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中国医学科学院 北京... [6]
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大连化学物理研究所 [4]
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Discovery of a highly potent kinase inhibitor capable of overcoming multiple imatinib-resistant ABL mutants for chronic myeloid leukemia (CML)
期刊论文
EUROPEAN JOURNAL OF PHARMACOLOGY, 2021, 卷号: 897
作者:
Lu, Tingting
;
Cao, Jiangyan
;
Zou, Fengming
;
Li, Xixiang
;
Wang, Aoli
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2021/04/26
BCR-ABL
ABL mutants
Chronic myeloid leukemia
Kinase inhibitor
Imatinib resistance
Adverse events associated with nilotinib in chronic myeloid leukemia: mechanisms and management strategies
期刊论文
EXPERT REVIEW OF CLINICAL PHARMACOLOGY, 2021
作者:
Wang, Zeng
;
Jiang, Liyu
;
Yan, Hao
;
Xu, Zhifei
;
Luo, Peihua
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2021/04/26
Adverse events
chronic myeloid leukemia
management
mechanisms
molecular target
nilotinib
An ultra-long circulating nanoparticle for reviving a highly selective BCR-ABL inhibitor in long-term effective and safe treatment of chronic myeloid leukemia
期刊论文
NANOMEDICINE-NANOTECHNOLOGY BIOLOGY AND MEDICINE, 2020, 卷号: 29
作者:
Fu, Liyi
;
Zou, Fengming
;
Liu, Qingwang
;
Wang, Beilei
;
Wang, Junqing
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2020/11/30
Chronic myeloid leukemia
BCR-ABL
Long-circulating nanoparticle
Drug delivery
Nilotinib combined with multi-agent chemotherapy in newly diagnosed Philadelphia chromosome-positive acute lymphoblastic leukemia: a single-center prospective study with long-term follow-up
期刊论文
2019, 卷号: 98, 期号: 3, 页码: 633-645
作者:
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2020/01/03
HRFS
MRFS
Nilotinib
OS
Ph plus ALL
UGT1A10 Is a High Activity and Important Extrahepatic Enzyme: Why Has Its Role in Intestinal Glucuronidation Been Frequently Underestimated?
期刊论文
MOLECULAR PHARMACEUTICS, 2017, 卷号: 14, 期号: 9, 页码: 2875-2883
作者:
Yang, Ling
;
Ge, Guang-Bo
;
Jarvinen, Erkka
;
Troberg, Johanna
;
Finel, Moshe
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2017/12/20
UDP-glucuronosyltransferase
recombinant UGT1A10
intestine microsomes
intestinal glucuronidation
estradiol
estrone
morphine
SN-38
AMC
NCHN
bavachinin
UGT1A10 Is a High Activity and Important Extrahepatic Enzyme: Why Has Its Role in Intestinal Glucuronidation Been Frequently Underestimated?
期刊论文
MOLECULAR PHARMACEUTICS, 2017, 卷号: 14, 期号: 9, 页码: 2875-2883
作者:
Troberg, Johanna
;
Jarvinen, Erkka
;
Ge, Guang-Bo
;
Yang, Ling
;
Finel, Moshe
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2017/12/20
UDP-glucuronosyltransferase
recombinant UGT1A10
intestine microsomes
intestinal glucuronidation
estradiol
estrone
morphine
SN-38
AMC
NCHN
bavachinin
AKT is critically involved in the antagonism of BRAF inhibitor sorafenib against dabrafenib in colorectal cancer cells harboring both wild-type and mutant (V600E) BRAF genes
期刊论文
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2017, 卷号: 489, 期号: 1, 页码: 14-20
作者:
Wang, Hongbin
;
Quan, Haitian
;
Lou, Liguang
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/01/08
Antagonism
AKT
BRAF
Dabrafenib
Sorafenib
RUXOLITINIB/NILOTINIB COTREATMENT BETTER INHIBITS LEUKEMIA-PROPAGATING CELLS IN PHILADELPHIA CHROMOSOME-POSITIVE ALL
期刊论文
HAEMATOLOGICA, 2017
Kong, Y.
;
Wu, Y.L.
;
Song, Y.
;
Shi, M.M.
;
Cao, X.N.
;
Zhao, H.Y.
;
Qin, Y.Z.
;
Lai, Y.Y.
;
Jiang, H.
;
Jiang, Q.
;
Huang, X.J.
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
RUXOLITINIB/NILOTINIB COTREATMENT BETTER INHIBITS LEUKEMIA-PROPAGATING CELLS IN PHILADELPHIA CHROMOSOME-POSITIVE ALL
其他
2017-01-01
Kong, Y.
;
Wu, Y.L.
;
Song, Y.
;
Shi, M.M.
;
Cao, X.N.
;
Zhao, H.Y.
;
Qin, Y.Z.
;
Lai, Y.Y.
;
Jiang, H.
;
Jiang, Q.
;
Huang, X.J.
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
Ruxolitinib/nilotinib cotreatment inhibits leukemia-propagating cells in Philadelphia chromosome-positive ALL
期刊论文
JOURNAL OF TRANSLATIONAL MEDICINE, 2017
Kong, Yuan
;
Wu, Yi-Lin
;
Song, Yang
;
Shi, Min-Min
;
Cao, Xie-Na
;
Zhao, Hong-Yan
;
Qin, Ya-Zhen
;
Lai, Yue-Yun
;
Jiang, Hao
;
Jiang, Qian
;
Huang, Xiao-Jun
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2017/12/03
Acute lymphoblastic leukemia
Ph-chromosome
Leukemia-propagating cells
Nilotinib
Ruxolitinib
ACUTE MYELOID-LEUKEMIA
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