 25
作者:
Yu, Ling[1]
;
Cao, Lijuan[1]
;
Sun, Jing[2]
;
Li, Zhongyi[3]
;
Yao, Fengzhen[1]
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/17
Transcriptional up-regulation of relaxin-3 by Nur77 attenuates -adrenergic agonist-induced apoptosis in cardiomyocytes
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2018, 卷号: Vol.293 No.36, 页码: 14001-14011
-
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  |  
浏览/下载:3/0
  |  
提交时间:2019/12/26
transcription
factor
nuclear
receptor
cardiomyocyte
apoptosis
relaxin
isoprenoid
Nur77
relaxin-3
beta-adrenergic
receptor
transcriptional
regulator
promoter
A validated UPLC-MS/MS method coupled with protein precipitation and ion exchange solid phase extraction for the quantitation of porcine relaxin B29 in dog plasma and its application to a pharmacokinetic study
期刊论文
ANALYTICAL AND BIOANALYTICAL CHEMISTRY, 2017, 卷号: 409, 期号: 28, 页码: 6559-6565
作者:
Su, Chong
;
Sun, Hui
;
Yang, Hong
;
Yin, Lei
;
Zhang, Jiwen
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2019/01/08
Ion exchange solid phase extraction
LC-MS/MS
Porcine relaxin
Ultrahigh performance liquid chromatography
Relaxin in paraventricular nucleus contributes to sympathetic overdrive and hypertension via PI3K-Akt pathway
期刊论文
NEUROPHARMACOLOGY, 2016, 卷号: 103, 期号: [db:dc_citation_issue], 页码: 247-256
作者:
Sun, Hai-Jian
;
Chen, Dan
;
Han, Ying
;
Zhou, Ye-Bo
;
Wang, Jue-Jin
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/02
Sympathetic
Hypertension
Relaxin
Vasopressin
Paraventricular nucleus
Bioactivity assay of porcine relaxin based on cAMP accumulation in THP-1 cells quantified by LC-MS/MS
期刊论文
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2015, 卷号: 111, 页码: 320-323
作者:
Ren, Xiaohong
;
Wang, Caifen
;
Wu, Li
;
Li, Haiyan
;
Chi, Liandi
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  |  
浏览/下载:24/0
  |  
提交时间:2019/01/08
Porcine relaxin
Bioactivity
cAMP
LC-MS/MS
ELISA
H2 relaxin expression and its effect on clinical outcomes in patients with chronic heart failure
期刊论文
INTERNATIONAL JOURNAL OF CLINICAL AND EXPERIMENTAL MEDICINE, 2015, 卷号: 8, 期号: 3
作者:
Xie, Juan
;
Chen, Yuan
;
Li, Liang
;
Zhang, Shan
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/19
Relaxin
chronic heart failure
cardiovascular events
The Formation and Stabilization of a Novel G-Quadruplex in the 5 '-Flanking Region of the Relaxin Gene
期刊论文
PLOS ONE, 2012, 卷号: 7, 期号: 2
作者:
Gao, Wei
;
Lin, Sen
;
Gu, Huiping
;
Xu, Ming
;
Cui, Xiaojie
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/06/20
Up-Regulating Relaxin Expression by G-Quadruplex Interactive Ligand to Achieve Antifibrotic Action
期刊论文
endocrinology, 2012
Gu, Hui-Ping
;
Lin, Sen
;
Xu, Ming
;
Yu, Hai-Yi
;
Du, Xiao-Jun
;
Zhang, You-Yi
;
Yuan, Gu
;
Gao, Wei
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2015/11/14
SPONTANEOUSLY HYPERTENSIVE-RATS
CARDIAC FIBROBLASTS
BERBERINE DERIVATIVES
CIRCULAR-DICHROISM
ANGIOTENSIN-II
HEART-FAILURE
HUMAN GENOME
FIBROSIS
GENE
CELLS
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